JP2005528459A5 - - Google Patents
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- Publication number
- JP2005528459A5 JP2005528459A5 JP2004511291A JP2004511291A JP2005528459A5 JP 2005528459 A5 JP2005528459 A5 JP 2005528459A5 JP 2004511291 A JP2004511291 A JP 2004511291A JP 2004511291 A JP2004511291 A JP 2004511291A JP 2005528459 A5 JP2005528459 A5 JP 2005528459A5
- Authority
- JP
- Japan
- Prior art keywords
- amino
- het
- methyl
- independently
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02012590A EP1369420A1 (en) | 2002-06-06 | 2002-06-06 | Inhibitors of the GPib - vWF interaction |
| PCT/EP2003/005955 WO2003104221A1 (en) | 2002-06-06 | 2003-06-06 | Inhibitors of the gpib -vwf interaction, their preparation and use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005528459A JP2005528459A (ja) | 2005-09-22 |
| JP2005528459A5 true JP2005528459A5 (https=) | 2006-04-06 |
| JP4455326B2 JP4455326B2 (ja) | 2010-04-21 |
Family
ID=29433122
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004511291A Expired - Fee Related JP4455326B2 (ja) | 2002-06-06 | 2003-06-06 | ＧＰＩｂ−ｖＷＦ相互作用の阻害薬、それらの製造および使用 |
Country Status (9)
| Country | Link |
|---|---|
| EP (2) | EP1369420A1 (https=) |
| JP (1) | JP4455326B2 (https=) |
| AT (1) | ATE353082T1 (https=) |
| AU (1) | AU2003274686A1 (https=) |
| BR (1) | BR0311826A (https=) |
| CA (1) | CA2488193A1 (https=) |
| DE (1) | DE60311578T2 (https=) |
| MX (1) | MXPA04011408A (https=) |
| WO (1) | WO2003104221A1 (https=) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004080950A1 (en) * | 2003-03-14 | 2004-09-23 | H. Lundbeck A/S | Substituted aniline derivatives |
| AR043507A1 (es) * | 2003-03-14 | 2005-08-03 | Lundbeck & Co As H | Derivados de anilina sustituidos y composiciones farmaceuticas |
| WO2005033079A1 (ja) | 2003-09-30 | 2005-04-14 | Eisai Co., Ltd. | ヘテロ環化合物を含有する新規な抗真菌剤 |
| WO2006016548A1 (ja) * | 2004-08-09 | 2006-02-16 | Eisai R & D Management Co., Ltd. | ヘテロ環化合物を含有する新規な抗マラリア剤 |
| JP4874958B2 (ja) | 2005-03-30 | 2012-02-15 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ピリジン誘導体を含有する抗真菌剤 |
| TWI385169B (zh) | 2005-10-31 | 2013-02-11 | Eisai R&D Man Co Ltd | 經雜環取代之吡啶衍生物及含有彼之抗真菌劑 |
| EP2065377B1 (en) | 2006-09-21 | 2011-11-23 | Eisai R&D Management Co., Ltd. | Pyridine derivative substituted by heteroaryl ring, and antifungal agent comprising the same |
| TW200841879A (en) | 2007-04-27 | 2008-11-01 | Eisai R&D Man Co Ltd | Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same |
| WO2008136279A1 (ja) | 2007-04-27 | 2008-11-13 | Eisai R & D Management Co., Ltd. | ヘテロ環置換ピリジン誘導体の塩またはその結晶 |
| EP3103791B1 (en) | 2007-06-27 | 2018-01-31 | Merck Sharp & Dohme Corp. | 4-carboxybenzylamino derivatives as histone deacetylase inhibitors |
| WO2009005638A2 (en) | 2007-06-27 | 2009-01-08 | Merck & Co., Inc. | Pyridyl and pyrimidinyl derivatives as histone deacetylase inhibitors |
| US8513287B2 (en) | 2007-12-27 | 2013-08-20 | Eisai R&D Management Co., Ltd. | Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same |
| US8188119B2 (en) | 2008-10-24 | 2012-05-29 | Eisai R&D Management Co., Ltd | Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same |
| EP2627324A4 (en) * | 2010-10-11 | 2014-05-07 | Univ Leland Stanford Junior | SUBSTITUTED BENZAMIDES AND USES THEREOF |
| US9296732B2 (en) | 2012-04-12 | 2016-03-29 | The Board Of Trustees Of The Leland Stanford Junior University | Substituted benzamides and their uses |
| JP2023078557A (ja) * | 2021-11-26 | 2023-06-07 | 学校法人東海大学 | フォンヴィルブランド因子と血小板との結合を阻害するための医薬組成物 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW301607B (https=) * | 1993-03-09 | 1997-04-01 | Takeda Pharm Industry Co Ltd | |
| AU5812498A (en) * | 1996-12-20 | 1998-07-17 | Merck & Co., Inc. | Substituted aminoquinolines as modulators of chemokine receptor activity |
| US5919776A (en) * | 1996-12-20 | 1999-07-06 | Merck & Co., Inc. | Substituted aminoquinolines as modulators of chemokine receptor activity |
-
2002
- 2002-06-06 EP EP02012590A patent/EP1369420A1/en not_active Withdrawn
-
2003
- 2003-06-06 EP EP03740199A patent/EP1509516B1/en not_active Expired - Lifetime
- 2003-06-06 DE DE60311578T patent/DE60311578T2/de not_active Expired - Lifetime
- 2003-06-06 MX MXPA04011408A patent/MXPA04011408A/es unknown
- 2003-06-06 AT AT03740199T patent/ATE353082T1/de not_active IP Right Cessation
- 2003-06-06 CA CA002488193A patent/CA2488193A1/en not_active Abandoned
- 2003-06-06 JP JP2004511291A patent/JP4455326B2/ja not_active Expired - Fee Related
- 2003-06-06 AU AU2003274686A patent/AU2003274686A1/en not_active Abandoned
- 2003-06-06 BR BR0311826-6A patent/BR0311826A/pt not_active IP Right Cessation
- 2003-06-06 WO PCT/EP2003/005955 patent/WO2003104221A1/en not_active Ceased
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