JP2006503857A5 - - Google Patents

Download PDF

Info

Publication number
JP2006503857A5
JP2006503857A5 JP2004540809A JP2004540809A JP2006503857A5 JP 2006503857 A5 JP2006503857 A5 JP 2006503857A5 JP 2004540809 A JP2004540809 A JP 2004540809A JP 2004540809 A JP2004540809 A JP 2004540809A JP 2006503857 A5 JP2006503857 A5 JP 2006503857A5
Authority
JP
Japan
Prior art keywords
piperazine
amide
ethyl
sulfonyl
thiophen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2004540809A
Other languages
English (en)
Japanese (ja)
Other versions
JP4713152B2 (ja
JP2006503857A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2003/050640 external-priority patent/WO2004031182A1/en
Publication of JP2006503857A publication Critical patent/JP2006503857A/ja
Publication of JP2006503857A5 publication Critical patent/JP2006503857A5/ja
Application granted granted Critical
Publication of JP4713152B2 publication Critical patent/JP4713152B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2004540809A 2002-09-20 2003-09-19 ピペラジン誘導体及び使用方法 Expired - Fee Related JP4713152B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US41230802P 2002-09-20 2002-09-20
US60/412,308 2002-09-20
PCT/EP2003/050640 WO2004031182A1 (en) 2002-09-20 2003-09-19 Piperazine derivatives and methods of use

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2011000050A Division JP5436462B2 (ja) 2002-09-20 2011-01-04 ピペラジン誘導体及び使用方法

Publications (3)

Publication Number Publication Date
JP2006503857A JP2006503857A (ja) 2006-02-02
JP2006503857A5 true JP2006503857A5 (enExample) 2010-08-05
JP4713152B2 JP4713152B2 (ja) 2011-06-29

Family

ID=32069711

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2004540809A Expired - Fee Related JP4713152B2 (ja) 2002-09-20 2003-09-19 ピペラジン誘導体及び使用方法
JP2011000050A Expired - Fee Related JP5436462B2 (ja) 2002-09-20 2011-01-04 ピペラジン誘導体及び使用方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2011000050A Expired - Fee Related JP5436462B2 (ja) 2002-09-20 2011-01-04 ピペラジン誘導体及び使用方法

Country Status (8)

Country Link
US (3) US7754722B2 (enExample)
EP (1) EP1542993B1 (enExample)
JP (2) JP4713152B2 (enExample)
AU (1) AU2003299124A1 (enExample)
CA (1) CA2499732A1 (enExample)
ES (1) ES2399047T3 (enExample)
NO (1) NO20051844L (enExample)
WO (1) WO2004031182A1 (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1592389B1 (en) 2003-02-14 2009-04-22 Laboratoires Serono SA Piperazine-2-carboxamide derivatives
US8017612B2 (en) 2006-04-18 2011-09-13 Japan Tobacco Inc. Piperazine compound and use thereof as a HCV polymerase inhibitor
TW200944523A (en) * 2008-02-08 2009-11-01 Organon Nv (Dihydro)pyrrolo[2,1-a]isoquinolines
US8071587B2 (en) 2009-05-27 2011-12-06 N. V. Organon (Dihydro)imidazoiso[5,1-A]quinolines
TW201116531A (en) 2009-07-29 2011-05-16 Organon Nv Ring-annulated dihydropyrrolo[2,1-a]isoquinolines
US8431564B2 (en) 2009-07-29 2013-04-30 Merck Sharp & Dohme B.V. Ring-annulated dihydropyrrolo[2,1-α]isoquinolines
TW201116515A (en) 2009-07-31 2011-05-16 Organon Nv Dihydrobenzoindazoles
CA2801074A1 (en) 2010-06-04 2011-12-08 Albany Molecular Research, Inc. Glycine transporter-1 inhibitors, methods of making them, and uses thereof
JP6162694B2 (ja) * 2011-07-18 2017-07-12 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングＭｅｒｃｋ Ｐａｔｅｎｔ Ｇｅｓｅｌｌｓｃｈａｆｔ ｍｉｔ ｂｅｓｃｈｒａｅｎｋｔｅｒ Ｈａｆｔｕｎｇ ベンズアミド類
AR095202A1 (es) * 2013-03-11 2015-09-30 Merck Patent Gmbh Heterociclos como moduladores de la actividad quinasa
KR20170054650A (ko) * 2015-11-10 2017-05-18 삼성전자주식회사 이동 정보에 기초하여 심박수를 추정하는 방법 및 장치
US10688224B1 (en) 2019-07-03 2020-06-23 King Abdulaziz University Prosthetic implantable antibacterial surgical mesh

