JP2007522210A5 - - Google Patents

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Publication number
JP2007522210A5
JP2007522210A5 JP2006553086A JP2006553086A JP2007522210A5 JP 2007522210 A5 JP2007522210 A5 JP 2007522210A5 JP 2006553086 A JP2006553086 A JP 2006553086A JP 2006553086 A JP2006553086 A JP 2006553086A JP 2007522210 A5 JP2007522210 A5 JP 2007522210A5
Authority
JP
Japan
Prior art keywords
amino
carboxamide
methyl
ethyl
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006553086A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007522210A (ja
Filing date
Publication date
Priority claimed from SE0400284A external-priority patent/SE0400284D0/xx
Application filed filed Critical
Publication of JP2007522210A publication Critical patent/JP2007522210A/ja
Publication of JP2007522210A5 publication Critical patent/JP2007522210A5/ja
Pending legal-status Critical Current

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JP2006553086A 2004-02-10 2005-02-07 JAK3キナーゼ修飾物質としての新規なキノリン−カルボキシアミド(carbaxamide) Pending JP2007522210A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0400284A SE0400284D0 (sv) 2004-02-10 2004-02-10 Novel compounds
PCT/SE2005/000156 WO2005075429A1 (en) 2004-02-10 2005-02-07 Novel quinoline-carbaxamides as jack3 kinase modulators

Publications (2)

Publication Number Publication Date
JP2007522210A JP2007522210A (ja) 2007-08-09
JP2007522210A5 true JP2007522210A5 (cg-RX-API-DMAC7.html) 2008-03-21

Family

ID=31885281

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006553086A Pending JP2007522210A (ja) 2004-02-10 2005-02-07 JAK3キナーゼ修飾物質としての新規なキノリン−カルボキシアミド(carbaxamide)

Country Status (9)

Country Link
US (1) US20080153799A1 (cg-RX-API-DMAC7.html)
EP (1) EP1718615A1 (cg-RX-API-DMAC7.html)
JP (1) JP2007522210A (cg-RX-API-DMAC7.html)
CN (1) CN1942445A (cg-RX-API-DMAC7.html)
AR (1) AR047609A1 (cg-RX-API-DMAC7.html)
SE (1) SE0400284D0 (cg-RX-API-DMAC7.html)
TW (1) TW200529838A (cg-RX-API-DMAC7.html)
UY (1) UY28745A1 (cg-RX-API-DMAC7.html)
WO (1) WO2005075429A1 (cg-RX-API-DMAC7.html)

