JP2005531526A5 - - Google Patents
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- Publication number
- JP2005531526A5 JP2005531526A5 JP2003580307A JP2003580307A JP2005531526A5 JP 2005531526 A5 JP2005531526 A5 JP 2005531526A5 JP 2003580307 A JP2003580307 A JP 2003580307A JP 2003580307 A JP2003580307 A JP 2003580307A JP 2005531526 A5 JP2005531526 A5 JP 2005531526A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- formula
- compound
- alkyl
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 CCCCC1=SC(N(*)N=C)=C(*)*1 Chemical compound CCCCC1=SC(N(*)N=C)=C(*)*1 0.000 description 2
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02290788A EP1348701A1 (en) | 2002-03-28 | 2002-03-28 | (2,4-disubstituted-thiazol-5-yl) amine compounds as PDE7 inhibitors |
| PCT/EP2003/002287 WO2003082839A1 (en) | 2002-03-28 | 2003-03-06 | (4,2-disubstituted-thiazol-5-yl)amine compounds as pde7 inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005531526A JP2005531526A (ja) | 2005-10-20 |
| JP2005531526A5 true JP2005531526A5 (enExample) | 2006-04-20 |
Family
ID=27798934
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003580307A Withdrawn JP2005531526A (ja) | 2002-03-28 | 2003-03-06 | Ｐｄｅ７阻害剤としての（４，２−２置換−チアゾール−５−イル）アミン化合物 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US6753340B2 (enExample) |
| EP (2) | EP1348701A1 (enExample) |
| JP (1) | JP2005531526A (enExample) |
| AU (1) | AU2003212310A1 (enExample) |
| BR (1) | BR0308765A (enExample) |
| CA (1) | CA2480679A1 (enExample) |
| MX (1) | MXPA04009476A (enExample) |
| WO (1) | WO2003082839A1 (enExample) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003282087A1 (en) * | 2002-11-13 | 2004-06-03 | Bayer Healthcare Ag | DIAGNOSTICS AND THERAPEUTICS FOR DISEASES ASSOCIATED WITH HUMAN PHOSPHODIESTERASE 7A1 (PDE7a1) |
| ES2217956B1 (es) * | 2003-01-23 | 2006-04-01 | Almirall Prodesfarma, S.A. | Nuevos derivados de 4-aminotieno(2,3-d)pirimidin-6-carbonitrilo. |
| AP2006003700A0 (en) | 2004-02-13 | 2006-08-31 | Warner Lambert Co | Androgen receptor modulators |
| WO2005100305A1 (en) | 2004-04-13 | 2005-10-27 | Warner-Lambert Company Llc | Androgen modulators |
| CA2562672C (en) | 2004-04-22 | 2009-09-29 | Warner-Lambert Company Llc | 4-cyano-phenoxy derivatives as androgen modulators |
| TW200724139A (en) | 2005-05-05 | 2007-07-01 | Warner Lambert Co | Androgen modulators |
| EP1956906A4 (en) | 2005-11-09 | 2009-12-30 | Combinatorx Inc | METHODS, COMPOSITIONS AND KITS FOR THE TREATMENT OF PATHOLOGIES |
| GB0701426D0 (en) * | 2007-01-25 | 2007-03-07 | Univ Sheffield | Compounds and their use |
| AU2008230710B2 (en) * | 2007-03-27 | 2014-04-10 | Omeros Corporation | The use of PDE7 inhibitors for the treatment of movement disorders |
| US8637528B2 (en) | 2007-03-27 | 2014-01-28 | Omeros Corporation | Use of PDE7 inhibitors for the treatment of movement disorders |
| FR2943673B1 (fr) | 2009-03-27 | 2013-03-29 | Sanofi Aventis | Applications therapeutiques de derives de quinazolinedione |
| US9220715B2 (en) | 2010-11-08 | 2015-12-29 | Omeros Corporation | Treatment of addiction and impulse-control disorders using PDE7 inhibitors |
| KR20230104760A (ko) | 2010-11-08 | 2023-07-10 | 오메로스 코포레이션 | Pde7 억제제를 사용한 중독 및 충동-조절 장애의 치료 |
| US20130184280A1 (en) * | 2011-12-21 | 2013-07-18 | Telik, Inc. | Substituted thiazoles as vegfr2 kinase inhibitors |
| CN109689649B (zh) | 2016-07-14 | 2022-07-19 | 百时美施贵宝公司 | 经二环杂芳基取代的化合物 |
| ES2823127T3 (es) | 2016-07-14 | 2021-05-06 | Bristol Myers Squibb Co | Compuestos tricíclicos de quinolina y azaquinolina sustituidos con heteroarilo como inhibidores de PAR4 |
| JP7058256B2 (ja) | 2016-07-14 | 2022-04-21 | ブリストル－マイヤーズ スクイブ カンパニー | 二環式ヘテロアリール置換化合物 |
| US11987981B2 (en) | 2016-07-28 | 2024-05-21 | Carboshield, Inc. | Structural element reinforcement systems and methods |
| US12195987B2 (en) | 2016-07-28 | 2025-01-14 | Carboshield, Inc. | Structural element reinforcement systems and methods |
| CA3264513A1 (en) | 2022-08-18 | 2024-02-22 | Mitodicure Gmbh | USE OF SUBSTITUTED BENZOFURAN AND BENZOXAZOLE COMPOUNDS FOR THE TREATMENT AND PREVENTION OF DISEASES ASSOCIATED WITH CHRONIC FATIGUE, EXHAUSTION AND/OR EXERCISE INTOLERANCE |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH10504542A (ja) * | 1994-07-27 | 1998-05-06 | ジー．ディー．サール アンド カンパニー | 炎症処置用の置換チアゾール化合物 |
| AU4298997A (en) * | 1996-08-26 | 1998-03-19 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Thiazole derivatives useful as selective inhibitors of pde-iv |
| US6313156B1 (en) * | 1999-12-23 | 2001-11-06 | Icos Corporation | Thiazole compounds as cyclic-AMP-specific phosphodiesterase inhibitors |
| ATE414079T1 (de) * | 2000-03-01 | 2008-11-15 | Janssen Pharmaceutica Nv | 2,4-disubstituierte thiazolyl derivate |
-
2002
- 2002-03-28 EP EP02290788A patent/EP1348701A1/en not_active Withdrawn
-
2003
- 2003-03-06 BR BR0308765-4A patent/BR0308765A/pt not_active IP Right Cessation
- 2003-03-06 EP EP03708184A patent/EP1492778A1/en not_active Withdrawn
- 2003-03-06 CA CA002480679A patent/CA2480679A1/en not_active Abandoned
- 2003-03-06 AU AU2003212310A patent/AU2003212310A1/en not_active Abandoned
- 2003-03-06 WO PCT/EP2003/002287 patent/WO2003082839A1/en not_active Ceased
- 2003-03-06 JP JP2003580307A patent/JP2005531526A/ja not_active Withdrawn
- 2003-03-06 MX MXPA04009476A patent/MXPA04009476A/es active IP Right Grant
- 2003-03-27 US US10/401,392 patent/US6753340B2/en not_active Expired - Fee Related
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