IT7849547A0 - Derivati esterei dell'acido nacetil-para-aminofenolico e loro preparazione - Google Patents

Derivati esterei dell'acido nacetil-para-aminofenolico e loro preparazione

Info

Publication number
IT7849547A0
IT7849547A0 IT7849547A IT4954778A IT7849547A0 IT 7849547 A0 IT7849547 A0 IT 7849547A0 IT 7849547 A IT7849547 A IT 7849547A IT 4954778 A IT4954778 A IT 4954778A IT 7849547 A0 IT7849547 A0 IT 7849547A0
Authority
IT
Italy
Prior art keywords
estere
aminophenolic
nacetyl
para
derivatives
Prior art date
Application number
IT7849547A
Other languages
English (en)
Other versions
IT1202822B (it
Original Assignee
Sterling Drug Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sterling Drug Inc filed Critical Sterling Drug Inc
Publication of IT7849547A0 publication Critical patent/IT7849547A0/it
Application granted granted Critical
Publication of IT1202822B publication Critical patent/IT1202822B/it

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT49547/78A 1977-05-26 1978-05-25 Derivati esterei dell'acido n-acetil-para-aminofenolico e loro preparazione IT1202822B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB22218/77A GB1583602A (en) 1977-05-26 1977-05-26 N-acetyl-para-aminophenyl-n'-acetyl-amino-thioalkanoic acid ester derivatives

Publications (2)

Publication Number Publication Date
IT7849547A0 true IT7849547A0 (it) 1978-05-25
IT1202822B IT1202822B (it) 1989-02-09

Family

ID=10175844

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49547/78A IT1202822B (it) 1977-05-26 1978-05-25 Derivati esterei dell'acido n-acetil-para-aminofenolico e loro preparazione

Country Status (15)

Country Link
US (4) US4181719A (it)
AT (1) AT368489B (it)
BE (1) BE867531A (it)
CH (1) CH644590A5 (it)
DE (1) DE2822789C2 (it)
DK (1) DK155832C (it)
FI (1) FI70208C (it)
FR (1) FR2391998A1 (it)
GB (1) GB1583602A (it)
IE (1) IE47072B1 (it)
IT (1) IT1202822B (it)
LU (1) LU79703A1 (it)
NL (1) NL176070C (it)
NO (1) NO146392C (it)
SE (1) SE448991B (it)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1111384B (it) * 1978-12-21 1986-01-13 Sigma Tau Ind Farmaceuti Guaiacil esteri di derivati dello acido mercaptopropionico procedimento per la loro preparazione e loro uso terapeutico
US4307073A (en) * 1980-08-08 1981-12-22 The Research Foundation Of State University Of New York Method and composition for reducing the toxicity of acetaminophen
US5103021A (en) * 1982-04-02 1992-04-07 Syntex (U.S.A.) Inc. Acetaminophen analogs, antigens, and antibodies
US4605754A (en) * 1982-04-02 1986-08-12 Syntex (U.S.A.) Inc. Acetaminophen analogs
US4504413A (en) * 1982-04-02 1985-03-12 Syva Company Acetaminophen analogs, antigens, and antibodies
CH654302A5 (de) * 1983-05-04 1986-02-14 Sandoz Ag Acylaminophenolderivate, ihre herstellung und arzneimittel, welche sie enthalten.
GB9305058D0 (en) * 1993-03-12 1993-04-28 Penn Pharm Ltd Pharmaceutical compositions
DE19711053C2 (de) * 1997-03-03 1999-09-02 Rommelspacher Kombinationspräparat aus 2-Methyl-thiazolidin-2,4-dicarbonsäure und Paracetamol
FR2814366A1 (fr) * 2000-09-22 2002-03-29 Rhodia Chimie Sa Procede de granulation de matieres actives par extrusion basse pression pour l'obtention de granules directement compressibles
WO2002036077A2 (en) * 2000-11-06 2002-05-10 Andrx Pharmaceuticals, Inc. Once a day antihistamine and decongestant formulation
GB0114069D0 (en) * 2001-06-08 2001-08-01 Smithkline Beecham Plc Composition
US8092831B2 (en) * 2002-11-08 2012-01-10 Andrx Pharmaceuticals, Llc Antihistamine and decongestant system
EP1603593A4 (en) * 2002-11-15 2007-08-01 Branded Products For The Futur PHARMACEUTICAL COMPOSITION
US20050220862A1 (en) * 2004-03-31 2005-10-06 Bernstein Joel E Compositions with reduced hepatotoxicity
US20090298923A1 (en) * 2008-05-13 2009-12-03 Genmedica Therapeutics Sl Salicylate Conjugates Useful for Treating Metabolic Disorders
CN102149412A (zh) * 2008-05-20 2011-08-10 纽罗吉斯克斯公司 肝脏保护剂对乙酰氨基酚协同前药
WO2010106082A1 (en) * 2009-03-16 2010-09-23 Genmedica Therapeutics Sl Anti-inflammatory and antioxidant conjugates useful for treating metabolic disorders
CN102421424A (zh) * 2009-03-16 2012-04-18 根梅迪卡治疗公司 用于治疗代谢性疾病的组合疗法
US8466197B2 (en) 2010-12-14 2013-06-18 Genmedica Therapeutics Sl Thiocarbonates as anti-inflammatory and antioxidant compounds useful for treating metabolic disorders

