JP2000507246A - 固体相のリポグリコペプチドライブラリー、組成物及び方法 - Google Patents

固体相のリポグリコペプチドライブラリー、組成物及び方法

Info

Publication number
JP2000507246A
JP2000507246A JP9533750A JP53375097A JP2000507246A JP 2000507246 A JP2000507246 A JP 2000507246A JP 9533750 A JP9533750 A JP 9533750A JP 53375097 A JP53375097 A JP 53375097A JP 2000507246 A JP2000507246 A JP 2000507246A
Authority
JP
Japan
Prior art keywords
substituent
mmol
substituents
library
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP9533750A
Other languages
English (en)
Japanese (ja)
Inventor
マイケル ソフィア
ナイジェル アランソン
アンナ チェン
ダシャン リュウ
ティン ヤウ チャン
Original Assignee
トランセル テクノロジーズ インク．
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by トランセル テクノロジーズ インク． filed Critical トランセル テクノロジーズ インク．
Publication of JP2000507246A publication Critical patent/JP2000507246A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/001—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence having less than 12 amino acids and not being part of a ring structure
    • C07K9/005—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence having less than 12 amino acids and not being part of a ring structure containing within the molecule the substructure with m, n > 0 and m+n > 0, A, B, D, E being heteroatoms; X being a bond or a chain, e.g. muramylpeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/047—Simultaneous synthesis of different peptide species; Peptide libraries

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Analytical Chemistry (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP9533750A 1996-03-21 1997-03-21 固体相のリポグリコペプチドライブラリー、組成物及び方法 Pending JP2000507246A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US1377796P 1996-03-21 1996-03-21
US60/013,777 1996-03-21
US2452896P 1996-08-26 1996-08-26
US60/024,528 1996-08-26
PCT/US1997/004637 WO1997034623A1 (en) 1996-03-21 1997-03-21 Solid phase lipoglycopeptide library, compositions and methods

Publications (1)

Publication Number Publication Date
JP2000507246A true JP2000507246A (ja) 2000-06-13

Family

ID=26685236

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9533750A Pending JP2000507246A (ja) 1996-03-21 1997-03-21 固体相のリポグリコペプチドライブラリー、組成物及び方法

Country Status (5)

Country Link
EP (1) EP0934076A1 (enrdf_load_stackoverflow)
JP (1) JP2000507246A (enrdf_load_stackoverflow)
AU (1) AU2341197A (enrdf_load_stackoverflow)
CA (1) CA2249323A1 (enrdf_load_stackoverflow)
WO (1) WO1997034623A1 (enrdf_load_stackoverflow)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005509615A (ja) * 2001-10-15 2005-04-14 ケミン・ファーマ・ヨーロッパ 抗菌及び細胞増殖抑制活性を有する炭水化物ベースの二環式環構造の製造及び使用

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19624345B4 (de) * 1996-06-19 2004-12-23 Südzucker AG Mannheim/Ochsenfurt Acylierte Kohlenhydrate mit mindestens einer mit dem Kohlenhydrat veretherten Carboxyalkyl-Gruppe, Verfahren zu deren Herstellung und deren Verwendung in Waschmitteln
DE19642751A1 (de) * 1996-10-16 1998-04-23 Deutsches Krebsforsch Saccharid-Bibliothek
ATE242783T1 (de) 1998-12-23 2003-06-15 Theravance Inc Glycopeptid-derivate und pharmazeutische zusammensetzungen, die sie enthalten
US20010051349A1 (en) 2000-02-17 2001-12-13 Glycominds Ltd. Combinatorial complex carbohydrate libraries and methods for the manufacture and uses thereof
AUPS213802A0 (en) 2002-05-03 2002-06-06 Alchemia Pty Ltd Disaccharides for drug discovery
AU2002952121A0 (en) 2002-10-17 2002-10-31 Alchemia Limited Novel carbohydrate based anti-bacterials
CN102796147A (zh) * 2005-10-04 2012-11-28 阿尔卡米亚有限公司 化合物库
US8835614B2 (en) 2008-12-16 2014-09-16 Genzyme Corporation Oligosaccharide-protein conjugates
CN113200935B (zh) * 2021-04-26 2022-07-08 威海海洋生物医药产业技术研究院有限公司 一种用于次氯酸检测的荧光探针及其制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU1602995A (en) * 1994-01-11 1995-08-01 Affymax Technologies N.V. Methods for the solid phase synthesis of glycoconjugates

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005509615A (ja) * 2001-10-15 2005-04-14 ケミン・ファーマ・ヨーロッパ 抗菌及び細胞増殖抑制活性を有する炭水化物ベースの二環式環構造の製造及び使用

Also Published As

Publication number Publication date
WO1997034623A1 (en) 1997-09-25
EP0934076A1 (en) 1999-08-11
EP0934076A4 (enrdf_load_stackoverflow) 1999-08-11
AU2341197A (en) 1997-10-10
CA2249323A1 (en) 1997-09-25

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