JP2007502264A5 - - Google Patents

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Publication number
JP2007502264A5
JP2007502264A5 JP2006523062A JP2006523062A JP2007502264A5 JP 2007502264 A5 JP2007502264 A5 JP 2007502264A5 JP 2006523062 A JP2006523062 A JP 2006523062A JP 2006523062 A JP2006523062 A JP 2006523062A JP 2007502264 A5 JP2007502264 A5 JP 2007502264A5
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JP
Japan
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compound
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JP2006523062A
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English (en)
Japanese (ja)
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JP2007502264A (ja
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Priority claimed from GBGB0319124.4A external-priority patent/GB0319124D0/en
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Publication of JP2007502264A publication Critical patent/JP2007502264A/ja
Publication of JP2007502264A5 publication Critical patent/JP2007502264A5/ja
Withdrawn legal-status Critical Current

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JP2006523062A 2003-08-14 2004-08-13 Ｈｍ７４ａ受容体アゴニストとしての２−置換安息香酸誘導体 Withdrawn JP2007502264A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0319124.4A GB0319124D0 (en) 2003-08-14 2003-08-14 Chemical compounds
PCT/GB2004/003528 WO2005016870A1 (en) 2003-08-14 2004-08-13 2-substituted benzoic acid derivatives as hm74a receptor agonists

Publications (2)

Publication Number Publication Date
JP2007502264A JP2007502264A (ja) 2007-02-08
JP2007502264A5 true JP2007502264A5 (enExample) 2007-09-13

Family

ID=28052522

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006523062A Withdrawn JP2007502264A (ja) 2003-08-14 2004-08-13 Ｈｍ７４ａ受容体アゴニストとしての２−置換安息香酸誘導体

Country Status (4)

Country Link
EP (1) EP1670749A1 (enExample)
JP (1) JP2007502264A (enExample)
GB (1) GB0319124D0 (enExample)
WO (1) WO2005016870A1 (enExample)

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JP5254620B2 (ja) 2004-12-03 2013-08-07 メルク・シャープ・アンド・ドーム・コーポレーション Ｃｂ１アンタゴニストとしての置換ピペラジン
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JP2009520820A (ja) * 2005-12-20 2009-05-28 メルク エンド カムパニー インコーポレーテッド ナイアシン受容体アゴニスト、前記化合物を含む組成物及び治療方法
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JP2009533436A (ja) * 2006-04-11 2009-09-17 メルク エンド カムパニー インコーポレーテッド ナイアシン受容体アゴニスト、かかる化合物を含有する組成物、及び治療法
WO2008016676A2 (en) * 2006-08-02 2008-02-07 Cytokinetics, Incorporated Certain chemical entities, compositions, and methods
US8063082B2 (en) * 2006-08-02 2011-11-22 Cytokinetics, Inc. Certain chemical entities, compositions, and methods
US8071625B2 (en) 2006-08-02 2011-12-06 Cytokinetics, Inc. Certain chemical entities, compositions, and methods
WO2008069611A1 (en) * 2006-12-08 2008-06-12 Korea Research Institute Of Chemical Technology N-phenylamide derivative, process for the preparation thereof, and composition for preventing or treating ischemic diseases comprising same
KR100832750B1 (ko) 2006-12-08 2008-05-27 한국화학연구원 Ｎ-페닐아마이드 유도체를 함유하는 허혈성 질환의 예방또는 치료용 조성물
WO2008144423A2 (en) * 2007-05-15 2008-11-27 Medical College Of Georgia Research Institute, Inc. Compositions comprising a gpr109 ligand for treating disorders of the digestive tract and/or cancer
JP5670731B2 (ja) 2007-08-15 2015-02-18 サイトキネティクス・インコーポレーテッドＣｙｔｏｋｉｎｅｔｉｃｓ Ｉｎｃｏｒｐｏｒａｔｅｄ ある種の化学物質、組成物、および方法
WO2009123241A1 (ja) 2008-03-31 2009-10-08 株式会社レナサイエンス プラスミノーゲンアクチベーターインヒビター－１阻害剤
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US8664425B2 (en) * 2010-02-02 2014-03-04 Honeywell International Inc. Bluegreen fluorescent compounds
WO2012034116A2 (en) * 2010-09-10 2012-03-15 The Johns Hopkins University Small molecules as epigenetic modulators of lysine-specific demethylase 1 and methods of treating disorders
WO2013092786A1 (en) * 2011-12-23 2013-06-27 Norgine B.V. Compositions comprising cetilistat
EP2990057B1 (en) 2013-04-15 2019-03-20 Renascience Co., Ltd. Pai-1 inhibitor for use in enhancing the antitumor effect of an antitumor agent in a patient
CN104418764B (zh) * 2013-09-11 2017-02-01 上海伊明化学科技有限公司 一种二氢燕麦酰基邻氨基苯甲酸d合成方法
ES2578377B1 (es) * 2014-12-22 2017-05-04 Consejo Superior De Investigaciones Científicas (Csic) Compuestos moduladores del sensor neuronal de calcio dream y sus usos terapéuticos.
CN106511110B (zh) * 2016-10-25 2019-10-01 福州美乐莲生物科技有限公司 二氢燕麦生物碱d盐类化合物作为化妆品活性成分的应用及其合成方法
WO2019034690A1 (en) 2017-08-15 2019-02-21 Inflazome Limited SULFONYLURATES AND SULFONYLTHIOURES AS INHIBITORS OF NLRP3
US11926600B2 (en) 2017-08-15 2024-03-12 Inflazome Limited Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors
UY37848A (es) 2017-08-15 2019-03-29 Inflazome Ltd Sulfonilureas y sulfoniltioureas útiles como inhibidores de nlrp3
EP3707134A1 (en) 2017-11-09 2020-09-16 Inflazome Limited Novel sulfonamide carboxamide compounds
US12221434B2 (en) 2017-11-09 2025-02-11 Inflazome Limited Sulfonamide carboxamide compounds
US11905252B2 (en) 2018-03-02 2024-02-20 Inflazome Limited Compounds
EP3662908A1 (en) * 2018-12-04 2020-06-10 Consejo Superior de Investigaciones Cientificas (CSIC) Modulating compounds of kchip2 and its use for the treatment of cardiovascular pathologies
CN109553550B (zh) * 2018-12-29 2022-02-22 上海克琴科技有限公司 一种合成二氢燕麦生物碱的方法
CN112939803B (zh) * 2021-02-07 2023-07-18 郑州轻工业大学 一种二氢燕麦生物碱d的制备工艺
CN114478296B (zh) * 2022-02-14 2024-07-19 河南旭瑞新材料科技有限公司 一种二氢燕麦生物碱的制备方法

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FR2763334A1 (fr) * 1997-05-13 1998-11-20 Lipha Derives anthraniliques
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WO2000027823A1 (en) * 1998-11-09 2000-05-18 James Black Foundation Limited Gastrin and cholecystokinin receptor ligands
AR022204A1 (es) * 1999-01-08 2002-09-04 Norgine Bv Compuesto, proceso para su preparacion, composicion farmaceutica y producto comestible que lo comprende.
AU2001234089B2 (en) * 2000-02-15 2005-08-11 Teijin Limited Cancer remedy comprising anthranilic acid derivative as active ingredient
DE10133665A1 (de) * 2001-07-11 2003-01-30 Boehringer Ingelheim Pharma Carbonsäurederivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Herstellung

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