JP2007500716A5 - - Google Patents

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Publication number
JP2007500716A5
JP2007500716A5 JP2006522073A JP2006522073A JP2007500716A5 JP 2007500716 A5 JP2007500716 A5 JP 2007500716A5 JP 2006522073 A JP2006522073 A JP 2006522073A JP 2006522073 A JP2006522073 A JP 2006522073A JP 2007500716 A5 JP2007500716 A5 JP 2007500716A5
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JP
Japan
Prior art keywords
alkyl
group
hydrogen
cycloalkyl
independently selected
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JP2006522073A
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English (en)
Japanese (ja)
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JP2007500716A (ja
JP4884219B2 (ja
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Priority claimed from PCT/US2004/024542 external-priority patent/WO2005011654A2/en
Publication of JP2007500716A publication Critical patent/JP2007500716A/ja
Publication of JP2007500716A5 publication Critical patent/JP2007500716A5/ja
Application granted granted Critical
Publication of JP4884219B2 publication Critical patent/JP4884219B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2006522073A 2003-07-29 2004-07-29 ピリジル誘導体および治療剤としてのその用途 Expired - Fee Related JP4884219B2 (ja)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
US49114003P 2003-07-29 2003-07-29
US60/491,140 2003-07-29
US49108003P 2003-07-30 2003-07-30
US49132203P 2003-07-30 2003-07-30
US49114103P 2003-07-30 2003-07-30
US49111603P 2003-07-30 2003-07-30
US60/491,322 2003-07-30
US60/491,141 2003-07-30
US60/491,116 2003-07-30
US60/491,080 2003-07-30
PCT/US2004/024542 WO2005011654A2 (en) 2003-07-29 2004-07-29 Pyridyl derivatives and their use as therapeutic agents

Publications (3)

Publication Number Publication Date
JP2007500716A JP2007500716A (ja) 2007-01-18
JP2007500716A5 true JP2007500716A5 (enExample) 2007-09-13
JP4884219B2 JP4884219B2 (ja) 2012-02-29

Family

ID=34120125

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006522073A Expired - Fee Related JP4884219B2 (ja) 2003-07-29 2004-07-29 ピリジル誘導体および治療剤としてのその用途

Country Status (17)

Country Link
US (3) US7763618B2 (enExample)
EP (1) EP1651605B1 (enExample)
JP (1) JP4884219B2 (enExample)
KR (1) KR20060036105A (enExample)
AT (1) ATE556056T1 (enExample)
AU (1) AU2004261250B2 (enExample)
BR (1) BRPI0413059A (enExample)
CA (1) CA2533898A1 (enExample)
EC (1) ECSP066314A (enExample)
ES (1) ES2386354T3 (enExample)
IL (1) IL173397A0 (enExample)
MA (1) MA28012A1 (enExample)
MX (1) MXPA06001202A (enExample)
NO (1) NO20060973L (enExample)
SG (1) SG145695A1 (enExample)
TN (1) TNSN06035A1 (enExample)
WO (1) WO2005011654A2 (enExample)

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BRPI0719122A2 (pt) 2006-08-24 2013-12-10 Novartis Ag Compostos orgânicos
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US7638541B2 (en) 2006-12-28 2009-12-29 Metabolex Inc. 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine
WO2008091863A1 (en) 2007-01-23 2008-07-31 Kalypsys, Inc. Sulfonyl-substituted bicyclic compounds as ppar modulators for the treatment of non-alcoholic steatohepatitis
WO2008096746A1 (ja) 2007-02-06 2008-08-14 Takeda Pharmaceutical Company Limited スピロ化合物およびその用途
EP2142529B1 (en) * 2007-04-27 2013-12-25 Purdue Pharma LP Trpv1 antagonists and uses thereof
US7842696B2 (en) 2007-06-21 2010-11-30 Forest Laboratories Holdings Limited Piperazine derivatives as inhibitors of stearoyl-CoA desaturase
AU2008279447A1 (en) 2007-07-19 2009-01-29 Metabolex, Inc. N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the RUP3 or GPR119 receptor for the treatment of diabetes and metabolic disorders
CN101821234B (zh) 2007-08-08 2014-06-25 格里斯威医药有限责任公司 苯氧基吡咯烷衍生物及其应用和组合物
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CN105596291B (zh) * 2014-11-24 2020-09-08 辽宁海思科制药有限公司 一种磺达肝癸钠注射液组合物
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MA47212A (fr) 2017-01-06 2019-11-13 Yumanity Therapeutics Inc Méthodes de traitement de troubles neurologiques
WO2019084157A1 (en) 2017-10-24 2019-05-02 Yumanity Therapeutics, Inc. COMPOUNDS AND USES THEREOF
CN111386272B (zh) 2017-10-27 2023-01-06 费森尤斯卡比肿瘤学有限公司 一种改进的瑞博西尼及其盐的制备方法
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EA202192047A1 (ru) 2019-11-13 2021-12-08 Юманити Терапьютикс, Инк. Соединения и их применение

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