JP2003513076A5 - - Google Patents

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Publication number
JP2003513076A5
JP2003513076A5 JP2001534779A JP2001534779A JP2003513076A5 JP 2003513076 A5 JP2003513076 A5 JP 2003513076A5 JP 2001534779 A JP2001534779 A JP 2001534779A JP 2001534779 A JP2001534779 A JP 2001534779A JP 2003513076 A5 JP2003513076 A5 JP 2003513076A5
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JP
Japan
Prior art keywords
alkyl
amino
partially
heteroaryl
halogenated
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2001534779A
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English (en)
Japanese (ja)
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JP4861585B2 (ja
JP2003513076A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2000/029891 external-priority patent/WO2001032627A1/en
Publication of JP2003513076A publication Critical patent/JP2003513076A/ja
Publication of JP2003513076A5 publication Critical patent/JP2003513076A5/ja
Application granted granted Critical
Publication of JP4861585B2 publication Critical patent/JP4861585B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2001534779A 1999-10-29 2000-10-27 置換ピラゾールの合成方法 Expired - Fee Related JP4861585B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US16247699P 1999-10-29 1999-10-29
US60/162,476 1999-10-29
US19265100P 2000-03-28 2000-03-28
US60/192,651 2000-03-28
PCT/US2000/029891 WO2001032627A1 (en) 1999-10-29 2000-10-27 Process of making substituted pyrazoles

Publications (3)

Publication Number Publication Date
JP2003513076A JP2003513076A (ja) 2003-04-08
JP2003513076A5 true JP2003513076A5 (https=) 2007-12-20
JP4861585B2 JP4861585B2 (ja) 2012-01-25

Family

ID=26858795

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001534779A Expired - Fee Related JP4861585B2 (ja) 1999-10-29 2000-10-27 置換ピラゾールの合成方法

Country Status (11)

Country Link
EP (1) EP1235810B1 (https=)
JP (1) JP4861585B2 (https=)
AT (1) ATE244704T1 (https=)
AU (1) AU1445001A (https=)
CA (1) CA2387762C (https=)
DE (1) DE60003846T2 (https=)
DK (1) DK1235810T3 (https=)
ES (1) ES2202189T3 (https=)
MX (1) MXPA02004004A (https=)
PT (1) PT1235810E (https=)
WO (1) WO2001032627A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6407238B1 (en) 1999-10-29 2002-06-18 Boehringer Ingelheim Pharmaceuticals, Inc. Process of making substituted pyrazoles
US6492529B1 (en) 2000-01-18 2002-12-10 Boehringer Ingelheim Pharmaceuticals, Inc. Bis pyrazole-1H-pyrazole intermediates and their synthesis
EP1362037A1 (en) 2001-02-15 2003-11-19 Boehringer Ingelheim Pharmaceuticals Inc. Process for synthesis of heteroaryl-substituted urea compounds useful as antiinflammatory agents
DE10315569A1 (de) * 2003-04-05 2004-10-14 Merck Patent Gmbh Substituierte Pyrazolverbindungen
DE10315573A1 (de) 2003-04-05 2004-10-14 Merck Patent Gmbh Substituierte Pyrazole
DE10315571A1 (de) 2003-04-05 2004-10-14 Merck Patent Gmbh Pyrazolverbindungen
WO2007044490A2 (en) 2005-10-06 2007-04-19 Boehringer Ingelheim International Gmbh Process for making heteroaryl amine intermediate compounds
EP2135865A1 (de) 2008-06-17 2009-12-23 Bayer CropScience AG Substituierte 1-(Diazinyl) pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
EP2194052A1 (de) 2008-12-06 2010-06-09 Bayer CropScience AG Substituierte 1-(Thiazolyl)- und 1-(Isothiazolyl)pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
WO2011073098A1 (de) 2009-12-15 2011-06-23 Bayer Cropscience Ag 1-(heteroaryl)-pyrazol-4-yl-essigsäuren, verfahren zu deren herstellung und deren verwendung als herbizide und pflanzenwachstumsregulatoren
WO2020113094A1 (en) 2018-11-30 2020-06-04 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4314851A1 (de) * 1993-05-05 1994-11-10 Huels Chemische Werke Ag Verfahren zur Herstellung von 3-Amino-5-methylpyrazol
US5698708A (en) * 1996-06-20 1997-12-16 Monsanto Company Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity
CA2258215A1 (en) * 1996-06-20 1997-12-24 Monsanto Company Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity
WO1999023091A1 (en) * 1997-11-03 1999-05-14 Boehringer Ingelheim Pharmaceuticals, Inc. Aromatic heterocyclic compounds as anti-inflammatory agents

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