JP2005538035A - グアニジニウム輸送試薬および結合体 - Google Patents

グアニジニウム輸送試薬および結合体 Download PDF

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Publication number
JP2005538035A
JP2005538035A JP2003550821A JP2003550821A JP2005538035A JP 2005538035 A JP2005538035 A JP 2005538035A JP 2003550821 A JP2003550821 A JP 2003550821A JP 2003550821 A JP2003550821 A JP 2003550821A JP 2005538035 A JP2005538035 A JP 2005538035A
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group
compound
transport
agent
biologically active
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Japanese (ja)
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JP2005538035A5 (https=
Inventor
ジョナサン ビー． ロスバード，
ポール エー． ウェンダー，
カナカ パタビラマン，
エリン ティー． ペルキー，
セオドア シー． ジェソップ，
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Leland Stanford Junior University
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Leland Stanford Junior University
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Publication of JP2005538035A publication Critical patent/JP2005538035A/ja
Publication of JP2005538035A5 publication Critical patent/JP2005538035A5/ja
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2003550821A 2001-12-11 2002-12-11 グアニジニウム輸送試薬および結合体 Pending JP2005538035A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33969601P 2001-12-11 2001-12-11
PCT/US2002/039698 WO2003049772A2 (en) 2001-12-11 2002-12-11 Guanidinium transport reagents and conjugates

Publications (2)

Publication Number Publication Date
JP2005538035A true JP2005538035A (ja) 2005-12-15
JP2005538035A5 JP2005538035A5 (https=) 2006-11-02

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JP2003550821A Pending JP2005538035A (ja) 2001-12-11 2002-12-11 グアニジニウム輸送試薬および結合体

Country Status (7)

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US (1) US7169814B2 (https=)
EP (1) EP1461084A2 (https=)
JP (1) JP2005538035A (https=)
AU (1) AU2002359679B2 (https=)
CA (1) CA2469336C (https=)
MX (1) MXPA04005611A (https=)
WO (1) WO2003049772A2 (https=)

Cited By (3)

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JP2010504929A (ja) * 2006-09-27 2010-02-18 ボッティ，パオロ 生体系への送達を高める手段及び方法
JP2013028633A (ja) * 2005-12-30 2013-02-07 Revance Therapeutics Inc 局所投与用アルギニンヘテロマー
JP2020527127A (ja) * 2017-05-19 2020-09-03 ルネラ・バイオテック・インコーポレーテッド アンチミトシン：癌幹細胞を根絶するためのミトコンドリア生合成の標的阻害薬

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JP2013028633A (ja) * 2005-12-30 2013-02-07 Revance Therapeutics Inc 局所投与用アルギニンヘテロマー
JP2010504929A (ja) * 2006-09-27 2010-02-18 ボッティ，パオロ 生体系への送達を高める手段及び方法
US9211340B2 (en) 2006-09-27 2015-12-15 Paolo Botti Means and methods of enhancing delivery to biological systems
JP2020527127A (ja) * 2017-05-19 2020-09-03 ルネラ・バイオテック・インコーポレーテッド アンチミトシン：癌幹細胞を根絶するためのミトコンドリア生合成の標的阻害薬

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CA2469336A1 (en) 2003-06-19
US7169814B2 (en) 2007-01-30
US20040161405A9 (en) 2004-08-19
AU2002359679A1 (en) 2003-06-23
WO2003049772A2 (en) 2003-06-19
AU2002359679B2 (en) 2009-01-08
US20030185788A1 (en) 2003-10-02
EP1461084A2 (en) 2004-09-29
MXPA04005611A (es) 2005-04-19
WO2003049772A3 (en) 2003-11-20
CA2469336C (en) 2013-06-11

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