JP2007526336A5 - - Google Patents
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- Publication number
- JP2007526336A5 JP2007526336A5 JP2007502061A JP2007502061A JP2007526336A5 JP 2007526336 A5 JP2007526336 A5 JP 2007526336A5 JP 2007502061 A JP2007502061 A JP 2007502061A JP 2007502061 A JP2007502061 A JP 2007502061A JP 2007526336 A5 JP2007526336 A5 JP 2007526336A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- trifluoromethyl
- cyano
- trifluoroethyl
- cyclopropylmethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US54979404P | 2004-03-03 | 2004-03-03 | |
| US60/549,794 | 2004-03-03 | ||
| PCT/US2005/007245 WO2005085185A1 (en) | 2004-03-03 | 2005-03-03 | Aniline derivatives as selective androgen receptor modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2007526336A JP2007526336A (ja) | 2007-09-13 |
| JP2007526336A5 true JP2007526336A5 (enExample) | 2008-04-17 |
| JP4805909B2 JP4805909B2 (ja) | 2011-11-02 |
Family
ID=34919539
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007502061A Expired - Lifetime JP4805909B2 (ja) | 2004-03-03 | 2005-03-03 | 選択的アンドロゲン受容体モジュレーターとしてのアニリン誘導体 |
Country Status (5)
| Country | Link |
|---|---|
| US (2) | US7514470B2 (enExample) |
| EP (1) | EP1725522B1 (enExample) |
| JP (1) | JP4805909B2 (enExample) |
| ES (1) | ES2523017T3 (enExample) |
| WO (1) | WO2005085185A1 (enExample) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1654221A2 (en) * | 2003-06-10 | 2006-05-10 | Smithkline Beecham Corporation | Aniline derivatived androgen-, glucocorticoid-, mineralcorticoid- and progesterone- receptor modulators |
| JP2007505164A (ja) * | 2003-06-10 | 2007-03-08 | スミスクライン ビーチャム コーポレーション | アンドロゲン、グルココルチコイド、ミネラルコルチコイドおよびプロゲステロン受容体のモジュレーターとしての１−アミノナフタレン類 |
| WO2006113552A2 (en) * | 2005-04-15 | 2006-10-26 | Smithkline Beecham Corporation | Cyanoarylamines |
| EP1954133A4 (en) * | 2005-11-30 | 2010-11-24 | Glaxosmithkline Llc | PYRROLIDINANILINE |
| JP5102985B2 (ja) * | 2006-07-18 | 2012-12-19 | 東ソ−・エフテック株式会社 | 含フッ素２級アミン化合物の製造方法 |
| JP5205379B2 (ja) * | 2006-08-09 | 2013-06-05 | グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー | プロゲステロン受容体モジュレータとしてのピロリジノンアニリン |
| JP5204438B2 (ja) * | 2007-07-31 | 2013-06-05 | 東ソ−・エフテック株式会社 | 含フッ素アミン化合物の製造方法 |
| BRPI0907844B8 (pt) | 2008-02-22 | 2021-05-25 | Radius Health Inc | compostos e método para modular um receptor de andrógeno, processos de preparação e composição farmacêutica dos mesmos e seus usos |
| US8268872B2 (en) | 2008-02-22 | 2012-09-18 | Radius Health, Inc. | Selective androgen receptor modulators |
| MX2010010799A (es) * | 2008-03-31 | 2011-03-25 | Univ Columbia | Metodo de diagnostico, prevencion y tratamiento de las enfermedades de la masa osea. |
| US8623909B2 (en) * | 2008-05-09 | 2014-01-07 | Aska Pharmaceutical Co., Ltd. | Prophylactic/therapeutic agents for lifestyle-related diseases |
| AT509045B1 (de) | 2010-01-29 | 2011-06-15 | Planta Naturstoffe Vertriebsges M B H | Verbindungen zur behandlung von asthma bronchiale |
| US8987319B2 (en) | 2010-02-04 | 2015-03-24 | Radius Health, Inc. | Selective androgen receptor modulators |
| PT2568806T (pt) | 2010-05-12 | 2016-08-05 | Radius Health Inc | Regimes terapêuticos |
