IT1245889B - Formulazioni farmaceutiche per uso orale gastroresistenti contenenti sali di acidi biliari. - Google Patents

Formulazioni farmaceutiche per uso orale gastroresistenti contenenti sali di acidi biliari.

Info

Publication number
IT1245889B
IT1245889B ITBO910112A ITBO910112A IT1245889B IT 1245889 B IT1245889 B IT 1245889B IT BO910112 A ITBO910112 A IT BO910112A IT BO910112 A ITBO910112 A IT BO910112A IT 1245889 B IT1245889 B IT 1245889B
Authority
IT
Italy
Prior art keywords
gastro
resistant
pharmaceutical formulations
tablets
oral use
Prior art date
Application number
ITBO910112A
Other languages
English (en)
Inventor
Egidio Marchi
Gianfranco Tamagnone
Leone Gabriele Rotini
Original Assignee
Alfa Wassermann Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alfa Wassermann Spa filed Critical Alfa Wassermann Spa
Publication of ITBO910112A0 publication Critical patent/ITBO910112A0/it
Priority to ITBO910112A priority Critical patent/IT1245889B/it
Priority to US07/861,461 priority patent/US5302398A/en
Priority to ES92105714T priority patent/ES2090394T3/es
Priority to TW081102516A priority patent/TW202389B/zh
Priority to DK92105714.7T priority patent/DK0510404T3/da
Priority to DE69212882T priority patent/DE69212882T2/de
Priority to EP92105714A priority patent/EP0510404B1/en
Priority to CA002065809A priority patent/CA2065809C/en
Priority to JP4091129A priority patent/JP2509044B2/ja
Priority to KR1019920006051A priority patent/KR970005175B1/ko
Publication of ITBO910112A1 publication Critical patent/ITBO910112A1/it
Application granted granted Critical
Publication of IT1245889B publication Critical patent/IT1245889B/it
Priority to GR960402160T priority patent/GR3020843T3/el

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4808—Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4891—Coated capsules; Multilayered drug free capsule shells
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Nutrition Science (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Formulazioni farmaceutiche per uso orale ricoperte da una pellicola gastroresistente enterosolubile, preferibilmente scelte tra granulati gastroresistenti, compresse gastroresistenti, capsule gastroresistenti di gelatina dura contenenti polveri o granulati o due o più compresse o sospensioni oleose, capsule gastroresistenti di gelatina molle contenenti sospensioni oleose e capsule di gelatina dura contenenti granulati gastroresistenti o due o più compresse gastroresistenti, contenenti quantità terapeuticamente efficaci di sali degli acidi biliari con metalli alcalini o con basi organiche, processo per la loro preparazione e loro uso terapeutico nel trattamento delle calcolosi biliari, delle dispepsie biliari, della cirrosi biliare e delle epatopatie croniche e colestatiche.
ITBO910112A 1991-04-12 1991-04-12 Formulazioni farmaceutiche per uso orale gastroresistenti contenenti sali di acidi biliari. IT1245889B (it)

Priority Applications (11)

Application Number Priority Date Filing Date Title
ITBO910112A IT1245889B (it) 1991-04-12 1991-04-12 Formulazioni farmaceutiche per uso orale gastroresistenti contenenti sali di acidi biliari.
US07/861,461 US5302398A (en) 1991-04-12 1992-04-01 Gastroresistant pharmaceutical formulations for oral administration containing salts of bile acids
EP92105714A EP0510404B1 (en) 1991-04-12 1992-04-02 Gastroresistant pharmaceutical formulations for oral administration containing salts of bile acids
TW081102516A TW202389B (it) 1991-04-12 1992-04-02
DK92105714.7T DK0510404T3 (da) 1991-04-12 1992-04-02 Gastroresistente farmaceutiske formuleringer til oral administration indeholdende galdesyresalte
DE69212882T DE69212882T2 (de) 1991-04-12 1992-04-02 Gallensäuresalze enthaltende magenstabile pharmazeutische Zusammensetzung zur oralen Verabreichung
ES92105714T ES2090394T3 (es) 1991-04-12 1992-04-02 Formulados farmaceuticos gastroresistentes para administracion oral conteniendo sales de acidos biliares.
CA002065809A CA2065809C (en) 1991-04-12 1992-04-10 Gastroresistant pharmaceutical formulations for oral administration containing salts of bile acids
JP4091129A JP2509044B2 (ja) 1991-04-12 1992-04-10 胆汁酸塩を含有する胃液耐性のある経口投与用製剤
KR1019920006051A KR970005175B1 (ko) 1991-04-12 1992-04-11 담즙산의 염을 함유하는 경구용 위내성 의약 포뮬레이션
GR960402160T GR3020843T3 (en) 1991-04-12 1996-08-22 Gastroresistant pharmaceutical formulations for oral administration containing salts of bile acids

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITBO910112A IT1245889B (it) 1991-04-12 1991-04-12 Formulazioni farmaceutiche per uso orale gastroresistenti contenenti sali di acidi biliari.

Publications (3)

Publication Number Publication Date
ITBO910112A0 ITBO910112A0 (it) 1991-04-12
ITBO910112A1 ITBO910112A1 (it) 1992-10-12
IT1245889B true IT1245889B (it) 1994-10-25

Family

ID=11337388

Family Applications (1)

Application Number Title Priority Date Filing Date
ITBO910112A IT1245889B (it) 1991-04-12 1991-04-12 Formulazioni farmaceutiche per uso orale gastroresistenti contenenti sali di acidi biliari.

