JP2005526813A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2005526813A5 JP2005526813A5 JP2003580313A JP2003580313A JP2005526813A5 JP 2005526813 A5 JP2005526813 A5 JP 2005526813A5 JP 2003580313 A JP2003580313 A JP 2003580313A JP 2003580313 A JP2003580313 A JP 2003580313A JP 2005526813 A5 JP2005526813 A5 JP 2005526813A5
- Authority
- JP
- Japan
- Prior art keywords
- hydrogen
- group
- independently
- heteroarylalkyl
- heteroalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 229910052739 hydrogen Inorganic materials 0.000 claims 22
- 239000001257 hydrogen Substances 0.000 claims 21
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 12
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 9
- 125000003342 alkenyl group Chemical group 0.000 claims 9
- 125000000304 alkynyl group Chemical group 0.000 claims 9
- 125000003710 aryl alkyl group Chemical group 0.000 claims 9
- 125000003118 aryl group Chemical group 0.000 claims 9
- 125000004404 heteroalkyl group Chemical group 0.000 claims 9
- 125000001072 heteroaryl group Chemical group 0.000 claims 9
- 125000004446 heteroarylalkyl group Chemical group 0.000 claims 9
- 125000000837 carbohydrate group Chemical group 0.000 claims 6
- 125000000217 alkyl group Chemical group 0.000 claims 4
- 125000004429 atom Chemical group 0.000 claims 4
- 125000002252 acyl group Chemical group 0.000 claims 3
- 125000005251 aryl acyl group Chemical group 0.000 claims 3
- 150000003999 cyclitols Chemical group 0.000 claims 3
- 125000005253 heteroarylacyl group Chemical group 0.000 claims 3
- 229910052757 nitrogen Inorganic materials 0.000 claims 3
- 125000001424 substituent group Chemical group 0.000 claims 3
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 2
- CURLTUGMZLYLDI-UHFFFAOYSA-N Carbon dioxide Chemical compound O=C=O CURLTUGMZLYLDI-UHFFFAOYSA-N 0.000 claims 2
- 125000005001 aminoaryl group Chemical group 0.000 claims 2
- 150000001875 compounds Chemical class 0.000 claims 2
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 2
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 150000001413 amino acids Chemical class 0.000 claims 1
- 125000004103 aminoalkyl group Chemical group 0.000 claims 1
- 125000005214 aminoheteroaryl group Chemical group 0.000 claims 1
- 125000004104 aryloxy group Chemical group 0.000 claims 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 1
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims 1
- -1 heteroalkynyl Chemical group 0.000 claims 1
- 125000005553 heteroaryloxy group Chemical group 0.000 claims 1
- 150000002431 hydrogen Chemical class 0.000 claims 1
- 150000002825 nitriles Chemical class 0.000 claims 1
- 239000001301 oxygen Substances 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 108090000765 processed proteins & peptides Proteins 0.000 claims 1
- 125000004001 thioalkyl group Chemical group 0.000 claims 1
- 125000005000 thioaryl group Chemical group 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AUPS1434A AUPS143402A0 (en) | 2002-03-28 | 2002-03-28 | Anomeric derivatives of monosaccharides |
| AUPS1434 | 2002-03-28 | ||
| PCT/AU2003/000384 WO2003082846A1 (en) | 2002-03-28 | 2003-03-28 | Anomeric derivatives of monosaccharides |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005526813A JP2005526813A (ja) | 2005-09-08 |
