IT1289522B1 - Processo per la preparazione di eteroaril-fenilalanine - Google Patents
Processo per la preparazione di eteroaril-fenilalanineInfo
- Publication number
- IT1289522B1 IT1289522B1 IT96MI002738A ITMI962738A IT1289522B1 IT 1289522 B1 IT1289522 B1 IT 1289522B1 IT 96MI002738 A IT96MI002738 A IT 96MI002738A IT MI962738 A ITMI962738 A IT MI962738A IT 1289522 B1 IT1289522 B1 IT 1289522B1
- Authority
- IT
- Italy
- Prior art keywords
- preparation
- heteroaryl
- formula
- compounds
- eteroaril
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/26—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/55—Acids; Esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/12—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/30—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Priority Applications (15)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT96MI002738A IT1289522B1 (it) | 1996-12-24 | 1996-12-24 | Processo per la preparazione di eteroaril-fenilalanine |
| DE69705640T DE69705640T2 (de) | 1996-12-24 | 1997-12-15 | Verfahren zur herstellung von heteroaryl-phenylalaninen |
| PCT/EP1997/007024 WO1998028284A1 (en) | 1996-12-24 | 1997-12-15 | Process for the preparation of heteroaryl-phenylalanines |
| IL13036497A IL130364A (en) | 1996-12-24 | 1997-12-15 | Process for the preparation of heteroarylphenylalanines |
| CZ0230799A CZ296240B6 (cs) | 1996-12-24 | 1997-12-15 | Zpusob výroby heteroarylfenylalaninových derivátu |
| PT97952942T PT948492E (pt) | 1996-12-24 | 1997-12-15 | Processo para a preparacao de heteroaril-fenilalaninas |
| BRPI9713924-6A BR9713924B1 (pt) | 1996-12-24 | 1997-12-15 | processo para a preparaÇço de heteroarilafenilalaninas. |
| JP52833298A JP4226659B2 (ja) | 1996-12-24 | 1997-12-15 | ヘテロアリール−フェニルアラニン類の製造方法 |
| EP97952942A EP0948492B1 (en) | 1996-12-24 | 1997-12-15 | Process for the preparation of heteroaryl-phenylalanines |
| DK97952942T DK0948492T3 (da) | 1996-12-24 | 1997-12-15 | Fremgangsmåde til fremstilling af heteroarylphenylalaniner |
| AT97952942T ATE203017T1 (de) | 1996-12-24 | 1997-12-15 | Verfahren zur herstellung von heteroaryl- phenylalaninen |
| CA002275764A CA2275764C (en) | 1996-12-24 | 1997-12-15 | Process for the preparation of heteroaryl-phenylalanines |
| ES97952942T ES2159892T3 (es) | 1996-12-24 | 1997-12-15 | Procedimiento de preparacion de heteroaril - fenilalaninas |
| US09/331,164 US6448408B1 (en) | 1996-12-24 | 1997-12-15 | Process for the preparation of heteroaryl-phenylalanines |
| GR20010401721T GR3036855T3 (en) | 1996-12-24 | 2001-10-10 | Process for the preparation of heteroaryl-phenylalanines |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT96MI002738A IT1289522B1 (it) | 1996-12-24 | 1996-12-24 | Processo per la preparazione di eteroaril-fenilalanine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ITMI962738A1 ITMI962738A1 (it) | 1998-06-24 |
| IT1289522B1 true IT1289522B1 (it) | 1998-10-15 |
Family
ID=11375489
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT96MI002738A IT1289522B1 (it) | 1996-12-24 | 1996-12-24 | Processo per la preparazione di eteroaril-fenilalanine |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US6448408B1 (it) |
| EP (1) | EP0948492B1 (it) |
| JP (1) | JP4226659B2 (it) |
| AT (1) | ATE203017T1 (it) |
| BR (1) | BR9713924B1 (it) |
| CA (1) | CA2275764C (it) |
| CZ (1) | CZ296240B6 (it) |
| DE (1) | DE69705640T2 (it) |
| DK (1) | DK0948492T3 (it) |
| ES (1) | ES2159892T3 (it) |
| GR (1) | GR3036855T3 (it) |
| IL (1) | IL130364A (it) |
| IT (1) | IT1289522B1 (it) |
| PT (1) | PT948492E (it) |
| WO (1) | WO1998028284A1 (it) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4452899B2 (ja) * | 2001-12-13 | 2010-04-21 | 味の素株式会社 | 新規フェニルアラニン誘導体 |
| US8993599B2 (en) | 2003-07-18 | 2015-03-31 | Santarus, Inc. | Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1277737B1 (it) | 1995-12-28 | 1997-11-12 | Zambon Spa | Derivati tiolici ad attivita' inibitrice delle metallopeptidasi |
-
1996
- 1996-12-24 IT IT96MI002738A patent/IT1289522B1/it active IP Right Grant
-
1997
- 1997-12-15 IL IL13036497A patent/IL130364A/xx not_active IP Right Cessation
- 1997-12-15 DE DE69705640T patent/DE69705640T2/de not_active Expired - Lifetime
- 1997-12-15 EP EP97952942A patent/EP0948492B1/en not_active Expired - Lifetime
- 1997-12-15 AT AT97952942T patent/ATE203017T1/de active
- 1997-12-15 PT PT97952942T patent/PT948492E/pt unknown
- 1997-12-15 DK DK97952942T patent/DK0948492T3/da active
- 1997-12-15 ES ES97952942T patent/ES2159892T3/es not_active Expired - Lifetime
- 1997-12-15 JP JP52833298A patent/JP4226659B2/ja not_active Expired - Fee Related
- 1997-12-15 CZ CZ0230799A patent/CZ296240B6/cs not_active IP Right Cessation
- 1997-12-15 WO PCT/EP1997/007024 patent/WO1998028284A1/en active IP Right Grant
- 1997-12-15 CA CA002275764A patent/CA2275764C/en not_active Expired - Fee Related
- 1997-12-15 BR BRPI9713924-6A patent/BR9713924B1/pt not_active IP Right Cessation
- 1997-12-15 US US09/331,164 patent/US6448408B1/en not_active Expired - Lifetime
-
2001
- 2001-10-10 GR GR20010401721T patent/GR3036855T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ATE203017T1 (de) | 2001-07-15 |
| EP0948492A1 (en) | 1999-10-13 |
| WO1998028284A1 (en) | 1998-07-02 |
| US6448408B1 (en) | 2002-09-10 |
| PT948492E (pt) | 2001-11-30 |
| US20020028946A1 (en) | 2002-03-07 |
| DK0948492T3 (da) | 2001-10-15 |
| GR3036855T3 (en) | 2002-01-31 |
| JP2001506662A (ja) | 2001-05-22 |
| ITMI962738A1 (it) | 1998-06-24 |
| BR9713924B1 (pt) | 2009-01-13 |
| CA2275764C (en) | 2007-09-18 |
| ES2159892T3 (es) | 2001-10-16 |
| CA2275764A1 (en) | 1998-07-02 |
| IL130364A0 (en) | 2000-06-01 |
| BR9713924A (pt) | 2000-03-21 |
| DE69705640T2 (de) | 2002-05-02 |
| DE69705640D1 (de) | 2001-08-16 |
| CZ296240B6 (cs) | 2006-02-15 |
| EP0948492B1 (en) | 2001-07-11 |
| CZ230799A3 (cs) | 1999-12-15 |
| IL130364A (en) | 2003-07-06 |
| JP4226659B2 (ja) | 2009-02-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 0001 | Granted |