JP2009051812A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2009051812A5 JP2009051812A5 JP2008128074A JP2008128074A JP2009051812A5 JP 2009051812 A5 JP2009051812 A5 JP 2009051812A5 JP 2008128074 A JP2008128074 A JP 2008128074A JP 2008128074 A JP2008128074 A JP 2008128074A JP 2009051812 A5 JP2009051812 A5 JP 2009051812A5
- Authority
- JP
- Japan
- Prior art keywords
- xrpd
- powder
- formula
- hydroxydiphenylmethyl
- oxobutyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Description
式（Ｉ）の得られたケト：４−｛［４−（４−ヒドロキシジフェニルメチル）−１−ピペリジニル］−１−オキソブチル｝−α，α−ジメチルベンゼン酢酸は、ＸＲＰＤ（ここで、最も強い回折ピークが、２θにおいて５．７；８．８；１０．３；１１．５；１６．１；１７．３；１８．１；１９．４；２０．０；２２．８±０．２°である）を有する結晶構造を有する。前記結晶形態の式（Ｉ）のケトンは、新規化合物であり、本発明の目的物である。
Claims (1)
- 最も強い回折ピークが、２θにおいて５．７；８．８；１０．３；１１．５；１６．１；１７．３；１８．１；１９．４；２０．０；２２．８±０．２°であるＸＲＰＤを有する結晶形態にある、４−｛［４−（４−ヒドロキシジフェニルメチル）−１−ピペリジニル］−１−オキソブチル｝−α，α−ジメチルベンゼン酢酸。
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI2007A000987 | 2007-05-16 | ||
| IT000987A ITMI20070987A1 (it) | 2007-05-16 | 2007-05-16 | Procedimento per la preparazione di composti chetonici |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2009051812A JP2009051812A (ja) | 2009-03-12 |
| JP2009051812A6 JP2009051812A6 (ja) | 2009-06-18 |
| JP2009051812A5 true JP2009051812A5 (ja) | 2011-05-26 |
| JP5342169B2 JP5342169B2 (ja) | 2013-11-13 |
Family
ID=39666057
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008128074A Expired - Fee Related JP5342169B2 (ja) | 2007-05-16 | 2008-05-15 | ケト化合物の製法 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US8236961B2 (ja) |
| EP (1) | EP1992615B1 (ja) |
| JP (1) | JP5342169B2 (ja) |
| AT (1) | ATE554068T1 (ja) |
| AU (1) | AU2008202097A1 (ja) |
| BR (1) | BRPI0801557A2 (ja) |
| CA (1) | CA2631376A1 (ja) |
| IL (1) | IL191460A0 (ja) |
| IT (1) | ITMI20070987A1 (ja) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2403130B1 (es) * | 2010-06-15 | 2014-09-29 | Chemelectiva S.R.L. | Forma polimórfica de clorhidrato de fexofenadina, compuestos intermedios y procedimiento para su preparación |
| ITMI20131652A1 (it) | 2013-10-07 | 2015-04-08 | Dipharma Francis Srl | Procedimento per la purificazione di derivati dell'acido 2-fenil-2-metil-propanoico |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4254130A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
| US4254129A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
| MX9302076A (es) | 1992-04-10 | 1994-03-31 | Merrell Dow Pharma | Proceso novedoso para preparar derivados de piperidina. |
| US6153754A (en) | 1995-12-21 | 2000-11-28 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
| US6201124B1 (en) | 1995-12-21 | 2001-03-13 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
| ITRM20010260A1 (it) * | 2001-05-17 | 2002-11-18 | Dinamite Dipharma S P A In For | Processo per la preparazione della fexofenadina o acido 4 1-idrossi-4-4- (idrossidifenilmetil)-1-piperidinil|-butil|-alfa,alfa-dimetilbenz |
| JP2005537218A (ja) * | 2001-11-08 | 2005-12-08 | テバ ファーマシューティカル インダストリーズ リミティド | フェキソフェナジン塩基の多形体 |
| GB0319935D0 (en) * | 2003-08-26 | 2003-09-24 | Cipla Ltd | Polymorphs |
| ITMI20041143A1 (it) * | 2004-06-08 | 2004-09-08 | Dipharma Spa | Polimorfi di fexofenadina e procedimento per la loro preparazione |
| EP1616861A3 (en) | 2004-06-15 | 2006-02-08 | Dipharma S.p.A. | A process for the preparation of keto compounds |
| JP2008514641A (ja) * | 2004-09-28 | 2008-05-08 | テバ ファーマシューティカル インダストリーズ リミティド | 結晶形フェキソフェナジン、およびその調製方法 |
-
2007
- 2007-05-16 IT IT000987A patent/ITMI20070987A1/it unknown
-
2008
- 2008-05-12 AU AU2008202097A patent/AU2008202097A1/en not_active Abandoned
- 2008-05-15 BR BRPI0801557-0A patent/BRPI0801557A2/pt not_active IP Right Cessation
- 2008-05-15 IL IL191460A patent/IL191460A0/en unknown
- 2008-05-15 US US12/121,294 patent/US8236961B2/en not_active Expired - Fee Related
- 2008-05-15 JP JP2008128074A patent/JP5342169B2/ja not_active Expired - Fee Related
- 2008-05-15 AT AT08156214T patent/ATE554068T1/de active
- 2008-05-15 EP EP08156214A patent/EP1992615B1/en not_active Not-in-force
- 2008-05-15 CA CA002631376A patent/CA2631376A1/en not_active Abandoned
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| WO2009028553A1 (ja) | チタン酸化合物及びその製造方法並びに該チタン酸化合物を含む電極活物質、電極活物質を用いてなる蓄電デバイス | |
| JP2009520765A5 (ja) | ||
| EP1667971B1 (en) | Fexofenadine polymorphs and processes of preparing the same | |
| JP2010533203A5 (ja) | ||
| JP2010533191A5 (ja) | ||
| JP2010521514A5 (ja) | ||
| RU2011107128A (ru) | Новая молекулярно-ситовая композиция емм-12, способы ее получения и применения | |
| BRPI0617506A2 (pt) | derivados de Ácido dicarboxÍlico e seu uso | |
| JP2009051812A5 (ja) | ||
| JP2009521414A5 (ja) | ||
| JP2010265452A5 (ja) | 顔料の製造方法 | |
| JP2010511649A5 (ja) | ||
| Khandavilli et al. | High solubility crystalline hydrates of Na and K furosemide salts | |
| JP2012533550A5 (ja) | ||
| JP2021514967A5 (ja) | ||
| JP2013503145A5 (ja) | ||
| JP2009541344A5 (ja) | ||
| BG108435A (en) | Novel crystalline forms of 4-[4-[4-(hydroxydiphenyl methyl)-1-piperidinyl]-1-hydroxybutyl]-alpha, alpha-dimethylbenzene acetic acid and its hydrochloride | |
| JPWO2020037164A5 (ja) | ||
| RU2008105987A (ru) | Новые пиперидиновые производные | |
| US20050277775A1 (en) | Process for the preparation of keto compounds | |
| JP2016503041A5 (ja) | ||
| WO2007146768A3 (en) | Compounds for the treatment of metabolic disorders | |
| JP7252978B2 (ja) | ２－（１－（ｔｅｒｔ－ブトキシカルボニル）ピペリジン－４－イル）安息香酸を調製するためのプロセス | |
| EP1992615B1 (en) | A process for the preparation of keto compounds |