JP2008501649A5 - - Google Patents
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- Publication number
- JP2008501649A5 JP2008501649A5 JP2007513783A JP2007513783A JP2008501649A5 JP 2008501649 A5 JP2008501649 A5 JP 2008501649A5 JP 2007513783 A JP2007513783 A JP 2007513783A JP 2007513783 A JP2007513783 A JP 2007513783A JP 2008501649 A5 JP2008501649 A5 JP 2008501649A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- compound
- formula
- lower alkyl
- alkyl group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 description 3
- 125000000217 alkyl group Chemical group 0.000 description 2
- 125000003884 phenylalkyl group Chemical group 0.000 description 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 description 1
- 125000003545 alkoxy group Chemical group 0.000 description 1
- 125000005843 halogen group Chemical group 0.000 description 1
- 229910052739 hydrogen Inorganic materials 0.000 description 1
- 239000001257 hydrogen Substances 0.000 description 1
- 125000002768 hydroxyalkyl group Chemical group 0.000 description 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04102460 | 2004-06-02 | ||
| PCT/EP2005/005594 WO2005117865A1 (en) | 2004-06-02 | 2005-05-24 | Naphthaline derivatives useful as histamine-3-receptor ligands |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2008501649A JP2008501649A (ja) | 2008-01-24 |
| JP2008501649A5 true JP2008501649A5 (enExample) | 2010-09-24 |
| JP4594386B2 JP4594386B2 (ja) | 2010-12-08 |
Family
ID=34982058
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007513783A Expired - Fee Related JP4594386B2 (ja) | 2004-06-02 | 2005-05-24 | ヒスタミン３受容体のリガンドとして有用なナフタレン誘導体 |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US7259158B2 (enExample) |
| EP (1) | EP1755593B1 (enExample) |
| JP (1) | JP4594386B2 (enExample) |
| KR (1) | KR100854212B1 (enExample) |
| CN (1) | CN1960727B (enExample) |
| AR (1) | AR049433A1 (enExample) |
| AT (1) | ATE383857T1 (enExample) |
| AU (1) | AU2005249196B2 (enExample) |
| BR (1) | BRPI0511778A (enExample) |
| CA (1) | CA2566526C (enExample) |
| DE (1) | DE602005004404T2 (enExample) |
| DK (1) | DK1755593T3 (enExample) |
| ES (1) | ES2299074T3 (enExample) |
| IL (1) | IL179370A (enExample) |
| MX (1) | MXPA06014017A (enExample) |
| MY (1) | MY139704A (enExample) |
| NO (1) | NO20065733L (enExample) |
| NZ (1) | NZ550764A (enExample) |
| PL (1) | PL1755593T3 (enExample) |
| PT (1) | PT1755593E (enExample) |
| RU (1) | RU2387638C2 (enExample) |
| TW (1) | TWI299992B (enExample) |
| WO (1) | WO2005117865A1 (enExample) |
| ZA (1) | ZA200609678B (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1988143A4 (en) | 2006-02-20 | 2009-11-25 | Konica Minolta Holdings Inc | ORGANIC ELECTROLUMINESCENT ELEMENT, WHITE LIGHT EMITTING ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE |
| WO2008083124A1 (en) | 2006-12-28 | 2008-07-10 | Rigel Pharmaceuticals, Inc. | N-substituted-heterocycloalkyloxybenzamide compounds and methods of use |
| CN101679237A (zh) | 2007-05-03 | 2010-03-24 | 赛福伦公司 | 制备(r)-2-甲基吡咯烷和(s)-2-甲基吡咯烷及其酒石酸盐的方法 |
| CA2705947C (en) | 2007-11-16 | 2016-08-09 | Rigel Pharmaceuticals, Inc. | Carboxamide, sulfonamide and amine compounds for metabolic disorders |
| JP5650540B2 (ja) * | 2007-12-12 | 2015-01-07 | ライジェル ファーマシューティカルズ， インコーポレイテッド | 代謝障害のためのカルボキサミド、スルホンアミド、およびアミン化合物 |
| NZ588652A (en) | 2008-04-23 | 2012-09-28 | Rigel Pharmaceuticals Inc | Carboxamide compounds for the treatment of metabolic disorders |
| TW201202251A (en) | 2010-05-11 | 2012-01-16 | Sanofi Aventis | Substituted N-heteroaryl spirolactam bipyrrolidines, preparation and therapeutic use thereof |
| JP5784110B2 (ja) | 2010-05-11 | 2015-09-24 | サノフイ | 置換されたｎ−ヘテロアリールテトラヒドロ−イソキノリン誘導体、その製造及び治療上の使用 |
| EP2569297A1 (en) | 2010-05-11 | 2013-03-20 | Sanofi | Substituted n-heterocycloalkyl bipyrrolidinylphenyl amide derivatives, preparation and therapeutic use thereof |