Country Status (11)

Country Link
US (1) US5302398A (it)
EP (1) EP0510404B1 (it)
JP (1) JP2509044B2 (it)
KR (1) KR970005175B1 (it)
CA (1) CA2065809C (it)
DE (1) DE69212882T2 (it)
DK (1) DK0510404T3 (it)
ES (1) ES2090394T3 (it)
GR (1) GR3020843T3 (it)
IT (1) IT1245889B (it)
TW (1) TW202389B (it)

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US7303768B2 (en) * 1998-07-24 2007-12-04 Seo Hong Yoo Preparation of aqueous clear solution dosage forms with bile acids
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FR2796272B1 (fr) 1999-07-15 2003-09-19 Oreal Composition sans cire structuree sous forme rigide par un polymere
FR2796271B1 (fr) 1999-07-15 2002-01-11 Oreal Composition sans cire structuree sous forme rigide par un polymere
ATE293425T1 (de) * 1999-12-28 2005-05-15 Oreal Strukturierte langhaltige zubereitung enthaltend ein polymer und pastöse fettstoffe
FR2804018B1 (fr) * 2000-01-24 2008-07-11 Oreal Composition sans transfert structuree sous forme rigide par un polymere
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AU2001220877A1 (en) * 2000-12-12 2002-06-24 L'oreal S.A. Cosmetic composition comprising heteropolymers and a solid substance and method of using same
US20020168335A1 (en) * 2000-12-12 2002-11-14 Nathalie Collin Cosmetic composition comprising a wax and a polymer
WO2002047630A1 (fr) * 2000-12-12 2002-06-20 L'oreal Composition cosmetique comprenant un melange de polymeres
WO2002047623A1 (en) 2000-12-12 2002-06-20 L'oreal Sa Composition comprising at least one heteropolymer and at least one inert filler and methods for use
FR2817740B1 (fr) * 2000-12-12 2006-08-04 Oreal Procede de fabrication d'une composition cosmetique coloree de maquillage a transmittance controlee
US8080257B2 (en) * 2000-12-12 2011-12-20 L'oreal S.A. Cosmetic compositions containing at least one hetero polymer and at least one film-forming silicone resin and methods of using
AU2002256544A1 (en) * 2000-12-12 2002-06-24 L'oreal Sa Cosmetic compositions containing at least one heteropolymer and at least one gelling agent and methods of using the same
US6881400B2 (en) * 2000-12-12 2005-04-19 L'oreal S.A. Use of at least one polyamide polymer in a mascara composition for increasing the adhesion of and/or expressly loading make-up deposited on eyelashes
FR2817739B1 (fr) * 2000-12-12 2005-01-07 Oreal Composition cosmetique coloree transparente ou translucide
US7276547B2 (en) * 2000-12-12 2007-10-02 L'oreal S.A. Compositions comprising heteropolymers and at least one oil-soluble polymers chosen from alkyl celluloses and alkylated guar gums
US6835399B2 (en) * 2000-12-12 2004-12-28 L'ORéAL S.A. Cosmetic composition comprising a polymer blend
US20020107314A1 (en) * 2000-12-12 2002-08-08 Carlos Pinzon Compositions containing heteropolymers and oil-soluble esters and methods of using same
AU2001225392A1 (en) * 2000-12-13 2002-06-24 L Oreal Composition structured with a polymer containing a heteroatom and an organogelator
FR2819400B1 (fr) * 2001-01-15 2004-12-03 Oreal Composition cosmetique de maquillage ou de soin des matieres keratiniques comprenant un melange de polymeres
US7025953B2 (en) * 2001-01-17 2006-04-11 L'oreal S.A. Nail polish composition comprising a polymer
FR2819399B1 (fr) * 2001-01-17 2003-02-21 Oreal Composition cosmetique contenant un polymere et une huile fluoree
CA2403670C (en) * 2001-01-31 2010-02-09 Rohm Gmbh & Co. Kg Multiparticulate drug form comprising at least two differently coated pellet forms
US6716420B2 (en) 2001-10-05 2004-04-06 L′Oreal Methods of use and of making a mascara comprising at least one coloring agent and at least one heteropolymer
FR2832060B1 (fr) * 2001-11-09 2004-07-09 Oreal Composition contenant un ester n-acyle d'acide amine et un filtre uv structuree par un polyamide
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US20050008598A1 (en) 2003-07-11 2005-01-13 Shaoxiang Lu Cosmetic compositions comprising a structuring agent, silicone powder and swelling agent
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US20040166133A1 (en) * 2003-01-21 2004-08-26 L'oreal Method of making a mascara composition comprising polyamide polymer and at least one solid substance having a melting point of 45oC or greater
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AU2005295541B2 (en) * 2004-10-15 2011-02-17 Seo Hong Yoo Methods and compositions for reducing toxicity of a pharmaceutical compound
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Also Published As

Publication number Publication date
CA2065809A1 (en) 1992-10-13
ES2090394T3 (es) 1996-10-16
KR970005175B1 (ko) 1997-04-14
ITBO910112A0 (it) 1991-04-12
GR3020843T3 (en) 1996-11-30
KR920019358A (ko) 1992-11-19
DE69212882T2 (de) 1997-01-23
CA2065809C (en) 1999-01-12
EP0510404A1 (en) 1992-10-28
US5302398A (en) 1994-04-12
EP0510404B1 (en) 1996-08-21
DK0510404T3 (da) 1996-09-09
JPH0597678A (ja) 1993-04-20
JP2509044B2 (ja) 1996-06-19
DE69212882D1 (de) 1996-09-26
ITBO910112A1 (it) 1992-10-12
TW202389B (it) 1993-03-21

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19960307