JP2002534519A5 - - Google Patents

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Publication number
JP2002534519A5
JP2002534519A5 JP2000593604A JP2000593604A JP2002534519A5 JP 2002534519 A5 JP2002534519 A5 JP 2002534519A5 JP 2000593604 A JP2000593604 A JP 2000593604A JP 2000593604 A JP2000593604 A JP 2000593604A JP 2002534519 A5 JP2002534519 A5 JP 2002534519A5
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JP
Japan
Prior art keywords
phenyl
alkyl
triazol
halogen
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2000593604A
Other languages
English (en)
Japanese (ja)
Other versions
JP2002534519A (ja
JP4933694B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2000/000177 external-priority patent/WO2000042036A1/de
Publication of JP2002534519A publication Critical patent/JP2002534519A/ja
Publication of JP2002534519A5 publication Critical patent/JP2002534519A5/ja
Application granted granted Critical
Publication of JP4933694B2 publication Critical patent/JP4933694B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2000593604A 1999-01-12 2000-01-12 ドーパミン−ｄ３−レセプター親和性を有するトリアゾール化合物 Expired - Fee Related JP4933694B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19900811 1999-01-12
DE19900811.6 1999-01-12
PCT/EP2000/000177 WO2000042036A1 (de) 1999-01-12 2000-01-12 Triazolverbindungen mit dopamin-d3-rezeptoraffinität

Publications (3)

Publication Number Publication Date
JP2002534519A JP2002534519A (ja) 2002-10-15
JP2002534519A5 true JP2002534519A5 (https=) 2010-10-28
JP4933694B2 JP4933694B2 (ja) 2012-05-16

Family

ID=7894006

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2000593605A Expired - Fee Related JP4615125B2 (ja) 1999-01-12 2000-01-12 ドーパミン−ｄ３−レセプター親和性を有するトリアゾール化合物
JP2000593606A Ceased JP2002534521A (ja) 1999-01-12 2000-01-12 ドーパミン−３−レセプター親和性を有するトリアゾール化合物
JP2000593604A Expired - Fee Related JP4933694B2 (ja) 1999-01-12 2000-01-12 ドーパミン−ｄ３−レセプター親和性を有するトリアゾール化合物

Family Applications Before (2)

Application Number Title Priority Date Filing Date
JP2000593605A Expired - Fee Related JP4615125B2 (ja) 1999-01-12 2000-01-12 ドーパミン−ｄ３−レセプター親和性を有するトリアゾール化合物
JP2000593606A Ceased JP2002534521A (ja) 1999-01-12 2000-01-12 ドーパミン−３−レセプター親和性を有するトリアゾール化合物

Country Status (28)

Country Link
US (3) US6602867B1 (https=)
EP (3) EP1144405B1 (https=)
JP (3) JP4615125B2 (https=)
KR (3) KR100775720B1 (https=)
CN (3) CN1267430C (https=)
AR (3) AR022230A1 (https=)
AT (3) ATE366729T1 (https=)
AU (3) AU2289700A (https=)
BG (2) BG65105B1 (https=)
BR (2) BR0007500A (https=)
CA (3) CA2359948C (https=)
CO (3) CO5150182A1 (https=)
CZ (2) CZ20012550A3 (https=)
DE (3) DE50014472D1 (https=)
ES (2) ES2288839T3 (https=)
HK (1) HK1045311B (https=)
HR (1) HRP20010590A2 (https=)
HU (2) HUP0200709A3 (https=)
ID (2) ID29552A (https=)
IL (3) IL144136A0 (https=)
NO (2) NO20013444L (https=)
NZ (2) NZ512830A (https=)
PL (2) PL201889B1 (https=)
SK (2) SK9862001A3 (https=)
TR (2) TR200102026T2 (https=)
TW (1) TWI274750B (https=)
WO (3) WO2000042036A1 (https=)
ZA (2) ZA200106584B (https=)

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BRPI0518823A2 (pt) 2004-12-02 2008-12-09 Abbott Gmbh & Co Kg compostos de triazol adequados para o tratamento de transtornos que respondam À modulaÇço do receptor d3 da dopamina
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JP5118039B2 (ja) 2005-08-18 2013-01-16 シンタ ファーマシューティカルズ コーポレーション Ｈｓｐ９０活性を調節するトリアゾール化合物
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CN102264733B (zh) 2008-10-10 2014-07-30 中国人民解放军军事医学科学院毒物药物研究所 新型多巴胺d3受体配体，其制备方法及其医药用途
US9326955B2 (en) * 2008-10-31 2016-05-03 Loyola University Chicago Combination pharmaceuticals and methods thereof using proteinacious channels as treatments for medical conditions
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JPWO2012124744A1 (ja) * 2011-03-14 2014-07-24 大正製薬株式会社 含窒素縮合複素環化合物
PE20142366A1 (es) * 2012-05-30 2015-01-10 Hoffmann La Roche Compuestos triazolo como inhibidores de pde 10
RU2561063C1 (ru) * 2014-07-01 2015-08-20 Общество с ограниченной ответственностью "Научно-производственное объединение "Фарматрон" (НПО "Фарматрон") Способ коррекции неврологических нарушений при хронической алкогольной интоксикации
GB201415573D0 (en) 2014-09-03 2014-10-15 Cancer Therapeutics Crc Pty Ltd Compounds
WO2016034673A1 (en) 2014-09-03 2016-03-10 Ctxt Pty Ltd Tetrahydroisoquinoline derived prmt5-inhibitors
EP3189048B1 (en) 2014-09-03 2021-03-17 Ctxt Pty Ltd Aminoindane-, aminotetrahydronaphthalene- and aminobenzocyclobutane-derived prmt5-inhibitors
GB201604030D0 (en) 2016-03-09 2016-04-20 Ctxt Pty Ltd Compounds
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GB201604022D0 (en) 2016-03-09 2016-04-20 Ctxt Pty Ltd Compounds
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EP3634406B1 (en) * 2017-05-12 2023-09-06 Board of Trustees of The Southern Illinois University on behalf of Southern Illinois University Edwardsville 3,4,5-trisubstituted-1,2,4-triazoles and 3,4,5-trisubstituted-3-thio-1,2,4-triazoles and uses thereof
US10941153B2 (en) * 2018-05-31 2021-03-09 Regents Of The University Of Minnesota Substituted phenethylamine derivatives
GB202117129D0 (en) * 2021-11-26 2022-01-12 Epidarex Exeed Ltd Compounds

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