JP2003516393A5 - - Google Patents

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Publication number
JP2003516393A5
JP2003516393A5 JP2001543517A JP2001543517A JP2003516393A5 JP 2003516393 A5 JP2003516393 A5 JP 2003516393A5 JP 2001543517 A JP2001543517 A JP 2001543517A JP 2001543517 A JP2001543517 A JP 2001543517A JP 2003516393 A5 JP2003516393 A5 JP 2003516393A5
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JP
Japan
Prior art keywords
oxo
compound
acid
substituted
embedded image
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JP2001543517A
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English (en)
Japanese (ja)
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JP2003516393A (ja
JP5021131B2 (ja
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Priority claimed from PCT/US2000/033260 external-priority patent/WO2001042216A2/en
Publication of JP2003516393A publication Critical patent/JP2003516393A/ja
Publication of JP2003516393A5 publication Critical patent/JP2003516393A5/ja
Application granted granted Critical
Publication of JP5021131B2 publication Critical patent/JP5021131B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2001543517A 1999-12-08 2000-12-08 カスパーゼインヒビターおよびその使用 Expired - Fee Related JP5021131B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16981299P 1999-12-08 1999-12-08
US60/169,812 1999-12-08
PCT/US2000/033260 WO2001042216A2 (en) 1999-12-08 2000-12-08 Caspase inhibitors and uses thereof

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2007315252A Division JP2008101019A (ja) 1999-12-08 2007-12-05 カスパーゼインヒビターおよびその使用
JP2011234386A Division JP2012021032A (ja) 1999-12-08 2011-10-25 カスパーゼインヒビターおよびその使用

Publications (3)

Publication Number Publication Date
JP2003516393A JP2003516393A (ja) 2003-05-13
JP2003516393A5 true JP2003516393A5 (enExample) 2008-01-31
JP5021131B2 JP5021131B2 (ja) 2012-09-05

Family

ID=22617272

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2001543517A Expired - Fee Related JP5021131B2 (ja) 1999-12-08 2000-12-08 カスパーゼインヒビターおよびその使用
JP2007315252A Withdrawn JP2008101019A (ja) 1999-12-08 2007-12-05 カスパーゼインヒビターおよびその使用
JP2011234386A Withdrawn JP2012021032A (ja) 1999-12-08 2011-10-25 カスパーゼインヒビターおよびその使用

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2007315252A Withdrawn JP2008101019A (ja) 1999-12-08 2007-12-05 カスパーゼインヒビターおよびその使用
JP2011234386A Withdrawn JP2012021032A (ja) 1999-12-08 2011-10-25 カスパーゼインヒビターおよびその使用

Country Status (24)

Country Link
US (4) US7517987B2 (enExample)
EP (4) EP1244626A2 (enExample)
JP (3) JP5021131B2 (enExample)
KR (3) KR100904697B1 (enExample)
CN (2) CN101348455A (enExample)
AP (1) AP2002002535A0 (enExample)
AR (1) AR026748A1 (enExample)
AU (3) AU2428301A (enExample)
BR (1) BR0016282A (enExample)
CA (2) CA2733434A1 (enExample)
CO (1) CO5261609A1 (enExample)
CZ (1) CZ20021970A3 (enExample)
EA (1) EA200200645A1 (enExample)
HU (1) HUP0300782A3 (enExample)
IL (1) IL150077A0 (enExample)
IS (1) IS6411A (enExample)
MX (1) MXPA02005779A (enExample)
NO (2) NO324776B1 (enExample)
NZ (2) NZ530485A (enExample)
PL (1) PL356066A1 (enExample)
SK (1) SK8072002A3 (enExample)
TW (1) TWI275586B (enExample)
WO (1) WO2001042216A2 (enExample)
ZA (1) ZA200204390B (enExample)

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WO2008116107A2 (en) 2007-03-21 2008-09-25 Takeda San Diego, Inc. Piperazine derivatives as glucokinase activators
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EP2699091B1 (en) 2011-03-28 2017-06-21 DeuteRx, LLC 2',6'-dioxo-3'-deutero-piperdin-3-yl-isoindoline compounds
DK2697246T3 (en) 2011-04-15 2018-05-28 Genesis Tech Limited SELECTIVE CYSTEIN PROTEASE INHIBITORS AND USES THEREOF
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US9540340B2 (en) 2013-01-14 2017-01-10 Deuterx, Llc 3-(5-substituted-4-oxoquinazolin-3(4H)-yl)-3-deutero-piperidine-2,6-dione derivatives and compositions comprising and methods of using the same
WO2014152833A1 (en) 2013-03-14 2014-09-25 Deuterx, Llc 3-(substituted-4-oxo-quinazolin-3(4h)-yl)-3-deutero-piperidine-2,6-dione derivatives
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WO2018133870A1 (zh) 2017-01-23 2018-07-26 正大天晴药业集团股份有限公司 作为Caspase抑制剂的联环化合物
CN106749045B (zh) * 2017-03-03 2020-02-14 上海交通大学 一种d-氨基酸氧化酶抑制剂及其制法和应用
SG11202002913QA (en) * 2017-10-04 2020-04-29 Battelle Memorial Institute Probe for selectively characterizing enzymes involved in xenobiotic metabolism and method of making and using the same
CA3171430A1 (en) * 2020-03-13 2021-09-16 Brent R. Stockwell Gpx4 compounds and compositions and methods of treatment using same
AU2021321068B2 (en) * 2020-08-05 2025-01-02 Lg Chem, Ltd. Use of caspase inhibitor for alleviating or treating osteoarthritis
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CN120265616A (zh) * 2022-09-26 2025-07-04 艾知怀斯治疗学公司 1,4-二氢喹唑啉酮化合物及其用途
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