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5639639A (en) * 1983-11-02 1997-06-17 Genzyme Corporation Recombinant heterodimeric human fertility hormones, and methods, cells, vectors and DNA for the production thereof
IT1206302B (it) * 1987-06-26 1989-04-14 Serono Cesare Ist Ricerca Ormone follicolo-stimolante urinario
US5017557A (en) * 1987-07-24 1991-05-21 Industria Farmaceutica Serono S.P.A. Treatment of infertility with somatotrophin releasing factor
IL117798A (en) * 1995-04-07 2001-11-25 Schering Plough Corp Tricyclic compounds useful for inhibiting the function of protein - G and for the treatment of malignant diseases, and pharmaceutical preparations containing them
US5880128A (en) * 1996-05-08 1999-03-09 Schering Corporation Carbonyl piperazinyl and piperidinyl compounds
ES2224408T3 (es) 1997-06-17 2005-03-01 Schering Corporation Compuestos de benzopiridocicloheptano utiles para la inhibicion de la farnesil-proteina-transferasa.
ES2221227T3 (es) 1997-11-24 2004-12-16 MERCK & CO., INC. Derivados sustituidos de beta-alanina como inhibidores de la adhesion celular.
PT1102763E (pt) 1998-08-07 2005-01-31 Applied Research Systems Mimeticos fsh para o tratamento da infertilidade
US6432959B1 (en) * 1998-12-23 2002-08-13 Schering Corporation Inhibitors of farnesyl-protein transferase
ES2242444T3 (es) * 1998-12-23 2005-11-01 Schering Corporation Nuevos inhibidores de la farnesil-proteina-transferasa.
US6426357B1 (en) * 1999-07-27 2002-07-30 Affymax, Inc. Antagonists of follicle stimulating hormone activity
JP2001294572A (ja) 2000-02-09 2001-10-23 Dai Ichi Seiyaku Co Ltd 新規スルホニル誘導体
WO2002009706A1 (en) 2000-07-27 2002-02-07 Smithkline Beecham Corporation Agonists of follicle stimulating hormone activity
EP1592389B1 (en) * 2003-02-14 2009-04-22 Laboratoires Serono SA Piperazine-2-carboxamide derivatives

Similar Documents

Publication Publication Date Title
ES2795366T3 (es) Compuestos de indol carboxamida útiles como inhibidores de cinasas
ES2316784T3 (es) Derivados de 2-hidroxi-3-heteroarilindol como inhibidores de gsk3.
JP6193922B2 (ja) ハロアルキルヘテロアリールベンズアミド化合物
RU2386620C2 (ru) Производные пиридазин-3(2н)-она и их применение в качестве ингибиторов фдэ4
EA200500304A1 (ru) Производные 3-(сульфонамидоэтил)индола, предназначенные для использования в качестве миметиков глюкокортикоидов при лечении воспалительных, аллергических и пролиферативных заболеваний
JP5436462B2 (ja) ピペラジン誘導体及び使用方法
JP2008513498A5 (enExample)
JP2006503857A5 (enExample)
JP2007511467A (ja) ジペプチジルペプチダーゼインヒビター
NO20061766L (no) 1,1,1-trifluor-4-fenyl-4-metyl-2-(1H-Pyrrolo'2,3-Cl Pyridin-2-ylmetyl)pentan-2-ol derivater og beslektede forbindelser som glukokortikoidligander for behandling av inflammatoriske sykdommer og diabetes
AR054127A1 (es) Imidazoquinolinas como inhibidores de quinasa de lipido
CA2485850A1 (en) 8-azaprostaglandin analogs as agents for lowering intraocular pressure
UY29389A1 (es) Derivados sustituidos del ácido1-((4-((((3,3-dimetil-2-oxo-2,3-dihidro-1h-indol-1-il)carbonil)amino)metil)piperidin-1-il)metil)ciclobutanocarboxílico, sales farmaceuticamente aceptables, composiciones que los contienen y aplicaciones.
KR20200038473A (ko) 히스톤 데아세틸라제 1 및 2 (hdac1-2)의 선택적인 저해제로서 새로운 헤테로아릴 아미드 유도체
AU2015241022A1 (en) Inhibitors of histone demethylases
JP2012507525A5 (enExample)
RU2007122485A (ru) Ингибиторы киназы
JP2005531526A5 (enExample)
JP2004525183A5 (enExample)
JP6434528B2 (ja) 置換ピリドン及びピラジノン、並びに好中球エラスターゼ活性の阻害剤としてのその使用
JP2005527521A5 (enExample)
US6245768B1 (en) 1-(N′-(arylalkylaminoalkyl)) aminoisoindoles; a new class of dopamine receptor subtype specific ligands
JP6713000B2 (ja) 抗腫瘍活性を有する化合物
US5591866A (en) (1H-indol-1-yl)-2-(amino)acetamide derivatives and preparation thereof
RU2007128080A (ru) Производные пирролидиния в качестве мускариновых рецепторов мз