| US8642632B2 (en) | 2010-07-02 | 2014-02-04 | Radius Health, Inc. | Selective androgen receptor modulators |
| WO2012047617A1 (en) | 2010-09-28 | 2012-04-12 | Radius Health, Inc. | Selective androgen receptor modulators |
| PL3122426T3 (pl) | 2014-03-28 | 2023-05-15 | Duke University | Leczenie raka sutka z zastosowaniem selektywnych modulatorów receptora estrogenowego |
| US9421264B2 (en) | 2014-03-28 | 2016-08-23 | Duke University | Method of treating cancer using selective estrogen receptor modulators |
| RU2019117364A (ru) * | 2014-10-16 | 2019-08-05 | ДжиТиИкс, ИНК. | Способы лечения урологических нарушений с применением селективных модуляторов андрогеновых рецепторов |
| SMT202200199T1 (it) | 2016-06-22 | 2022-07-21 | Ellipses Pharma Ltd | Metodi di trattamento del cancro del seno ar+. |
| EP4374925A3 (en) | 2017-01-05 | 2025-01-15 | Radius Pharmaceuticals, Inc. | Polymorphic forms of rad1901-2hcl |
| CN112566666A (zh) | 2018-05-14 | 2021-03-26 | 努瓦申生物公司 | 靶向抗癌核激素受体的化合物 |
| CN112423844B (zh) | 2018-07-04 | 2024-08-13 | 雷迪厄斯制药公司 | Rad1901-2hcl的多晶型形式 |
| CN119390714A (zh) | 2019-02-12 | 2025-02-07 | 雷迪厄斯制药公司 | 方法和化合物 |
| AU2020274113A1 (en) | 2019-05-14 | 2021-11-11 | Nuvation Bio Inc. | Anti-cancer nuclear hormone receptor-targeting compounds |
| WO2021097046A1 (en) | 2019-11-13 | 2021-05-20 | Nuvation Bio Inc. | Anti-cancer nuclear hormone receptor-targeting compounds |
| JP2024510792A (ja) | 2021-03-23 | 2024-03-11 | ニューベイション・バイオ・インコーポレイテッド | 抗がん核内ホルモン受容体標的化化合物 |
| JP2024516024A (ja) | 2021-05-03 | 2024-04-11 | ニューベイション・バイオ・インコーポレイテッド | 抗がん核内ホルモン受容体標的化化合物 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2272433A1 (en) * | 1996-11-22 | 1998-05-28 | James E. Audia | N-(aryl/heteroaryl) amino acid esters, pharmaceutical compositions, and methods for inhibiting beta-amyloid peptide release and/or its synthesis |
| JP2001519769A (ja) | 1996-11-22 | 2001-10-23 | エラン・ファーマシューティカルズ・インコーポレイテッド | Ｎ―（アリール／ヘテロアリール）アミノ酸誘導体、その医薬組成物および該化合物を用いたβ―アミロイドペプチドの放出および／またはその合成を阻害する方法 |
| US6506782B1 (en) * | 1998-02-27 | 2003-01-14 | Athena Neurosciences, Inc. | Heterocyclic compounds, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds |
| ES2243500T3 (es) * | 2000-06-06 | 2005-12-01 | Warner-Lambert Company Llc | Ciclohexilaminas biciclicas y uso como antegonistas del receptor nmda. |
| MXPA03001632A (es) | 2000-08-24 | 2004-09-10 | Univ Tennessee Res Corp | Moduladores receptores de androgeno selectivos y metodos para usar los mismos. |
| CN1176905C (zh) * | 2002-03-22 | 2004-11-24 | 清华大学 | 甘氨酸乙酯邻苯二腈及其合成方法与应用 |
| EP1654221A2 (en) * | 2003-06-10 | 2006-05-10 | Smithkline Beecham Corporation | Aniline derivatived androgen-, glucocorticoid-, mineralcorticoid- and progesterone- receptor modulators |
-
2005
- 2005-03-03 JP JP2007502061A patent/JP4805909B2/ja not_active Expired - Lifetime
- 2005-03-03 US US10/598,508 patent/US7514470B2/en not_active Expired - Lifetime
- 2005-03-03 EP EP05730067.5A patent/EP1725522B1/en not_active Expired - Lifetime
- 2005-03-03 ES ES05730067.5T patent/ES2523017T3/es not_active Expired - Lifetime
- 2005-03-03 WO PCT/US2005/007245 patent/WO2005085185A1/en not_active Ceased
-
2009
- 2009-02-25 US US12/392,687 patent/US7723385B2/en not_active Expired - Lifetime
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