| EP2569303A1 (en) | 2010-05-11 | 2013-03-20 | Sanofi | Substituted n-alkyl and n-acyl tetrahydro-isoquinoline derivatives, preparation and therapeutic use thereof |
| AR081383A1 (es) | 2010-05-11 | 2012-08-29 | Sanofi Aventis | N-heteroaril bipirrolidin carboxamidas sustituidas, composiciones farmaceuticas que las contienen y uso de las mismas para el tratamiento de enfermedades del sistema nervioso central. |
| EP2569280B1 (en) | 2010-05-11 | 2015-02-25 | Sanofi | Substituted phenyl cycloalkyl pyrrolidine (piperidine) spirolactams and amides, preparation and therapeutic use thereof |
| KR101408699B1 (ko) | 2012-02-29 | 2014-06-19 | 중앙대학교 산학협력단 | 지르코늄 선택적 형광 프루브 |
| KR102127025B1 (ko) * | 2012-07-27 | 2020-06-25 | 비오겐 엠에이 아이엔씨. | S1p 조절제 및/또는 atx 조절제인 화합물들 |
| ES2684995T3 (es) | 2012-07-27 | 2018-10-05 | Biogen Ma Inc. | Derivados del ácido 2-(1-(1-(6-((ciclohexil)oxi)-5-(trifluorometil)naftalen-2-il)etil)piperidin-3-il)acético como moduladores de la autotaxina (atx) para el tratamiento de inflamaciones y trastornos autoinmunes |
| AP2014008139A0 (en) * | 2012-08-23 | 2014-12-31 | Suven Life Sciences Ltd | Acrylamide compounds as histamine H3 receptor ligands |
| CN117229207B (zh) * | 2023-09-01 | 2024-09-03 | 浙江工业大学 | 一种苯基萘类化合物及其制备与应用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19621483A1 (de) * | 1996-05-29 | 1997-12-04 | Hoechst Ag | Substituierte 2-Naphthoylguanidine, Verfahren zur ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| SI0923542T1 (en) * | 1996-05-31 | 2004-02-29 | Pharmacia & Upjohn Company | Aryl substituted cyclic amines as selective dopamine d3 ligands |
| CA2441080A1 (en) * | 2001-03-23 | 2002-10-03 | Eli Lilly And Company | Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses |
| GB0224557D0 (en) * | 2002-10-22 | 2002-11-27 | Glaxo Group Ltd | Novel compounds |
| JP4820094B2 (ja) * | 2002-11-12 | 2011-11-24 | アボット・ラボラトリーズ | ヒスタミン−３受容体リガンドとしての２環式置換アミン |
| MX2007004465A (es) * | 2004-10-19 | 2007-05-07 | Hoffmann La Roche | Derivados de quinolina. |
-
2005
- 2005-05-24 KR KR1020067025300A patent/KR100854212B1/ko not_active Expired - Fee Related
- 2005-05-24 CN CN2005800178164A patent/CN1960727B/zh not_active Expired - Fee Related
- 2005-05-24 AT AT05775021T patent/ATE383857T1/de active
- 2005-05-24 AU AU2005249196A patent/AU2005249196B2/en not_active Ceased
- 2005-05-24 JP JP2007513783A patent/JP4594386B2/ja not_active Expired - Fee Related
- 2005-05-24 PL PL05775021T patent/PL1755593T3/pl unknown
- 2005-05-24 NZ NZ550764A patent/NZ550764A/en unknown
- 2005-05-24 BR BRPI0511778-0A patent/BRPI0511778A/pt not_active IP Right Cessation
- 2005-05-24 DE DE602005004404T patent/DE602005004404T2/de not_active Expired - Lifetime
- 2005-05-24 CA CA2566526A patent/CA2566526C/en not_active Expired - Fee Related
- 2005-05-24 RU RU2006146621/04A patent/RU2387638C2/ru not_active IP Right Cessation
- 2005-05-24 MX MXPA06014017A patent/MXPA06014017A/es active IP Right Grant
- 2005-05-24 EP EP05775021A patent/EP1755593B1/en not_active Expired - Lifetime
- 2005-05-24 DK DK05775021T patent/DK1755593T3/da active
- 2005-05-24 WO PCT/EP2005/005594 patent/WO2005117865A1/en not_active Ceased
- 2005-05-24 ES ES05775021T patent/ES2299074T3/es not_active Expired - Lifetime
- 2005-05-24 PT PT05775021T patent/PT1755593E/pt unknown
- 2005-05-31 TW TW094117927A patent/TWI299992B/zh active
- 2005-05-31 AR ARP050102236A patent/AR049433A1/es not_active Application Discontinuation
- 2005-05-31 MY MYPI20052479A patent/MY139704A/en unknown
- 2005-06-01 US US11/142,738 patent/US7259158B2/en not_active Expired - Fee Related
-
2006
- 2006-11-16 IL IL179370A patent/IL179370A/en not_active IP Right Cessation
- 2006-11-21 ZA ZA200609678A patent/ZA200609678B/xx unknown
- 2006-12-12 NO NO20065733A patent/NO20065733L/no not_active Application Discontinuation
-
2007
- 2007-06-22 US US11/821,263 patent/US7608617B2/en not_active Expired - Fee Related
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