JP2005519866A5 - - Google Patents

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Publication number
JP2005519866A5
JP2005519866A5 JP2003532466A JP2003532466A JP2005519866A5 JP 2005519866 A5 JP2005519866 A5 JP 2005519866A5 JP 2003532466 A JP2003532466 A JP 2003532466A JP 2003532466 A JP2003532466 A JP 2003532466A JP 2005519866 A5 JP2005519866 A5 JP 2005519866A5
Authority
JP
Japan
Prior art keywords
membered
ring
heterocyclic
aromatic ring
amidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003532466A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005519866A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2002/031769 external-priority patent/WO2003029216A1/en
Publication of JP2005519866A publication Critical patent/JP2005519866A/ja
Publication of JP2005519866A5 publication Critical patent/JP2005519866A5/ja
Pending legal-status Critical Current

Links

JP2003532466A 2001-10-03 2002-10-03 凝固カスケードの選択阻害に有用な６員複素環式化合物 Pending JP2005519866A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US32672101P 2001-10-03 2001-10-03
US33862301P 2001-10-24 2001-10-24
US33285701P 2001-11-06 2001-11-06
US35005201P 2001-11-07 2001-11-07
US33189101P 2001-11-21 2001-11-21
US33210701P 2001-11-21 2001-11-21
PCT/US2002/031769 WO2003029216A1 (en) 2001-10-03 2002-10-03 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade

Publications (2)

Publication Number Publication Date
JP2005519866A JP2005519866A (ja) 2005-07-07
JP2005519866A5 true JP2005519866A5 (https=) 2006-01-12

Family

ID=27559729

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003532466A Pending JP2005519866A (ja) 2001-10-03 2002-10-03 凝固カスケードの選択阻害に有用な６員複素環式化合物

Country Status (7)

Country Link
US (2) US6969715B2 (https=)
EP (1) EP1438292A1 (https=)
JP (1) JP2005519866A (https=)
BR (1) BR0213092A (https=)
CA (1) CA2462305A1 (https=)
MX (1) MXPA04003163A (https=)
WO (1) WO2003029216A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MD20140044A2 (ro) 2011-11-11 2014-08-31 Pfizer Inc. 2-Tiopirimidinone şi utilizarea lor pentru tratamentul afecţiunilor cardiovasculare
DK2785700T3 (en) 2011-11-29 2016-06-13 Perosphere Inc Agent for preventing the action of anti-coagulants.
AU2016257179A1 (en) 2015-05-05 2017-11-02 Pfizer Inc. 2-thiopyrimidinones
CN110117257B (zh) * 2018-02-05 2022-12-06 安徽省新星药物开发有限责任公司 一种含胍基的p2y12受体拮抗剂、制备方法及其用途

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