JP2008517936A5 - - Google Patents
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- Publication number
- JP2008517936A5 JP2008517936A5 JP2007538127A JP2007538127A JP2008517936A5 JP 2008517936 A5 JP2008517936 A5 JP 2008517936A5 JP 2007538127 A JP2007538127 A JP 2007538127A JP 2007538127 A JP2007538127 A JP 2007538127A JP 2008517936 A5 JP2008517936 A5 JP 2008517936A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- unsubstituted
- substituted
- alkoxy
- alkenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000000217 alkyl group Chemical group 0.000 claims 23
- 125000003342 alkenyl group Chemical group 0.000 claims 13
- 125000003545 alkoxy group Chemical group 0.000 claims 13
- 125000000304 alkynyl group Chemical group 0.000 claims 12
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 12
- -1 benzyloxy, phenoxy Chemical group 0.000 claims 11
- 125000004076 pyridyl group Chemical group 0.000 claims 10
- 150000001875 compounds Chemical class 0.000 claims 7
- 125000002541 furyl group Chemical group 0.000 claims 6
- DLFVBJFMPXGRIB-UHFFFAOYSA-N Acetamide Chemical compound CC(N)=O DLFVBJFMPXGRIB-UHFFFAOYSA-N 0.000 claims 4
- ZHNUHDYFZUAESO-UHFFFAOYSA-N Formamide Chemical compound NC=O ZHNUHDYFZUAESO-UHFFFAOYSA-N 0.000 claims 4
- 125000002047 benzodioxolyl group Chemical group O1OC(C2=C1C=CC=C2)* 0.000 claims 4
- 125000001164 benzothiazolyl group Chemical group S1C(=NC2=C1C=CC=C2)* 0.000 claims 4
- 125000004541 benzoxazolyl group Chemical group O1C(=NC2=C1C=CC=C2)* 0.000 claims 4
- 125000005102 carbonylalkoxy group Chemical group 0.000 claims 4
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 claims 4
- 125000004438 haloalkoxy group Chemical group 0.000 claims 4
- 125000001188 haloalkyl group Chemical group 0.000 claims 4
- 125000001624 naphthyl group Chemical group 0.000 claims 4
- 125000002971 oxazolyl group Chemical group 0.000 claims 4
- 125000000951 phenoxy group Chemical group [H]C1=C([H])C([H])=C(O*)C([H])=C1[H] 0.000 claims 4
- 125000000714 pyrimidinyl group Chemical group 0.000 claims 4
- 125000001424 substituent group Chemical group 0.000 claims 4
- 125000000335 thiazolyl group Chemical group 0.000 claims 4
- 125000001544 thienyl group Chemical group 0.000 claims 4
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 3
- 125000004001 thioalkyl group Chemical group 0.000 claims 3
- BOIUBJYPHIFHEJ-UHFFFAOYSA-N 2,4-difluoro-1,3-benzodioxole Chemical compound C1=CC(F)=C2OC(F)OC2=C1 BOIUBJYPHIFHEJ-UHFFFAOYSA-N 0.000 claims 2
- 125000005036 alkoxyphenyl group Chemical group 0.000 claims 2
- 150000005215 alkyl ethers Chemical group 0.000 claims 2
- 125000005189 alkyl hydroxy group Chemical group 0.000 claims 2
- 125000000051 benzyloxy group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])O* 0.000 claims 2
- 125000002619 bicyclic group Chemical group 0.000 claims 2
- 229910052801 chlorine Inorganic materials 0.000 claims 2
- 125000001309 chloro group Chemical group Cl* 0.000 claims 2
- RTZKZFJDLAIYFH-UHFFFAOYSA-N ether Substances CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 claims 2