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR462M (it) * 1958-10-13 1961-05-02
US3591686A (en) * 1967-08-01 1971-07-06 Mead Johnson & Co Anti-inflammatory compositions and methods utilizing n-acylcysteines and the beta-alkyl and carboxyl derivatives thereof
US4038306A (en) * 1967-08-07 1977-07-26 Merck & Co., Inc. N-t-butoxycarbonyl-s-lower alkanoylamidomethyl-cysteine and p-nitrophenyl esters
GB1428803A (en) * 1973-05-29 1976-03-17 Gallardo Antonio Sa 4-acetamidophenyl esters of aryl-alkane carboxylic acids and a process for their preparation
US3983138A (en) * 1973-09-25 1976-09-28 Merck & Co., Inc. Amino acid esters
GB1463505A (en) * 1973-11-21 1977-02-02 Nat Res Dev Pharmaceutical compositions
US3996268A (en) * 1974-09-03 1976-12-07 The Regents Of The University Of California Cross-linking reagent for insulin synthesis

Also Published As

Publication number Publication date
FR2391998A1 (fr) 1978-12-22
SE448991B (sv) 1987-03-30
NO781824L (no) 1978-11-28
FI70208B (fi) 1986-02-28
LU79703A1 (fr) 1978-11-06
NO146392B (no) 1982-06-14
IT1202822B (it) 1989-02-09
NO146392C (no) 1982-09-22
US4482495A (en) 1984-11-13
AT368489B (de) 1982-10-11
DK231578A (da) 1978-11-27
DK155832B (da) 1989-05-22
IE781047L (en) 1978-11-26
US4181719A (en) 1980-01-01
SE7806038L (sv) 1978-11-27
FI70208C (fi) 1986-09-15
CH644590A5 (de) 1984-08-15
BE867531A (fr) 1978-09-18
DE2822789C2 (de) 1984-01-12
NL176070B (nl) 1984-09-17
FI781610A (fi) 1978-11-27
IE47072B1 (en) 1983-12-14
NL176070C (nl) 1985-02-18
DK155832C (da) 1989-10-02
GB1583602A (en) 1981-01-28
US4405800A (en) 1983-09-20
US4361703A (en) 1982-11-30
NL7805675A (nl) 1978-11-28
ATA380178A (de) 1982-02-15
FR2391998B1 (it) 1981-11-13
DE2822789A1 (de) 1978-12-07

Similar Documents

Publication Publication Date Title
IT7828768A0 (it) Derivati dell'acido 3- e 4-azidoftalico e procedimento per la loro preparazione.
IT7967573A0 (it) Derivati dell acido 2 m ben zoilfenossi propionico e loro impiegocome medicamenti
IT7849547A0 (it) Derivati esterei dell'acido nacetil-para-aminofenolico e loro preparazione
IT1097233B (it) Nuovi derivati dell'acido fenilacetico
IT7868914A0 (it) Derivati dell acido cicloalchilidenmetilfenilacetico particolarmente utili come medicamenti e procedimento per la loro preparazione
IT1097950B (it) Derivati dell'acido glicil-metil-fisfinico,loro preparazione e loro impiego
IT8067576A0 (it) Derivati dell acido penem 3 carbossilico loro preparazione ed impiego
IT1087384B (it) Derivati radiomarcati dell'acido folico
IT1117313B (it) Derivati dell'acido pirrol-1-carbossilico e procedimento per la loro preparazione
IT1133091B (it) Derivati dell acido penicillanico e procedimento per la loro preparazione
IT1109830B (it) Derivati di acido 1-azaxantone-3-carbossilico e procedimento per la loro preparazione
IT8167783A0 (it) Carbossilico e procedimento per la derivati dell acido penicil 3loro preparazione
IT1117314B (it) Derivati dell'acido pirrol-1-carbossilico e procedimento per la loro preparazione
IT7849300A0 (it) Derivati dell'acido 2-triclorometil4-nitrobenzolsolfenico
IT1075675B (it) Derivati dell'acido oleanoico
IT1097445B (it) Nuovi derivati dell'acido vincinico e procedimento per la loro preparazione
IT1126405B (it) Derivati esteri dell'acido farnesilacetico
IT1121530B (it) Nuovi derivati dell'acido 1-pirrolo-e 1-pirrolidin-carbossilico e procedimento per la loro preparazione
IT1113270B (it) Derivati dell'acido piridilfosforico e procedimento per la loro produzione
IT1122310B (it) Derivati dell'acido tio-propanoilamminico
IT1081510B (it) Derivati dell'acido 2-cianoesanoico
IT7967402A0 (it) Derivati dell'acido imidazolininil3 cloro 3 cefem 4 carbossilico eprocedimento per la loro preparazione
IT1141125B (it) Derivati dell'acido carbotioico di mercaptoacilamminocidi
IT1195761B (it) Derivati dell'acido ossayohimban-carbossilico
IT7828770A0 (it) Derivati dell'acido bis-azidoftalico e procedimento per la loro preparazione.