JP2005504101A5 - - Google Patents

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Publication number
JP2005504101A5
JP2005504101A5 JP2003530847A JP2003530847A JP2005504101A5 JP 2005504101 A5 JP2005504101 A5 JP 2005504101A5 JP 2003530847 A JP2003530847 A JP 2003530847A JP 2003530847 A JP2003530847 A JP 2003530847A JP 2005504101 A5 JP2005504101 A5 JP 2005504101A5
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JP
Japan
Prior art keywords
amino
triazole
anilino
pharmaceutical composition
phenylaminothiazol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003530847A
Other languages
English (en)
Japanese (ja)
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JP2005504101A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2002/030059 external-priority patent/WO2003027275A1/en
Publication of JP2005504101A publication Critical patent/JP2005504101A/ja
Publication of JP2005504101A5 publication Critical patent/JP2005504101A5/ja
Pending legal-status Critical Current

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JP2003530847A 2001-09-27 2002-09-23 緑内障を治療するためのグリコゲンシンターゼキナーゼ−３（ｇｓｋ−３）インヒビター Pending JP2005504101A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32539001P 2001-09-27 2001-09-27
PCT/US2002/030059 WO2003027275A1 (en) 2001-09-27 2002-09-23 Inhibitors of glycogen synthase kinase-3 (gsk-3) for treating glaucoma

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2005211956A Division JP2005320350A (ja) 2001-09-27 2005-07-21 緑内障を治療するためのグリコゲンシンターゼキナーゼ−３（ｇｓｋ−３）インヒビター

Publications (2)

Publication Number Publication Date
JP2005504101A JP2005504101A (ja) 2005-02-10
JP2005504101A5 true JP2005504101A5 (enExample) 2006-01-05

Family

ID=23267686

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2003530847A Pending JP2005504101A (ja) 2001-09-27 2002-09-23 緑内障を治療するためのグリコゲンシンターゼキナーゼ−３（ｇｓｋ−３）インヒビター
JP2005211956A Pending JP2005320350A (ja) 2001-09-27 2005-07-21 緑内障を治療するためのグリコゲンシンターゼキナーゼ−３（ｇｓｋ−３）インヒビター

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2005211956A Pending JP2005320350A (ja) 2001-09-27 2005-07-21 緑内障を治療するためのグリコゲンシンターゼキナーゼ−３（ｇｓｋ−３）インヒビター

Country Status (15)

Country Link
US (2) US7598288B2 (enExample)
EP (2) EP1430120A4 (enExample)
JP (2) JP2005504101A (enExample)
KR (1) KR20040047824A (enExample)
CN (2) CN101380319A (enExample)
AR (1) AR036684A1 (enExample)
AU (1) AU2002334635B2 (enExample)
BR (1) BR0212924A (enExample)
CA (1) CA2460000C (enExample)
MX (1) MXPA04002137A (enExample)
PL (1) PL207022B1 (enExample)
RU (1) RU2297243C2 (enExample)
TW (2) TWI335221B (enExample)
WO (1) WO2003027275A1 (enExample)
ZA (1) ZA200401846B (enExample)

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EP1616568A3 (en) * 2002-04-30 2006-06-21 Alcon, Inc GSK-3 inhibitors and CDK inhibitors as anti-glaucoma agents
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TW200526224A (en) * 2003-12-22 2005-08-16 Alcon Inc Short form c-Maf transcription factor antagonists for treatment of glaucoma
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US7872000B2 (en) 2006-12-29 2011-01-18 Rigel Pharmaceuticals, Inc. Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as Axl inhibitors
EP2484679B1 (en) 2006-12-29 2016-09-28 Rigel Pharmaceuticals, Inc. N3-heteroaryl substituted triazoles and n5-heteroaryl substitued triazoles useful as axl inhibitors
PT2114955E (pt) 2006-12-29 2013-04-18 Rigel Pharmaceuticals Inc Triazoles substituídos com arilo bicíclico em ponte ou heteroarilo bicíclico em ponte úteis como inibidores de axl
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WO2010005876A2 (en) 2008-07-09 2010-01-14 Rigel Pharmaceuticals, Inc. Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
PT2328888E (pt) 2008-07-09 2013-01-29 Rigel Pharmaceuticals Inc Triazóis bicíclicos em ponte substituídos com heteroarilos úteis como inibidores axl
US8546433B2 (en) 2009-01-16 2013-10-01 Rigel Pharmaceuticals, Inc. Axl inhibitors for use in combination therapy for preventing, treating or managing metastatic cancer
UA103918C2 (en) * 2009-03-02 2013-12-10 Айерем Элелси N-(hetero)aryl, 2-(hetero)aryl-substituted acetamides for use as wnt signaling modulators
RU2456266C1 (ru) * 2011-04-06 2012-07-20 Максим Эдуардович Запольский Производные 4,4'-бифениламидов, обладающие фармакологической активностью, и лекарственные средства на их основе
EP2975138A2 (en) 2013-03-15 2016-01-20 Fundació Institut de Recerca Biomèdica (IRB Barcelona) Method for the diagnosis, prognosis and treatment of cancer metastasis
EP3089748A4 (en) * 2014-01-02 2017-09-27 Massachusetts Eye & Ear Infirmary Treating ocular neovascularization
US20170165230A1 (en) 2014-04-09 2017-06-15 Christopher Rudd Use of gsk-3 inhibitors or activators which modulate pd-1 or t-bet expression to modulate t cell immunity
US11045352B2 (en) 2014-05-12 2021-06-29 Gholam A. Peyman Methods for treatment of dry eye and other acute or chronic inflammatory processes
US10925889B2 (en) 2014-05-12 2021-02-23 Gholam A. Peyman Method of treating, reducing, or alleviating a medical condition in a patient
US10583221B2 (en) 2014-05-12 2020-03-10 Gholam A. Peyman Method of corneal transplantation or corneal inlay implantation with cross-linking
US11666777B2 (en) 2014-05-12 2023-06-06 Gholam A. Peyman Photodynamic therapy technique for preventing damage to the fovea of the eye or another body portion of a patient
US10881503B2 (en) 2014-05-12 2021-01-05 Gholam A. Peyman Method of corneal transplantation or corneal inlay implantation with cross-linking
US11338059B2 (en) 2014-05-12 2022-05-24 Gholam A. Peyman Method of corneal and scleral inlay crosslinking and preservation
US12396889B2 (en) 2014-05-12 2025-08-26 Gholam A. Peyman Lamellar corneal autologous or homologous graft in refractive surgery
US11565023B2 (en) 2014-05-12 2023-01-31 Gholam A. Peyman Method of corneal transplantation or corneal inlay implantation with cross-linking
US11648261B2 (en) 2014-05-12 2023-05-16 Gholam A. Peyman Method of treating, reducing, or alleviating a medical condition in a patient
TWI744723B (zh) 2014-06-20 2021-11-01 美商基利科學股份有限公司 多環型胺甲醯基吡啶酮化合物之合成
WO2019221959A1 (en) * 2018-05-16 2019-11-21 Peyman Gholam A Method of treating, reducing, or alleviating a medical condition in a patient
US11707518B2 (en) 2019-04-28 2023-07-25 Gholam A. Peyman Method of treating, reducing, or alleviating a medical condition in a patient
US12226478B2 (en) 2019-04-28 2025-02-18 Gholam A. Peyman Method of treating, reducing, or alleviating a medical condition in a patient
US12110278B2 (en) * 2020-10-13 2024-10-08 Yale University Selective JAK2 pseudokinase ligands and methods of use

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