- 229910052731 fluorine Inorganic materials 0.000 claims 2
- 230000002538 fungal effect Effects 0.000 claims 2
- 230000000855 fungicidal effect Effects 0.000 claims 2
- 229910052736 halogen Inorganic materials 0.000 claims 2
- 125000005843 halogen group Chemical group 0.000 claims 2
- 150000002367 halogens Chemical class 0.000 claims 2
- 125000005059 halophenyl group Chemical group 0.000 claims 2
- 125000005842 heteroatom Chemical group 0.000 claims 2
- 125000000623 heterocyclic group Chemical group 0.000 claims 2
- 229910052739 hydrogen Inorganic materials 0.000 claims 2
- 230000009545 invasion Effects 0.000 claims 2
- 229910052740 iodine Inorganic materials 0.000 claims 2
- 125000005647 linker group Chemical group 0.000 claims 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 2
- 125000002950 monocyclic group Chemical group 0.000 claims 2
- 125000002757 morpholinyl group Chemical group 0.000 claims 2
- 125000003373 pyrazinyl group Chemical group 0.000 claims 2
- 125000000168 pyrrolyl group Chemical group 0.000 claims 2
- 241000233866 Fungi Species 0.000 claims 1
- 206010061217 Infestation Diseases 0.000 claims 1
- 229910052794 bromium Inorganic materials 0.000 claims 1
- 229910052799 carbon Inorganic materials 0.000 claims 1
- 239000012876 carrier material Substances 0.000 claims 1
- 125000004093 cyano group Chemical group *C#N 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 239000002689 soil Substances 0.000 claims 1
- 238000005507 spraying Methods 0.000 claims 1
- 125000004963 sulfonylalkyl group Chemical group 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US62157704P | 2004-10-21 | 2004-10-21 | |
| US60/621,577 | 2004-10-21 | ||
| PCT/US2005/038145 WO2006047397A1 (en) | 2004-10-21 | 2005-10-21 | Thieno-pyrimidine compounds having fungicidal activity |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012104644A Division JP5572664B2 (ja) | 2004-10-21 | 2012-05-01 | 殺真菌活性を有するチエノ−ピリミジン化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2008517936A JP2008517936A (ja) | 2008-05-29 |
| JP2008517936A5 true JP2008517936A5 (enExample) | 2009-01-22 |
| JP5122293B2 JP5122293B2 (ja) | 2013-01-16 |
Family
ID=35722379
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007538127A Expired - Fee Related JP5122293B2 (ja) | 2004-10-21 | 2005-10-21 | 殺真菌活性を有するチエノ−ピリミジン化合物 |
| JP2012104644A Expired - Fee Related JP5572664B2 (ja) | 2004-10-21 | 2012-05-01 | 殺真菌活性を有するチエノ−ピリミジン化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012104644A Expired - Fee Related JP5572664B2 (ja) | 2004-10-21 | 2012-05-01 | 殺真菌活性を有するチエノ−ピリミジン化合物 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US8008487B2 (enExample) |
| EP (1) | EP1802632B1 (enExample) |
| JP (2) | JP5122293B2 (enExample) |
| KR (3) | KR101386797B1 (enExample) |
| CN (1) | CN101084224B (enExample) |
| AT (1) | ATE516291T1 (enExample) |
| BR (1) | BRPI0516242B1 (enExample) |
| WO (1) | WO2006047397A1 (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101084224B (zh) * | 2004-10-21 | 2013-12-04 | 美国陶氏益农公司 | 具有杀真菌活性的噻吩并-嘧啶化合物 |
