JP2006526656A - 5員ヘテロ環ベースのp−38阻害剤 - Google Patents

5員ヘテロ環ベースのp−38阻害剤 Download PDF

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JP2006526656A
JP2006526656A JP2006515154A JP2006515154A JP2006526656A JP 2006526656 A JP2006526656 A JP 2006526656A JP 2006515154 A JP2006515154 A JP 2006515154A JP 2006515154 A JP2006515154 A JP 2006515154A JP 2006526656 A JP2006526656 A JP 2006526656A
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alkyl
substituted
methyl
aryl
cycloalkyl
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ドン・チン
ファブリス・ピエール
ワン・チアンチアン
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ノバルティス アクチエンゲゼルシャフト
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    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/071,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
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    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D263/34Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Neurology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
JP2006515154A 2003-06-03 2004-06-02 5員ヘテロ環ベースのp−38阻害剤 Pending JP2006526656A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US47566203P 2003-06-03 2003-06-03
US53154103P 2003-12-19 2003-12-19
PCT/US2004/017580 WO2005000298A2 (en) 2003-06-03 2004-06-02 5-membered heterocycle-based p-38 inhibitors

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JP2006526656A true JP2006526656A (ja) 2006-11-24
JP2006526656A5 JP2006526656A5 (https=) 2007-08-16

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JP2006515154A Pending JP2006526656A (ja) 2003-06-03 2004-06-02 5員ヘテロ環ベースのp−38阻害剤

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US (2) US7652044B2 (https=)
EP (1) EP1635824B1 (https=)
JP (1) JP2006526656A (https=)
AT (1) ATE439837T1 (https=)
AU (1) AU2004251668B2 (https=)
BR (1) BRPI0410905A (https=)
CA (1) CA2528438A1 (https=)
DE (1) DE602004022668D1 (https=)
ES (1) ES2332135T3 (https=)
MX (1) MXPA05013075A (https=)
PL (1) PL1635824T3 (https=)
PT (1) PT1635824E (https=)
WO (1) WO2005000298A2 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
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JP2007509130A (ja) * 2003-10-23 2007-04-12 アブ サイエンス チロシンキナーゼ阻害薬としての2−アミノアリールオキサゾール化合物

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