| JP2005526813A5 true JP2005526813A5 (enExample) | 2006-03-16 |
| JP4610197B2 JP4610197B2 (ja) | 2011-01-12 |
Family
ID=3835023
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003580313A Expired - Fee Related JP4610197B2 (ja) | 2002-03-28 | 2003-03-28 | 単糖のアノマー誘導体 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US7737287B2 (enExample) |
| EP (1) | EP1487812A4 (enExample) |
| JP (1) | JP4610197B2 (enExample) |
| CN (1) | CN100537556C (enExample) |
| AU (1) | AUPS143402A0 (enExample) |
| CA (1) | CA2480578C (enExample) |
| DE (1) | DE03745223T1 (enExample) |
| WO (1) | WO2003082846A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7138531B2 (en) | 2001-10-15 | 2006-11-21 | Kemin Pharma B.V.B.A. | Preparation and use of carbohydrate-based bicyclic ring structures with antimicrobial and cytostatic activity |
| AU2002950657A0 (en) | 2002-08-08 | 2002-09-12 | Alchemia Limited | Derivatives of monosaccharides for drug discovery |
| AU2002951995A0 (en) | 2002-10-11 | 2002-10-31 | Alchemia Limited | Classes of compounds that interact with gpcrs |
| CN100347184C (zh) | 2003-01-07 | 2007-11-07 | 凯敏制药欧洲股份有限公司 | 可用于治疗由黄病毒科病毒如丙型肝炎及牛病毒性腹泻病毒引起的感染的双环糖类化合物 |
| WO2004062590A2 (en) | 2003-01-07 | 2004-07-29 | Kemin Pharma Europe B.V.B.A. | Bicyclic carbohydrates as antiprotozoal bioactive for the treatment of infections caused by parasites |
| US7368475B2 (en) | 2003-03-12 | 2008-05-06 | Kemin Pharma Bvba | Furanose-type bicyclic carbohydrates with biological activity |
| US7098243B2 (en) | 2003-09-16 | 2006-08-29 | Kemin Pharma Europe B.V.B.A. | Bicyclic carbohydrates as antiviral bioactives for the treatment of infections caused by the alphaherpesvirinae HSV-1 and HSV-2 |
| US20080176936A1 (en) * | 2005-02-04 | 2008-07-24 | Wim Meutermans | Classes of Compounds that Interact with Integrins |
| AU2006209794B2 (en) * | 2005-02-04 | 2010-07-08 | Alchemia Limited | Classes of compounds that interact with integrins |
| ES2400509T3 (es) * | 2005-10-04 | 2013-04-10 | Alchemia Ltd | Método de diseño de fármacos |
| WO2007070947A1 (en) * | 2005-12-22 | 2007-06-28 | Alchemia Ltd | Antibacterial agents |
| AU2021213822A1 (en) | 2020-01-31 | 2022-09-22 | Avilar Therapeutics, Inc. | ASGPR-binding compounds for the degradation of extracellular proteins |
| TW202308703A (zh) | 2021-05-03 | 2023-03-01 | 美商亞維拉治療公司 | 用於降解免疫球蛋白及其他蛋白質之有效asgpr結合化合物 |
| WO2024118503A1 (en) | 2022-11-28 | 2024-06-06 | Hongene Biotech Corporation | Functionalized n-acetylgalactosamine analogs |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5331664A (en) * | 1976-09-02 | 1978-03-25 | Suami T | Production of novel nitroso urea derivatives |
| DE3347522A1 (de) * | 1983-12-30 | 1985-07-11 | Troponwerke GmbH & Co KG, 5000 Köln | N-glycosylierte carbonsaeureamid-derivate als mittel bei der bekaempfung von erkrankungen des rheumatischen formenkreises |
| DE3521994A1 (de) * | 1985-06-20 | 1987-01-02 | Bayer Ag | N-(2-aminoacylamido-2-desoxy-hexosyl)-amide-, -carbamate und -harnstoffe, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln |
| HU208146B (en) * | 1989-11-14 | 1993-08-30 | Biogal Gyogyszergyar | Process for producing aminobenzoic acid-n-glycoside derivatives |
| US5449785A (en) * | 1991-07-24 | 1995-09-12 | Hoffmann-La Roche Inc. | Cyclohexane derivatives |
| JPH07242684A (ja) * | 1994-03-02 | 1995-09-19 | Japan Tobacco Inc | 新規なグルクロン酸化合物 |
