JP2005517741A - インシュリン及びｉｇｆ−１レセプターのアゴニスト及びアンタゴニスト - Google Patents

インシュリン及びｉｇｆ−１レセプターのアゴニスト及びアンタゴニスト Download PDF

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JP2005517741A
JP2005517741A JP2003569654A JP2003569654A JP2005517741A JP 2005517741 A JP2005517741 A JP 2005517741A JP 2003569654 A JP2003569654 A JP 2003569654A JP 2003569654 A JP2003569654 A JP 2003569654A JP 2005517741 A JP2005517741 A JP 2005517741A
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seq
sequence
amino acid
group
formula
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Japanese (ja)
Inventor
レヌーカ ピルートラ，
レニー ブリセット，
アーサー， ジェイ． ブルーム，
ラウゲ シェファー，
ヤコブ ブラント，
ニール， アイ． ゴールドスタイン，
ジェーン スペツラー，
ソーレン オステルガール，
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ノボ・ノルデイスク・エー／エス
ディージーアイ バイオテクノロジーズ
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/65—Insulin-like growth factors, i.e. somatomedins, e.g. IGF-1, IGF-2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/62—Insulins

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Toxicology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
JP2003569654A 2001-09-24 2002-09-24 インシュリン及びｉｇｆ−１レセプターのアゴニスト及びアンタゴニスト Pending JP2005517741A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/962,756 US6875741B2 (en) 1998-09-02 2001-09-24 Insulin and IGF-1 receptor agonists and antagonists
PCT/US2002/030312 WO2003070747A2 (en) 2001-09-24 2002-09-24 Insulin and igf-1 receptor agonists and antagonists

Publications (1)

Publication Number Publication Date
JP2005517741A true JP2005517741A (ja) 2005-06-16

Family

ID=25506313

Family Applications (2)

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JP2003530818A Pending JP2005505579A (ja) 2001-09-24 2002-09-24 アンタゴニスト
JP2003569654A Pending JP2005517741A (ja) 2001-09-24 2002-09-24 インシュリン及びｉｇｆ−１レセプターのアゴニスト及びアンタゴニスト

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2003530818A Pending JP2005505579A (ja) 2001-09-24 2002-09-24 アンタゴニスト

Country Status (6)

Country Link
US (1) US6875741B2 (cg-RX-API-DMAC7.html)
EP (2) EP1432433A4 (cg-RX-API-DMAC7.html)
JP (2) JP2005505579A (cg-RX-API-DMAC7.html)
AU (2) AU2002366384A1 (cg-RX-API-DMAC7.html)
CA (2) CA2459999A1 (cg-RX-API-DMAC7.html)
WO (2) WO2003027246A2 (cg-RX-API-DMAC7.html)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009511446A (ja) * 2005-10-05 2009-03-19 ノボ・ノルデイスク・エー／エス インスリンレセプターアンタゴニストと、関連した組成物、使用及び方法

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009511446A (ja) * 2005-10-05 2009-03-19 ノボ・ノルデイスク・エー／エス インスリンレセプターアンタゴニストと、関連した組成物、使用及び方法

Also Published As

Publication number Publication date
AU2002341834A1 (en) 2003-04-07
EP1496935A2 (en) 2005-01-19
EP1432433A2 (en) 2004-06-30
WO2003070747A3 (en) 2004-11-11
EP1432433A4 (en) 2006-08-30
CA2460055A1 (en) 2003-08-28
CA2459999A1 (en) 2003-04-03
WO2003027246A3 (en) 2003-07-31
WO2003027246A2 (en) 2003-04-03
US6875741B2 (en) 2005-04-05
US20030195147A1 (en) 2003-10-16
JP2005505579A (ja) 2005-02-24
AU2002366384A1 (en) 2003-09-09
AU2002366384A8 (en) 2003-09-09
EP1496935A4 (en) 2006-06-07
WO2003070747A2 (en) 2003-08-28

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