| EP2078721B1 (en) * | 2005-10-21 | 2014-01-22 | Dow AgroSciences LLC | Thieno-pyrimidine compounds having fungicidal activity |
| AP2008004687A0 (en) * | 2006-05-22 | 2008-12-31 | Basf Se | Insecticidal methods using 4-amino-5-chloro-thieno(2,3-d)-pyrimidine compounds |
| US8318384B2 (en) | 2007-04-30 | 2012-11-27 | The Governors Of The University Of Alberta | Anode catalyst and methods of making and using the same |
| AU2009291783A1 (en) * | 2008-09-10 | 2010-03-18 | Alcon Research, Ltd | Aminopyrimidine inhibitors of histamine receptors for the treatment of disease |
| TWI485138B (zh) * | 2009-07-16 | 2015-05-21 | Sds Biotech Corp | 4- (3-butynyl) aminopyrimidine derivatives as a pest control agent for agricultural and horticulture |
| BR112012002164B1 (pt) | 2009-07-30 | 2021-04-20 | Merial, Inc | compostos inseticidas de 4-amino-tieno[2,3-d]-pirimidina e métodos para seu uso |
| JP5902100B2 (ja) * | 2011-01-14 | 2016-04-13 | 株式会社エス・ディー・エス バイオテック | ４−（３−ブチニル）アミノピリミジン誘導体を含む農園芸用有害生物防除剤組成物 |
| BR112013033568B1 (pt) * | 2011-06-27 | 2020-11-24 | Merial, Inc | Compostos eter amidopiridil e composiqoes, e seu uso contra parasitas |
| WO2013012918A1 (en) | 2011-07-19 | 2013-01-24 | Infinity Pharmaceuticals Inc. | Heterocyclic compounds and uses thereof |
| AR090037A1 (es) | 2011-11-15 | 2014-10-15 | Xention Ltd | Derivados de tieno y/o furo-pirimidinas y piridinas inhibidores de los canales de potasio |
| CN105315296B (zh) * | 2014-07-04 | 2018-04-03 | 沈阳中化农药化工研发有限公司 | 取代芳氧吡啶类化合物及其用途 |
| CN104725398B (zh) * | 2015-01-29 | 2017-01-18 | 杨威 | 一种jak/stat3磷酸化抑制剂及其制备方法与用途 |
| CN109776427B (zh) * | 2017-11-13 | 2022-08-23 | 沈阳中化农药化工研发有限公司 | 嘧啶双胺类化合物及其用途 |
| WO2020180768A1 (en) * | 2019-03-01 | 2020-09-10 | Revolution Medicines, Inc. | Bicyclic heteroaryl compounds and uses thereof |
| CN115626893B (zh) * | 2022-10-10 | 2024-04-02 | 山西永津集团有限公司 | 一种2-羟基-5-羟甲基吡啶的合成方法 |
Family Cites Families (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1570494A (en) | 1975-11-28 | 1980-07-02 | Ici Ltd | Thienopyrimidine derivatives and their use as pesticides |
| ZA782648B (en) * | 1977-05-23 | 1979-06-27 | Ici Australia Ltd | The prevention,control or eradication of infestations of ixodid ticks |
| GB2043061B (en) | 1979-03-05 | 1983-05-11 | Ici Ltd | Thienopyrimidine and quinazoline derivatives |
| JPS5942387A (ja) * | 1982-07-21 | 1984-03-08 | Sankyo Co Ltd | チエノピリミジン誘導体および殺虫、殺ダニ剤 |
| EP0193885B1 (de) | 1985-03-02 | 1989-06-14 | BASF Aktiengesellschaft | Thiophenderivate |
| JPS6267A (ja) * | 1985-03-14 | 1987-01-06 | Sankyo Co Ltd | フエノキシアルキルアミン誘導体、その製法および殺虫殺ダニ剤 |
| US5141941A (en) * | 1988-11-21 | 1992-08-25 | Ube Industries, Ltd. | Aralkylamine derivatives, and fungicides containing the same |
| US5124333A (en) * | 1989-08-02 | 1992-06-23 | Ube Industries, Ltd. | Aminopyrimidine derivatives and harmful organisms preventive agent |
| JPH0363265A (ja) * | 1989-08-02 | 1991-03-19 | Ube Ind Ltd | アルキルアミノピリミジン誘導体、その製造法及び殺虫・殺ダニ・殺線虫剤 |
| JPH075569B2 (ja) | 1989-08-02 | 1995-01-25 | 宇部興産株式会社 | アラルキルアミン誘導体、その製法及び殺菌、殺虫剤 |
