JP2004525873A5 - - Google Patents

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Publication number
JP2004525873A5
JP2004525873A5 JP2002551496A JP2002551496A JP2004525873A5 JP 2004525873 A5 JP2004525873 A5 JP 2004525873A5 JP 2002551496 A JP2002551496 A JP 2002551496A JP 2002551496 A JP2002551496 A JP 2002551496A JP 2004525873 A5 JP2004525873 A5 JP 2004525873A5
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JP
Japan
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alkyl
amino
mono
alkoxy
alkynyl
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JP2002551496A
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English (en)
Japanese (ja)
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JP5260818B2 (ja
JP2004525873A (ja
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Priority claimed from PCT/US2000/026816 external-priority patent/WO2002049993A2/en
Publication of JP2004525873A publication Critical patent/JP2004525873A/ja
Publication of JP2004525873A5 publication Critical patent/JP2004525873A5/ja
Application granted granted Critical
Publication of JP5260818B2 publication Critical patent/JP5260818B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2002551496A 2000-09-29 2000-09-29 高親和性低分子Ｃ５ａ受容体調節物質 Expired - Fee Related JP5260818B2 (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2000/026816 WO2002049993A2 (en) 2000-09-29 2000-09-29 High affinity small molecule c5a receptor modulators

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2011092825A Division JP2011219476A (ja) 2011-04-19 2011-04-19 高親和性低分子Ｃ５ａ受容体調節物質

Publications (3)

Publication Number Publication Date
JP2004525873A JP2004525873A (ja) 2004-08-26
JP2004525873A5 true JP2004525873A5 (https=) 2007-11-22
JP5260818B2 JP5260818B2 (ja) 2013-08-14

Family

ID=21741822

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002551496A Expired - Fee Related JP5260818B2 (ja) 2000-09-29 2000-09-29 高親和性低分子Ｃ５ａ受容体調節物質

Country Status (13)

Country Link
EP (1) EP1322309B1 (https=)
JP (1) JP5260818B2 (https=)
KR (1) KR20030060887A (https=)
CN (1) CN1454086A (https=)
AT (1) ATE404553T1 (https=)
AU (1) AU7622500A (https=)
BR (1) BR0017338A (https=)
DE (1) DE60039921D1 (https=)
IL (1) IL154993A0 (https=)
MX (1) MXPA03002788A (https=)
NO (1) NO20031370L (https=)
WO (1) WO2002049993A2 (https=)
YU (1) YU23503A (https=)

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WO2006060424A2 (en) 2004-12-01 2006-06-08 Kalypsys, Inc. Inducible nitric oxide synthase dimerization inhibitors
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RS54998B1 (sr) 2008-12-22 2016-11-30 Chemocentryx Inc Antagonisti c5ar
RS56332B1 (sr) 2010-06-24 2017-12-29 Chemocentryx Inc Antagonisti c5ar
MX2015014688A (es) * 2013-04-22 2016-02-19 Abbvie Inc Tiazoles y usos de los mismos.
DK3200791T3 (da) 2014-09-29 2020-05-25 Chemocentryx Inc Fremgangsmåder og mellemprodukter i fremstilling af C5AR- antagonister
EP3072891A1 (en) * 2015-03-24 2016-09-28 Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. New Toll-Like Receptor 9 Antagonists
JP7339733B2 (ja) 2016-01-14 2023-09-06 ケモセントリックス，インコーポレイティド Ｃ３腎症を処置する方法
EP3439658B1 (en) 2016-04-04 2021-11-24 ChemoCentryx, Inc. Soluble c5ar antagonists
WO2018222601A1 (en) 2017-05-31 2018-12-06 Chemocentryx, Inc. 5-5 FUSED RINGS AS C5a INHIBITORS
US10562896B2 (en) 2017-05-31 2020-02-18 Chemocentryx, Inc. 6-5 fused rings as C5a inhibitors
CA3077395A1 (en) 2017-10-30 2019-05-09 Chemocentryx, Inc. Deuterated compounds as immunomodulators
WO2019126424A1 (en) 2017-12-22 2019-06-27 Chemocentryx, Inc. DIARYL SUBSTITUTED 6,5-FUSED RING COMPOUNDS AS C5aR INHIBITORS
MX2020006460A (es) 2017-12-22 2020-11-06 Chemocentryx Inc Compuestos de anillo 5,5 fusionado sustituido con diarilo como inhibidores de c5ar.
BR112020019822A2 (pt) 2018-04-02 2021-03-16 Chemocentryx, Inc. Profármacos de antagonistas bicíclicos fundidos de c5ar
CN114957165A (zh) * 2021-02-26 2022-08-30 清华大学 一种抗病毒化合物及其制备方法和应用

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