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US7297700B2 (en) 2005-03-24 2007-11-20 Renovis, Inc. Bicycloheteroaryl compounds as P2X7 modulators and uses thereof
US7470787B2 (en) * 2005-07-11 2008-12-30 Aerie Pharmaceuticals, Inc. Isoquinoline compounds
TWI464148B (zh) 2006-03-16 2014-12-11 Evotec Us Inc 作為p2x7調節劑之雙環雜芳基化合物與其用途
TW200808732A (en) * 2006-04-14 2008-02-16 Astrazeneca Ab Chemical compounds
EP2526948A1 (en) 2006-09-20 2012-11-28 Aerie Pharmaceuticals, Inc. RHO kinase inhibitors
TW200831488A (en) 2006-11-29 2008-08-01 Astrazeneca Ab Novel compounds
US8455513B2 (en) 2007-01-10 2013-06-04 Aerie Pharmaceuticals, Inc. 6-aminoisoquinoline compounds
JO2704B1 (en) 2007-09-21 2013-03-03 جانسين فارماسوتيكا ان في Interference inhibition factors between MD2 and B53
US8455514B2 (en) * 2008-01-17 2013-06-04 Aerie Pharmaceuticals, Inc. 6-and 7-amino isoquinoline compounds and methods for making and using the same
US8450344B2 (en) 2008-07-25 2013-05-28 Aerie Pharmaceuticals, Inc. Beta- and gamma-amino-isoquinoline amide compounds and substituted benzamide compounds
EP2361902A4 (en) * 2008-11-21 2012-04-25 Astellas Pharma Inc 4,6-DIAMINONICOTINSÄUREAMIDVERBINDUNG
US8575153B2 (en) 2008-11-28 2013-11-05 Kowa Company, Ltd. Pyridine-3-carboxyamide derivative
ES2834451T3 (es) 2009-05-01 2021-06-17 Aerie Pharmaceuticals Inc Inhibidores de mecanismo doble para el tratamiento de enfermedades
US20120065199A1 (en) * 2009-05-20 2012-03-15 Clanotech Ab Substituted quinolines for use as vegf inhibitors
WO2012061557A2 (en) * 2010-11-05 2012-05-10 Glaxosmithkline Llc Chemical compounds
HK1217092A1 (zh) 2013-02-15 2016-12-23 Kala Pharmaceuticals, Inc. 治疗性化合物及其用途
ES2831625T3 (es) 2013-02-20 2021-06-09 Kala Pharmaceuticals Inc Compuestos terapéuticos y sus usos
US9688688B2 (en) 2013-02-20 2017-06-27 Kala Pharmaceuticals, Inc. Crystalline forms of 4-((4-((4-fluoro-2-methyl-1H-indol-5-yl)oxy)-6-methoxyquinazolin-7-yl)oxy)-1-(2-oxa-7-azaspiro[3.5]nonan-7-yl)butan-1-one and uses thereof
CN110396085B (zh) 2013-03-15 2024-11-15 爱尔康公司 联合治疗
US9890173B2 (en) 2013-11-01 2018-02-13 Kala Pharmaceuticals, Inc. Crystalline forms of therapeutic compounds and uses thereof
KR20160099084A (ko) 2013-11-01 2016-08-19 칼라 파마슈티컬스, 인크. 치료 화합물의 결정질 형태 및 그의 용도
WO2017086941A1 (en) 2015-11-17 2017-05-26 Aerie Pharmaceuticals, Inc. Process for the preparation of kinase inhibitors and intermediates thereof
US9643927B1 (en) 2015-11-17 2017-05-09 Aerie Pharmaceuticals, Inc. Process for the preparation of kinase inhibitors and intermediates thereof
CN109640966A (zh) 2016-08-31 2019-04-16 爱瑞制药公司 眼用组合物
US10253036B2 (en) 2016-09-08 2019-04-09 Kala Pharmaceuticals, Inc. Crystalline forms of therapeutic compounds and uses thereof
KR20190051010A (ko) 2016-09-08 2019-05-14 칼라 파마슈티컬스, 인크. 치료 화합물의 결정형 및 그의 용도
US10392399B2 (en) 2016-09-08 2019-08-27 Kala Pharmaceuticals, Inc. Crystalline forms of therapeutic compounds and uses thereof
KR20190135027A (ko) 2017-03-31 2019-12-05 에어리 파마슈티컬즈, 인코포레이티드 아릴 시클로프로필-아미노-이소퀴놀리닐 아미드 화합물
CA3112391A1 (en) 2018-09-14 2020-03-19 Aerie Pharmaceuticals, Inc. Aryl cyclopropyl-amino-isoquinolinyl amide compounds
CN111269215B (zh) * 2020-04-01 2021-10-26 中科利健制药(广州)有限公司 含氮杂环有机化合物及其制备方法和应用
TW202345806A (zh) 2022-03-31 2023-12-01 美商艾伯維有限公司 噻唑并〔5,4-b〕吡啶malt-1抑制劑

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GB8621425D0 (en) * 1986-09-05 1986-10-15 Smith Kline French Lab Compounds
GB8804447D0 (en) * 1988-02-25 1988-03-23 Smithkline Beckman Intercredit Compounds
DK273689A (da) * 1988-06-06 1989-12-07 Sanofi Sa 4-amino-3-carboxyquinoliner og -naphthyridiner, fremgangsmaade til deres fremstilling og anvendelse deraf i laegemidler
AU634880B2 (en) * 1990-03-28 1993-03-04 Otsuka Pharmaceutical Co., Ltd. Quinoline derivative, antiulcer drug containing the same, and production of said derivative
UA73073C2 (uk) * 1997-04-03 2005-06-15 Уайт Холдінгз Корпорейшн Заміщені 3-ціанохіноліни, спосіб їх одержання та фармацевтична композиція
SE0101675D0 (sv) * 2001-05-11 2001-05-11 Astrazeneca Ab Novel composition

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