JP2008523126A5 - - Google Patents

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Publication number
JP2008523126A5
JP2008523126A5 JP2007545891A JP2007545891A JP2008523126A5 JP 2008523126 A5 JP2008523126 A5 JP 2008523126A5 JP 2007545891 A JP2007545891 A JP 2007545891A JP 2007545891 A JP2007545891 A JP 2007545891A JP 2008523126 A5 JP2008523126 A5 JP 2008523126A5
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JP
Japan
Prior art keywords
lower alkyl
halogen
hydrogen
substituted
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2007545891A
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English (en)
Japanese (ja)
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JP4709849B2 (ja
JP2008523126A (ja
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Application filed filed Critical
Priority claimed from PCT/EP2005/012994 external-priority patent/WO2006063709A1/en
Publication of JP2008523126A publication Critical patent/JP2008523126A/ja
Publication of JP2008523126A5 publication Critical patent/JP2008523126A5/ja
Application granted granted Critical
Publication of JP4709849B2 publication Critical patent/JP4709849B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2007545891A 2004-12-15 2005-12-05 アルツハイマー病治療のためのグリシントランスポーターｉ（ｇｌｙｔ−１）インヒビターとしての二環式及び三環式置換フェニルメタノン類 Expired - Fee Related JP4709849B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP04106597.0 2004-12-15
EP04106597 2004-12-15
PCT/EP2005/012994 WO2006063709A1 (en) 2004-12-15 2005-12-05 Bi- and tricyclic substituted phenyl methanones as glycine transporter i (glyt-1) inhibitors for the treatment of alzheimer’s disease

Publications (3)

Publication Number Publication Date
JP2008523126A JP2008523126A (ja) 2008-07-03
JP2008523126A5 true JP2008523126A5 (https=) 2009-02-19
JP4709849B2 JP4709849B2 (ja) 2011-06-29

Family

ID=35841863

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007545891A Expired - Fee Related JP4709849B2 (ja) 2004-12-15 2005-12-05 アルツハイマー病治療のためのグリシントランスポーターｉ（ｇｌｙｔ−１）インヒビターとしての二環式及び三環式置換フェニルメタノン類

Country Status (20)

Country Link
US (1) US7375226B2 (https=)
EP (1) EP1828200B1 (https=)
JP (1) JP4709849B2 (https=)
KR (1) KR100883003B1 (https=)
CN (1) CN100586951C (https=)
AR (1) AR052156A1 (https=)
AT (1) ATE457989T1 (https=)
AU (1) AU2005315914B2 (https=)
BR (1) BRPI0519054A2 (https=)
CA (1) CA2590316A1 (https=)
DE (1) DE602005019465D1 (https=)
ES (1) ES2338139T3 (https=)
IL (1) IL183592A0 (https=)
MX (1) MX2007006896A (https=)
NO (1) NO20072833L (https=)
NZ (1) NZ555476A (https=)
RU (1) RU2007121768A (https=)
TW (1) TWI299041B (https=)
WO (1) WO2006063709A1 (https=)
ZA (1) ZA200705044B (https=)

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US9365512B2 (en) 2012-02-13 2016-06-14 AbbVie Deutschland GmbH & Co. KG Isoindoline derivatives, pharmaceutical compositions containing them, and their use in therapy
CN104203951B (zh) * 2012-03-16 2016-11-02 生命医药公司 肝x受体调节剂
WO2013138568A1 (en) * 2012-03-16 2013-09-19 Vitae Pharmaceuticals, Inc. Liver x reception modulators
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US9650334B2 (en) 2013-03-15 2017-05-16 Abbvie Inc. Pyrrolidine derivatives, pharmaceutical compositions containing them, and their use in therapy
US9708322B2 (en) 2013-03-15 2017-07-18 Intra-Cellular Therapies, Inc. Substituted pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalines for inhibiting serotonin reuptake transporter activity
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