| US5491152A (en) * | 1994-03-23 | 1996-02-13 | The Du Pont Merck Pharmaceutical Company | Derivatives of cyclic ethers and sulfides for the treatment of atherosclerosis |
| AU7286696A (en) * | 1995-10-13 | 1997-05-07 | F. Hoffmann-La Roche Ag | Antisense oligomers |
| AUPO190596A0 (en) * | 1996-08-26 | 1996-09-19 | Alchemia Pty Ltd | Oligosaccharide synthesis |
| EP0998280A4 (en) * | 1997-05-29 | 2002-11-06 | Incara Pharmaceuticals Corp | CARBOHYDRATE COMPOUNDS WITH SCAFFOLDING STRUCTURE AND BANKS CONTAINING SAME |
| US6197963B1 (en) * | 1998-08-13 | 2001-03-06 | The Trustees Of The University Of Pennsylvania | Non-peptide peptidomimetics |
| CA2415368A1 (en) * | 2000-07-13 | 2002-01-31 | Yi Jin | Synthesis and antiviral evaluation of nucleic acid based (nab) libraries |
| AUPR079700A0 (en) * | 2000-10-17 | 2000-11-09 | Alchemia Pty Ltd | Combinatorial libraries of monosaccharides |
| AUPR084400A0 (en) * | 2000-10-18 | 2000-11-09 | Alchemia Pty Ltd | Immunoadjuvant systems |
-
2002
- 2002-03-28 AU AUPS1434A patent/AUPS143402A0/en not_active Abandoned
-
2003
- 2003-03-28 CA CA2480578A patent/CA2480578C/en not_active Expired - Lifetime
- 2003-03-28 JP JP2003580313A patent/JP4610197B2/ja not_active Expired - Fee Related
- 2003-03-28 DE DE03745223T patent/DE03745223T1/de active Pending
- 2003-03-28 US US10/509,092 patent/US7737287B2/en active Active
- 2003-03-28 CN CNB038073757A patent/CN100537556C/zh not_active Expired - Lifetime
- 2003-03-28 EP EP03745223A patent/EP1487812A4/en not_active Withdrawn
- 2003-03-28 WO PCT/AU2003/000384 patent/WO2003082846A1/en not_active Ceased
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2005526813A5 (enExample) | ||
| CA2389681A1 (en) | Npy y5 antagonist | |
| JP2005532287A5 (enExample) | ||
| HUP0500457A2 (hu) | Polialkilén polimervegyületek, ilyeneket tartalmazó készítmények és azok alkalmazása | |
| HUP0401729A2 (hu) | IV típusú foszfodiészteráz inhibitor hatású alkin-aril-naftiridin-4(1H)-on-származékok és ezeket tartalmazó gyógyszerkészítmények | |
| HUP0302943A2 (hu) | Új heterociklusos vegyületek, előállításuk és alkalmazásuk gyógyszerekként, különösen antibakteriális szerekként | |
| CA2457054A1 (en) | Activator of peroxisome proliferator-activated receptor .delta. | |
| TW200738682A (en) | Isoquinoline derivatives | |
| JP2008510828A5 (enExample) | ||
| JP2005502621A5 (enExample) | ||
| JP2009500423A5 (enExample) | ||
| MY134582A (en) | New fluorenecarboxylic acid esters, process for the manufacture thereof and use thereof as medicaments | |
| JP2008505157A5 (enExample) | ||
| HUP0002404A2 (hu) | Aminosavszármazékok, hatóanyagként ezeket tartalmazó gyógyszerkészítmények, eljárás előállításukra és alkalmazásuk | |
| JP2004532346A5 (enExample) | ||
| JP2011506490A5 (enExample) | ||
| JP2005536531A5 (enExample) | ||
| TW200616636A (en) | Novel compounds | |
| JPH10121091A5 (enExample) | ||
| JP2005529910A5 (enExample) | ||
| HUP0204501A2 (hu) | Gyűrűs vegyületek, ezeket tartalmazó gyógyászati készítmények, valamint eljárás a vegyületek előállítására és alkalmazásuk | |
| JP2007507472A5 (enExample) | ||
| NO20073736L (no) | Nye 3-fenylpropionsyrederivater for behandlingen av diabetes | |
| JP2003535868A5 (enExample) | ||
| CA2531484A1 (en) | Novel bioisosteres of actinonin |