JP2002523366A - ドーパミン再取込みインヒビターを含有する組成物及びその使用方法 - Google Patents
ドーパミン再取込みインヒビターを含有する組成物及びその使用方法Info
- Publication number
- JP2002523366A JP2002523366A JP2000565873A JP2000565873A JP2002523366A JP 2002523366 A JP2002523366 A JP 2002523366A JP 2000565873 A JP2000565873 A JP 2000565873A JP 2000565873 A JP2000565873 A JP 2000565873A JP 2002523366 A JP2002523366 A JP 2002523366A
- Authority
- JP
- Japan
- Prior art keywords
- didesmethylsibutramine
- desmethylsibutramine
- sibutramine
- metabolite
- pharmaceutically acceptable
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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Classifications
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- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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Landscapes
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Applications Claiming Priority (7)
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| PCT/US1999/019167 WO2000010551A2 (en) | 1998-08-24 | 1999-08-23 | Methods of using and compositions comprising dopamine reuptake inhibitors |
Publications (2)
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| JP (1) | JP2002523366A (enExample) |
| KR (3) | KR20080011354A (enExample) |
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| ES (1) | ES2226435T3 (enExample) |
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| NZ (1) | NZ510193A (enExample) |
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Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2003504303A (ja) * | 1998-12-02 | 2003-02-04 | ピーター・スターリング・ミュラー | 器質性障害から派生する障害の治療 |
| JP2003519087A (ja) * | 1999-03-19 | 2003-06-17 | クノール・ゲー・エム・ベー・ハー | 摂食障害を治療する方法 |
| JP2003519675A (ja) * | 2000-01-11 | 2003-06-24 | セプラコア インコーポレーテッド | シブトラミンのラセミ型又は光学的に純粋な代謝産物、それらの調製、それらを含有する組成物及びそれらのドーパミン再取込みインヒビターとしての使用 |
| JP2008526836A (ja) * | 2005-01-06 | 2008-07-24 | シージェー チェイルジェダン コーポレーション | シブトラミンの無機酸塩 |
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| US6339106B1 (en) * | 1999-08-11 | 2002-01-15 | Sepracor, Inc. | Methods and compositions for the treatment and prevention of sexual dysfunction |
| US6476078B2 (en) * | 1999-08-11 | 2002-11-05 | Sepracor, Inc. | Methods of using sibutramine metabolites in combination with a phosphodiesterase inhibitor to treat sexual dysfunction |
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| US6696495B2 (en) | 1998-12-02 | 2004-02-24 | Snowden Pharmaceuticals, Llc | Treatment of disorders secondary to organic impairments |
| KR100948757B1 (ko) * | 1999-07-01 | 2010-03-23 | 파마시아 앤드 업존 캄파니 엘엘씨 | 고선택성 노르에피네프린 재흡수 억제제 및 그의 이용 방법 |
| WO2002036540A2 (en) * | 2000-11-02 | 2002-05-10 | Torrent Pharmaceuticals Ltd | PROCESS FOR PREPARATION OF β-PHENETHYLAMINE DERIVATIVE |
| US20020115727A1 (en) * | 2000-12-04 | 2002-08-22 | Senanayake Chris H. | Synthesis, methods of using, and compositions of hydroxylated cyclobutylalkylamines |
| ATE409475T1 (de) * | 2001-02-20 | 2008-10-15 | Dinan Timothy Gerard | Behandlung von fibromyalgie mit pindolol |
| DE10142666A1 (de) * | 2001-08-31 | 2003-03-20 | Aventis Pharma Gmbh | Verwendung von C2-substituierten Indan-1-ol-Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas |
| US6602911B2 (en) * | 2001-11-05 | 2003-08-05 | Cypress Bioscience, Inc. | Methods of treating fibromyalgia |
| US7005138B2 (en) * | 2001-12-21 | 2006-02-28 | Duramed Pharmaceuticals, Inc. | Method of systematically delivering SSRIs |
| US20060263419A1 (en) * | 2002-03-12 | 2006-11-23 | Hans-Michael Wolff | Transdermal therapeutic system for Parkinson's Disease |
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| US20050267176A1 (en) * | 2004-02-18 | 2005-12-01 | Sepracor Inc. | Dopamine-agonist combination therapy for improving sleep quality |
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| WO2006115770A2 (en) * | 2005-04-22 | 2006-11-02 | Teva Pharmaceuticals Usa, Inc. | Orally disintegrating pharmaceutical tablet formulations of olanzapine |
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| WO2010093243A1 (en) | 2009-02-12 | 2010-08-19 | Coöperatieve Mirzorg U.A., Arnhem | Use of a combination of diazoxide and metformin for treating obesity or obesity related disorders |
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- 1999-08-11 US US09/372,158 patent/US6331571B1/en not_active Expired - Lifetime
- 1999-08-23 ES ES99945137T patent/ES2226435T3/es not_active Expired - Lifetime
- 1999-08-23 KR KR1020087001197A patent/KR20080011354A/ko not_active Ceased
- 1999-08-23 WO PCT/US1999/019167 patent/WO2000010551A2/en not_active Ceased
- 1999-08-23 NZ NZ510193A patent/NZ510193A/en not_active IP Right Cessation
- 1999-08-23 AT AT99945137T patent/ATE279184T1/de active
- 1999-08-23 DK DK99945137T patent/DK1107746T3/da active
- 1999-08-23 HU HU0103408A patent/HUP0103408A3/hu unknown
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- 1999-08-23 AU AU57817/99A patent/AU772303B2/en not_active Ceased
- 1999-08-23 PL PL346843A patent/PL200264B1/pl not_active IP Right Cessation
- 1999-08-23 KR KR1020017002288A patent/KR20010085553A/ko not_active Ceased
- 1999-08-23 EP EP04018454A patent/EP1475086A3/en not_active Withdrawn
- 1999-08-23 PT PT99945137T patent/PT1107746E/pt unknown
- 1999-08-23 CZ CZ2001677A patent/CZ2001677A3/cs unknown
- 1999-08-23 DE DE69921157T patent/DE69921157T2/de not_active Expired - Lifetime
- 1999-08-23 JP JP2000565873A patent/JP2002523366A/ja active Pending
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2001
- 2001-02-20 IL IL141531A patent/IL141531A/en not_active IP Right Cessation
- 2001-02-23 NO NO20010943A patent/NO20010943L/no not_active Application Discontinuation
- 2001-12-04 US US10/000,806 patent/US6538034B2/en not_active Expired - Lifetime
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2003
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| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2003504303A (ja) * | 1998-12-02 | 2003-02-04 | ピーター・スターリング・ミュラー | 器質性障害から派生する障害の治療 |
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| JP2003519675A (ja) * | 2000-01-11 | 2003-06-24 | セプラコア インコーポレーテッド | シブトラミンのラセミ型又は光学的に純粋な代謝産物、それらの調製、それらを含有する組成物及びそれらのドーパミン再取込みインヒビターとしての使用 |
| JP2008526836A (ja) * | 2005-01-06 | 2008-07-24 | シージェー チェイルジェダン コーポレーション | シブトラミンの無機酸塩 |
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