JP2003511437A - Ｎ−［３−［［２−（３，４−ジメトキシフェニル）エチル］アミノ］プロピル］−４−ニトロベンズアミド塩酸塩の多型相 - Google Patents

Ｎ−［３−［［２−（３，４−ジメトキシフェニル）エチル］アミノ］プロピル］−４−ニトロベンズアミド塩酸塩の多型相

Info

Publication number
JP2003511437A
JP2003511437A JP2001530092A JP2001530092A JP2003511437A JP 2003511437 A JP2003511437 A JP 2003511437A JP 2001530092 A JP2001530092 A JP 2001530092A JP 2001530092 A JP2001530092 A JP 2001530092A JP 2003511437 A JP2003511437 A JP 2003511437A
Authority
JP
Japan
Prior art keywords
polymorphic form
propyl
dimethoxyphenyl
ethyl
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2001530092A
Other languages
English (en)
Japanese (ja)
Inventor
デイビッド・バスビー
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Publication of JP2003511437A publication Critical patent/JP2003511437A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/77—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
    • C07C233/78—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2001530092A 1999-10-08 2000-10-06 Ｎ−［３−［［２−（３，４−ジメトキシフェニル）エチル］アミノ］プロピル］−４−ニトロベンズアミド塩酸塩の多型相 Pending JP2003511437A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9923933.7 1999-10-08
GBGB9923933.7A GB9923933D0 (en) 1999-10-08 1999-10-08 Novel pharmaceutical
PCT/GB2000/003847 WO2001027071A1 (en) 1999-10-08 2000-10-06 Polymorphic n-[3-[[2-(3,4-dimethoxyphenyl) ethyl] amino] propyl] -4-nitro benzamide hydrochloride

Publications (1)

Publication Number Publication Date
JP2003511437A true JP2003511437A (ja) 2003-03-25

Family

ID=10862442

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001530092A Pending JP2003511437A (ja) 1999-10-08 2000-10-06 Ｎ−［３−［［２−（３，４−ジメトキシフェニル）エチル］アミノ］プロピル］−４−ニトロベンズアミド塩酸塩の多型相

Country Status (18)

Country Link
EP (1) EP1218334A1 (no)
JP (1) JP2003511437A (no)
KR (1) KR20020043618A (no)
CN (1) CN1384817A (no)
AU (1) AU7546000A (no)
BR (1) BR0014591A (no)
CA (1) CA2386845A1 (no)
CZ (1) CZ20021189A3 (no)
GB (1) GB9923933D0 (no)
HK (1) HK1049147A1 (no)
HU (1) HUP0203582A2 (no)
IL (1) IL148966A0 (no)
MX (1) MXPA02003516A (no)
NO (1) NO20021639L (no)
PL (1) PL354137A1 (no)
TR (1) TR200200949T2 (no)
WO (1) WO2001027071A1 (no)
ZA (1) ZA200202679B (no)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010511689A (ja) * 2006-12-06 2010-04-15 ファイザー・インク （３Ｓ）−３−［Ｎ−（Ｎ’−（２−ｔｅｒｔ−ブチルフェニル）オキサミル）アラニニル］アミノ−５−（２’，３’，５’，６’−テトラフルオロフェノキシ）−４−オキソペンタン酸の結晶形態

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7227033B2 (en) 2002-01-09 2007-06-05 Emisphere Technologies, Inc. Polymorphs of sodium 4-[(4-chloro-2-hydroxybenzoyl) amino] butanoate

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2726267B1 (fr) * 1994-10-26 1998-01-02 Smithkline Beecham Lab Nouveaux agents anti-arythmiques, compositions pharmaceutiques les contenant, et procede pour les preparer
GB9706376D0 (en) * 1997-03-27 1997-05-14 Smithkline Beecham Plc Novel pharmaceutical

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010511689A (ja) * 2006-12-06 2010-04-15 ファイザー・インク （３Ｓ）−３−［Ｎ−（Ｎ’−（２−ｔｅｒｔ−ブチルフェニル）オキサミル）アラニニル］アミノ−５−（２’，３’，５’，６’−テトラフルオロフェノキシ）−４−オキソペンタン酸の結晶形態

Also Published As

Publication number Publication date
GB9923933D0 (en) 1999-12-08
EP1218334A1 (en) 2002-07-03
NO20021639L (no) 2002-05-30
PL354137A1 (en) 2003-12-29
WO2001027071A1 (en) 2001-04-19
HK1049147A1 (zh) 2003-05-02
NO20021639D0 (no) 2002-04-05
AU7546000A (en) 2001-04-23
BR0014591A (pt) 2002-06-11
MXPA02003516A (es) 2004-09-10
CA2386845A1 (en) 2001-04-19
TR200200949T2 (tr) 2002-08-21
IL148966A0 (en) 2002-11-10
HUP0203582A2 (en) 2004-03-01
ZA200202679B (en) 2003-05-28
CN1384817A (zh) 2002-12-11
KR20020043618A (ko) 2002-06-10
CZ20021189A3 (cs) 2002-09-11

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