DK0948492T3 - Fremgangsmåde til fremstilling af heteroarylphenylalaniner - Google Patents

Fremgangsmåde til fremstilling af heteroarylphenylalaniner

Info

Publication number
DK0948492T3
DK0948492T3 DK97952942T DK97952942T DK0948492T3 DK 0948492 T3 DK0948492 T3 DK 0948492T3 DK 97952942 T DK97952942 T DK 97952942T DK 97952942 T DK97952942 T DK 97952942T DK 0948492 T3 DK0948492 T3 DK 0948492T3
Authority
DK
Denmark
Prior art keywords
preparation
heteroaryl
formula
compounds
heteroarylphenylalanines
Prior art date
Application number
DK97952942T
Other languages
English (en)
Inventor
Marco Villa
Maurizio Paiocchi
Katiuscia Arrighi
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Application granted granted Critical
Publication of DK0948492T3 publication Critical patent/DK0948492T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/26Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/55Acids; Esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/12Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/30Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Catalysts (AREA)
  • Indole Compounds (AREA)
DK97952942T 1996-12-24 1997-12-15 Fremgangsmåde til fremstilling af heteroarylphenylalaniner DK0948492T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT96MI002738A IT1289522B1 (it) 1996-12-24 1996-12-24 Processo per la preparazione di eteroaril-fenilalanine
PCT/EP1997/007024 WO1998028284A1 (en) 1996-12-24 1997-12-15 Process for the preparation of heteroaryl-phenylalanines

Publications (1)

Publication Number Publication Date
DK0948492T3 true DK0948492T3 (da) 2001-10-15

Family

ID=11375489

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97952942T DK0948492T3 (da) 1996-12-24 1997-12-15 Fremgangsmåde til fremstilling af heteroarylphenylalaniner

Country Status (15)

Country Link
US (1) US6448408B1 (da)
EP (1) EP0948492B1 (da)
JP (1) JP4226659B2 (da)
AT (1) ATE203017T1 (da)
BR (1) BR9713924B1 (da)
CA (1) CA2275764C (da)
CZ (1) CZ296240B6 (da)
DE (1) DE69705640T2 (da)
DK (1) DK0948492T3 (da)
ES (1) ES2159892T3 (da)
GR (1) GR3036855T3 (da)
IL (1) IL130364A (da)
IT (1) IT1289522B1 (da)
PT (1) PT948492E (da)
WO (1) WO1998028284A1 (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002354224A1 (en) * 2001-12-13 2003-07-09 Ajinomoto Co., Inc. Novel phenylalanine derivative
US8993599B2 (en) 2003-07-18 2015-03-31 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1277737B1 (it) 1995-12-28 1997-11-12 Zambon Spa Derivati tiolici ad attivita' inibitrice delle metallopeptidasi

Also Published As

Publication number Publication date
CA2275764A1 (en) 1998-07-02
CA2275764C (en) 2007-09-18
BR9713924B1 (pt) 2009-01-13
BR9713924A (pt) 2000-03-21
WO1998028284A1 (en) 1998-07-02
ATE203017T1 (de) 2001-07-15
ES2159892T3 (es) 2001-10-16
CZ296240B6 (cs) 2006-02-15
DE69705640D1 (de) 2001-08-16
US20020028946A1 (en) 2002-03-07
EP0948492A1 (en) 1999-10-13
US6448408B1 (en) 2002-09-10
GR3036855T3 (en) 2002-01-31
JP4226659B2 (ja) 2009-02-18
JP2001506662A (ja) 2001-05-22
CZ230799A3 (cs) 1999-12-15
IT1289522B1 (it) 1998-10-15
IL130364A (en) 2003-07-06
IL130364A0 (en) 2000-06-01
DE69705640T2 (de) 2002-05-02
EP0948492B1 (en) 2001-07-11
ITMI962738A1 (it) 1998-06-24
PT948492E (pt) 2001-11-30

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