| EP0424125A3 (en) | 1989-10-18 | 1991-10-09 | Ube Industries, Ltd. | Aralkylamine derivatives, preparation method thereof and fungicides containing the same |
| DE4008726A1 (de) * | 1990-03-19 | 1991-09-26 | Basf Ag | Thieno(2,3-d)pyrimidinderivate |
| US5137879A (en) * | 1990-03-30 | 1992-08-11 | Dowelanco | Furopyrimidin-4-imine derivatives |
| AU651337B2 (en) * | 1990-03-30 | 1994-07-21 | Dowelanco | Thienopyrimidine derivatives |
| JP2730019B2 (ja) * | 1990-04-06 | 1998-03-25 | 宇部興産株式会社 | アラルキルアミン誘導体，その製造法及び殺菌剤 |
| JP2762430B2 (ja) | 1991-01-18 | 1998-06-04 | 宇部興産株式会社 | アラルキルアミノピリミジン類の製法 |
| EP0519211A1 (de) * | 1991-05-17 | 1992-12-23 | Hoechst Schering AgrEvo GmbH | Substituierte 4-Aminopyrimidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel |
| JP3063266B2 (ja) | 1991-08-30 | 2000-07-12 | セイコーエプソン株式会社 | 液晶パネル及びその製造方法 |
| JPH0710712A (ja) | 1993-06-25 | 1995-01-13 | Ube Ind Ltd | 花卉園芸用殺菌剤 |
| US5679683A (en) * | 1994-01-25 | 1997-10-21 | Warner-Lambert Company | Tricyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family |
| GB9424676D0 (en) * | 1994-12-07 | 1995-02-01 | Sandoz Ltd | Organic compounds |
| US6232320B1 (en) * | 1998-06-04 | 2001-05-15 | Abbott Laboratories | Cell adhesion-inhibiting antiinflammatory compounds |
| IL139811A0 (en) * | 1998-06-04 | 2002-02-10 | Abbott Lab | Cell adhesion-inhibiting antinflammatory compounds |
| CA2390948A1 (en) * | 1999-06-03 | 2000-12-14 | Abbott Laboratories | Cell adhesion-inhibiting antiinflammatory compounds |
| WO2003022214A2 (en) * | 2001-09-06 | 2003-03-20 | Millennium Pharmaceuticals, Inc. | Piperazine and homopiperazine compounds |
| US20050009845A1 (en) | 2001-12-19 | 2005-01-13 | Caferro Thomas R. | Thienopyrimidine compounds as protein tyrosine kinase inhibitors |
| WO2004092123A2 (en) * | 2003-04-10 | 2004-10-28 | Microbia, Inc. | Inhibitors of fungal invasion |
| KR101186678B1 (ko) * | 2003-06-11 | 2012-09-27 | 젠션 리미티드 | 포타슘 채널 억제제로서의 티에노피리미딘 유도체 |
| GB0315950D0 (en) * | 2003-06-11 | 2003-08-13 | Xention Discovery Ltd | Compounds |
| CN101084224B (zh) * | 2004-10-21 | 2013-12-04 | 美国陶氏益农公司 | 具有杀真菌活性的噻吩并-嘧啶化合物 |
-
2005
- 2005-10-21 CN CN2005800440617A patent/CN101084224B/zh not_active Expired - Fee Related
- 2005-10-21 US US11/256,117 patent/US8008487B2/en not_active Expired - Fee Related
- 2005-10-21 KR KR1020077011335A patent/KR101386797B1/ko not_active Expired - Fee Related
- 2005-10-21 KR KR1020147016709A patent/KR20140094626A/ko not_active Abandoned
- 2005-10-21 BR BRPI0516242-4A patent/BRPI0516242B1/pt not_active IP Right Cessation
- 2005-10-21 AT AT05812301T patent/ATE516291T1/de not_active IP Right Cessation
- 2005-10-21 JP JP2007538127A patent/JP5122293B2/ja not_active Expired - Fee Related
- 2005-10-21 WO PCT/US2005/038145 patent/WO2006047397A1/en not_active Ceased
- 2005-10-21 KR KR1020137034724A patent/KR20140008471A/ko not_active Withdrawn
- 2005-10-21 EP EP05812301A patent/EP1802632B1/en not_active Expired - Lifetime
-
2012
- 2012-05-01 JP JP2012104644A patent/JP5572664B2/ja not_active Expired - Fee Related
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