JP2005532289A - 持続放出性医薬製剤及びその製造方法 - Google Patents

持続放出性医薬製剤及びその製造方法 Download PDF

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Publication number
JP2005532289A
JP2005532289A JP2003583385A JP2003583385A JP2005532289A JP 2005532289 A JP2005532289 A JP 2005532289A JP 2003583385 A JP2003583385 A JP 2003583385A JP 2003583385 A JP2003583385 A JP 2003583385A JP 2005532289 A JP2005532289 A JP 2005532289A
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Prior art keywords
sustained release
albuterol
sustained
hours
formulation
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Japanese (ja)
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JP2005532289A5 (enExample
Inventor
ダヴェジバイ クンバニ
ハリシュ ビー パンディア
ハイレン パテル
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プリヴァ インコーポレイテッド
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Publication of JP2005532289A publication Critical patent/JP2005532289A/ja
Publication of JP2005532289A5 publication Critical patent/JP2005532289A5/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators

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  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
JP2003583385A 2002-04-12 2003-04-11 持続放出性医薬製剤及びその製造方法 Pending JP2005532289A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/120,501 US7125563B2 (en) 2002-04-12 2002-04-12 Sustained release pharmaceutical preparations and methods for producing the same
PCT/US2003/009210 WO2003086364A1 (en) 2002-04-12 2003-04-11 Sustained release pharmaceutical prepartations and methods for producing the same

Publications (2)

Publication Number Publication Date
JP2005532289A true JP2005532289A (ja) 2005-10-27
JP2005532289A5 JP2005532289A5 (enExample) 2006-06-01

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ID=29214431

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JP2003583385A Pending JP2005532289A (ja) 2002-04-12 2003-04-11 持続放出性医薬製剤及びその製造方法

Country Status (10)

Country Link
US (3) US7125563B2 (enExample)
EP (1) EP1494653A1 (enExample)
JP (1) JP2005532289A (enExample)
CN (1) CN1655765A (enExample)
AU (1) AU2003218397A1 (enExample)
CA (1) CA2481667A1 (enExample)
HR (1) HRP20040945A2 (enExample)
PL (1) PL373328A1 (enExample)
RU (1) RU2004133532A (enExample)
WO (1) WO2003086364A1 (enExample)

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GB0203296D0 (en) 2002-02-12 2002-03-27 Glaxo Group Ltd Novel composition
US8637512B2 (en) 2002-07-29 2014-01-28 Glaxo Group Limited Formulations and method of treatment
ATE341312T1 (de) * 2003-05-20 2006-10-15 Ethypharm Sa Orale pharmazeutische zusammensetzung mit verzögerter freisetzung
EP2112920B1 (en) 2003-06-26 2018-07-25 Intellipharmaceutics Corp. Proton pump-inhibitor-containing capsules which comprise subunits differently structured for a delayed release of the active ingredient
US8394409B2 (en) 2004-07-01 2013-03-12 Intellipharmaceutics Corp. Controlled extended drug release technology
US10624858B2 (en) 2004-08-23 2020-04-21 Intellipharmaceutics Corp Controlled release composition using transition coating, and method of preparing same
US10064828B1 (en) 2005-12-23 2018-09-04 Intellipharmaceutics Corp. Pulsed extended-pulsed and extended-pulsed pulsed drug delivery systems
EP2018160B1 (en) 2006-03-16 2011-12-14 Tris Pharma, Inc. Modified release formulations containing drug-ion exchange resin complexes
WO2007112581A1 (en) * 2006-04-03 2007-10-11 Isa Odidi Controlled release delivery device comprising an organosol coat
US10960077B2 (en) 2006-05-12 2021-03-30 Intellipharmaceutics Corp. Abuse and alcohol resistant drug composition
EP2296634A1 (en) * 2008-06-02 2011-03-23 Dexcel Pharma Technologies Ltd. Process for manufacture of a medicament with granulation and pan coating
WO2011102504A1 (ja) 2010-02-22 2011-08-25 第一三共株式会社 経口用徐放性固形製剤
EP2540294B1 (en) * 2010-02-22 2016-08-03 Daiichi Sankyo Company, Limited Sustained-release solid preparation for oral use
US8623409B1 (en) 2010-10-20 2014-01-07 Tris Pharma Inc. Clonidine formulation
KR102127625B1 (ko) 2012-09-03 2020-06-29 다이이찌 산쿄 가부시키가이샤 하이드로모르폰염산염 함유의 경구용 서방성 의약 조성물
US11590228B1 (en) 2015-09-08 2023-02-28 Tris Pharma, Inc Extended release amphetamine compositions
CR20190142A (es) * 2016-09-07 2019-05-22 Saniona As Composiciones de tesofensina
US12458592B1 (en) 2017-09-24 2025-11-04 Tris Pharma, Inc. Extended release amphetamine tablets
US11590081B1 (en) 2017-09-24 2023-02-28 Tris Pharma, Inc Extended release amphetamine tablets
US11918689B1 (en) 2020-07-28 2024-03-05 Tris Pharma Inc Liquid clonidine extended release composition

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JPH04235914A (ja) * 1991-01-18 1992-08-25 Kyowa Hakko Kogyo Co Ltd 徐放性製剤
JPH05262640A (ja) * 1991-11-13 1993-10-12 Glaxo Canada Inc 制御放出装置
JPH05339151A (ja) * 1992-05-30 1993-12-21 Kodama Kk 持効性塩酸オキシブチニン製剤
JPH10507210A (ja) * 1995-11-03 1998-07-14 エドワード メンデル カンパニー，インコーポレーテッド 放出制御製剤（アルブテロール）
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Also Published As

Publication number Publication date
US20080107730A1 (en) 2008-05-08
RU2004133532A (ru) 2005-06-10
CA2481667A1 (en) 2003-10-23
AU2003218397A1 (en) 2003-10-27
US20060105037A1 (en) 2006-05-18
EP1494653A1 (en) 2005-01-12
WO2003086364A1 (en) 2003-10-23
PL373328A1 (en) 2005-08-22
CN1655765A (zh) 2005-08-17
US20030198670A1 (en) 2003-10-23
US7125563B2 (en) 2006-10-24
HRP20040945A2 (en) 2005-02-28

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