JP2007523177A5 - - Google Patents

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Publication number
JP2007523177A5
JP2007523177A5 JP2006554220A JP2006554220A JP2007523177A5 JP 2007523177 A5 JP2007523177 A5 JP 2007523177A5 JP 2006554220 A JP2006554220 A JP 2006554220A JP 2006554220 A JP2006554220 A JP 2006554220A JP 2007523177 A5 JP2007523177 A5 JP 2007523177A5
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JP
Japan
Prior art keywords
compound
fluorophenyl
phenyl
tumor
ethyl
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JP2006554220A
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English (en)
Japanese (ja)
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JP4934432B2 (ja
JP2007523177A (ja
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Priority claimed from PCT/US2005/005151 external-priority patent/WO2005080352A2/en
Publication of JP2007523177A publication Critical patent/JP2007523177A/ja
Publication of JP2007523177A5 publication Critical patent/JP2007523177A5/ja
Application granted granted Critical
Publication of JP4934432B2 publication Critical patent/JP4934432B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2006554220A 2004-02-19 2005-02-17 キナゾリン誘導体およびキナゾリン誘導体の治療への使用 Expired - Fee Related JP4934432B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US54548704P 2004-02-19 2004-02-19
US60/545,487 2004-02-19
PCT/US2005/005151 WO2005080352A2 (en) 2004-02-19 2005-02-17 Quinazoline derivatives and therapeutic use thereof

Publications (3)

Publication Number Publication Date
JP2007523177A JP2007523177A (ja) 2007-08-16
JP2007523177A5 true JP2007523177A5 (https=) 2008-03-13
JP4934432B2 JP4934432B2 (ja) 2012-05-16

Family

ID=34886161

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006554220A Expired - Fee Related JP4934432B2 (ja) 2004-02-19 2005-02-17 キナゾリン誘導体およびキナゾリン誘導体の治療への使用

Country Status (11)

Country Link
US (2) US7388014B2 (https=)
EP (2) EP2650286A1 (https=)
JP (1) JP4934432B2 (https=)
KR (1) KR100942865B1 (https=)
CN (1) CN1956966B (https=)
AU (1) AU2005214373B2 (https=)
BR (1) BRPI0507903A (https=)
CA (1) CA2557433C (https=)
ES (1) ES2554330T3 (https=)
MX (1) MXPA06009475A (https=)
WO (1) WO2005080352A2 (https=)

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AU2007249762A1 (en) * 2006-05-15 2007-11-22 Senex Biotechnology, Inc Identification of CDKI pathway inhibitors
WO2008124823A1 (en) * 2007-04-10 2008-10-16 Myriad Genetics, Inc. Method of treating melanoma
CN101120945B (zh) * 2007-07-30 2010-11-24 浙江大学 8-芳胺基-3H-咪唑[4,5-g]喹唑啉类衍生物的用途
PH12012500097A1 (en) * 2009-07-21 2011-01-27 Shanghai Inst Organic Chem Potent small molecule inhibitors of autophagy, and methods of use thereof
WO2012006960A1 (en) * 2010-07-14 2012-01-19 Zhejiang Beta Pharma Inc. NOVEL FUSED HETEROCYCLIC DERIVATIVES USEFUL AS c-MET TYROSINE KINASE INHIBITORS
US20140309224A1 (en) * 2011-09-13 2014-10-16 Roninson Igor B TREATMENT OF DISEASES OR DISORDERS CAUSED BY INDUCED NFkB TRANSCRIPTIONAL ACTIVITY
CN103086984A (zh) * 2011-11-03 2013-05-08 南京大学 一类4-苯氨基喹唑啉类衍生物及其制备方法与用途
WO2013135671A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
CN102659692B (zh) 2012-05-04 2014-04-09 郑州泰基鸿诺药物科技有限公司 双联厄洛替尼及其制备方法
CN102875570B (zh) * 2012-10-23 2015-11-04 浙江大学 喹唑啉衍生物及其制备方法和用途
JP6464139B2 (ja) 2013-03-14 2019-02-06 コンバージーン・リミテッド・ライアビリティ・カンパニーＣｏｎｖｅｒｇｅｎｅ Ｌｌｃ ブロモドメイン含有タンパク質の阻害のための方法および組成物
WO2015036058A1 (en) 2013-09-16 2015-03-19 Basf Se Fungicidal pyrimidine compounds
WO2015036059A1 (en) 2013-09-16 2015-03-19 Basf Se Fungicidal pyrimidine compounds
RU2016112013A (ru) * 2013-09-19 2017-10-24 Пьер Фабр Медикамент Производные хиназолина и их применение в качестве ингибиторов днк-метилтрансферазы
CN104926798B (zh) * 2014-03-21 2019-06-18 江苏豪森药业集团有限公司 阿法替尼中间体的高纯度制备方法
CA3006300C (en) 2015-11-25 2024-02-27 Convergene Llc Bicyclic bet bromodomain inhibitors and uses thereof
JP7191446B2 (ja) * 2017-01-30 2022-12-19 塩野義製薬株式会社 キナゾリン誘導体を含有する固形製剤
EP3897651A4 (en) * 2018-12-21 2022-09-21 University of Notre Dame du Lac DISCOVERY OF BD-OXIDASE INHIBITORS FOR THE TREATMENT OF MYCOBACTERIAL DISEASES
EP4424379A3 (en) 2019-04-24 2024-10-30 Convergene Llc Small molecule bromodomain inhibitors and uses thereof
KR102397359B1 (ko) * 2019-09-30 2022-05-11 한국화학연구원 4-아미노-퀴나졸린 유도체 및 이를 포함하는 항바이러스용 조성물
KR20220132543A (ko) * 2019-12-27 2022-09-30 루핀 리미티드 치환된 삼환 화합물
TWI807787B (zh) * 2021-04-19 2023-07-01 大陸商昆藥集團股份有限公司 苯並嘧啶三環衍生物及製備方法和應用
CN116444443B (zh) * 2023-03-15 2025-09-05 广东省中医院（广州中医药大学第二附属医院、广州中医药大学第二临床医学院、广东省中医药科学院） 一种苯甲酰-喹唑啉酮衍生物及其制备方法与应用

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