JP2004525873A5 - - Google Patents

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Publication number
JP2004525873A5
JP2004525873A5 JP2002551496A JP2002551496A JP2004525873A5 JP 2004525873 A5 JP2004525873 A5 JP 2004525873A5 JP 2002551496 A JP2002551496 A JP 2002551496A JP 2002551496 A JP2002551496 A JP 2002551496A JP 2004525873 A5 JP2004525873 A5 JP 2004525873A5
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JP
Japan
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alkyl
amino
mono
alkoxy
alkynyl
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JP2002551496A
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English (en)
Japanese (ja)
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JP5260818B2 (ja
JP2004525873A (ja
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Priority claimed from PCT/US2000/026816 external-priority patent/WO2002049993A2/en
Publication of JP2004525873A publication Critical patent/JP2004525873A/ja
Publication of JP2004525873A5 publication Critical patent/JP2004525873A5/ja
Application granted granted Critical
Publication of JP5260818B2 publication Critical patent/JP5260818B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2002551496A 2000-09-29 2000-09-29 高親和性低分子Ｃ５ａ受容体調節物質 Expired - Fee Related JP5260818B2 (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2000/026816 WO2002049993A2 (en) 2000-09-29 2000-09-29 High affinity small molecule c5a receptor modulators

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2011092825A Division JP2011219476A (ja) 2011-04-19 2011-04-19 高親和性低分子Ｃ５ａ受容体調節物質

Publications (3)

Publication Number Publication Date
JP2004525873A JP2004525873A (ja) 2004-08-26
JP2004525873A5 true JP2004525873A5 (https=) 2007-11-22
JP5260818B2 JP5260818B2 (ja) 2013-08-14

Family

ID=21741822

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002551496A Expired - Fee Related JP5260818B2 (ja) 2000-09-29 2000-09-29 高親和性低分子Ｃ５ａ受容体調節物質

Country Status (13)

Country Link
EP (1) EP1322309B1 (https=)
JP (1) JP5260818B2 (https=)
KR (1) KR20030060887A (https=)
CN (1) CN1454086A (https=)
AT (1) ATE404553T1 (https=)
AU (1) AU7622500A (https=)
BR (1) BR0017338A (https=)
DE (1) DE60039921D1 (https=)
IL (1) IL154993A0 (https=)
MX (1) MXPA03002788A (https=)
NO (1) NO20031370L (https=)
WO (1) WO2002049993A2 (https=)
YU (1) YU23503A (https=)

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JP2007284352A (ja) * 2004-08-05 2007-11-01 Dai Ichi Seiyaku Co Ltd ピラゾール誘導体
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EP1856126A2 (en) 2005-02-17 2007-11-21 Wyeth a Corporation of the State of Delaware Cycloalkylfused indole, benzothiophene, benzofuran and indene derivatives
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AU2017246228B2 (en) 2016-04-04 2021-04-15 Chemocentryx, Inc. Soluble C5aR antagonists
WO2018222601A1 (en) 2017-05-31 2018-12-06 Chemocentryx, Inc. 5-5 FUSED RINGS AS C5a INHIBITORS
CN110997674B (zh) 2017-05-31 2022-12-20 凯莫森特里克斯股份有限公司 作为C5a抑制剂的6-5稠合环类
KR20200109298A (ko) 2017-10-30 2020-09-22 케모센트릭스, 인크. 면역조절제로서의 중수소화된 화합물
MX2020006460A (es) 2017-12-22 2020-11-06 Chemocentryx Inc Compuestos de anillo 5,5 fusionado sustituido con diarilo como inhibidores de c5ar.
ES2980175T3 (es) 2017-12-22 2024-09-30 Chemocentryx Inc Compuestos anulares fusionados en 6,5 sustituidos con diarilo como inhibidores de C5aR
WO2019195159A1 (en) 2018-04-02 2019-10-10 Chemocentryx, Inc. PRODRUGS OF FUSED-BICYCLIC C5aR ANTAGONISTS
CN114957165A (zh) * 2021-02-26 2022-08-30 清华大学 一种抗病毒化合物及其制备方法和应用

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