IT1237772B - Derivati di macrolidi polienici. - Google Patents

Derivati di macrolidi polienici.

Info

Publication number
IT1237772B
IT1237772B IT02239689A IT2239689A IT1237772B IT 1237772 B IT1237772 B IT 1237772B IT 02239689 A IT02239689 A IT 02239689A IT 2239689 A IT2239689 A IT 2239689A IT 1237772 B IT1237772 B IT 1237772B
Authority
IT
Italy
Prior art keywords
amines
partricin
radicals
reacting
prepared
Prior art date
Application number
IT02239689A
Other languages
English (en)
Other versions
IT8922396A0 (it
IT8922396A1 (it
Inventor
Tiberio Bruzzese
Franco Ottoni
Original Assignee
Tiberio Bruzzese
Franco Ottoni
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tiberio Bruzzese, Franco Ottoni filed Critical Tiberio Bruzzese
Publication of IT8922396A0 publication Critical patent/IT8922396A0/it
Priority to IT02239689A priority Critical patent/IT1237772B/it
Priority to DE69022196T priority patent/DE69022196T2/de
Priority to AT90121400T priority patent/ATE127471T1/de
Priority to EP90121400A priority patent/EP0434943B1/en
Priority to ES90121400T priority patent/ES2079417T3/es
Priority to US07/612,912 priority patent/US5296597A/en
Priority to PT95910A priority patent/PT95910B/pt
Priority to KR1019900018555A priority patent/KR0185200B1/ko
Priority to JP02308956A priority patent/JP3094065B2/ja
Publication of IT8922396A1 publication Critical patent/IT8922396A1/it
Application granted granted Critical
Publication of IT1237772B publication Critical patent/IT1237772B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/10—Preparation of carboxylic acid amides from compounds not provided for in groups C07C231/02 - C07C231/08
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Steroid Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
IT02239689A 1989-11-16 1989-11-16 Derivati di macrolidi polienici. IT1237772B (it)

Priority Applications (9)

Application Number Priority Date Filing Date Title
IT02239689A IT1237772B (it) 1989-11-16 1989-11-16 Derivati di macrolidi polienici.
ES90121400T ES2079417T3 (es) 1989-11-16 1990-11-08 Procedimiento de preparacion de derivados de la partricina.
AT90121400T ATE127471T1 (de) 1989-11-16 1990-11-08 Polyen-makrolidderivate.
EP90121400A EP0434943B1 (en) 1989-11-16 1990-11-08 Polyene macrolide derivatives
DE69022196T DE69022196T2 (de) 1989-11-16 1990-11-08 Polyen-Makrolidderivate.
US07/612,912 US5296597A (en) 1989-11-16 1990-11-14 Amide derivatives of Partricin A & Partricin B
PT95910A PT95910B (pt) 1989-11-16 1990-11-15 Processo para a preparacao de derivados macrolido de polieno
KR1019900018555A KR0185200B1 (ko) 1989-11-16 1990-11-16 폴리엔 마크로라이드 유도체
JP02308956A JP3094065B2 (ja) 1989-11-16 1990-11-16 ポリエン・マクロライド誘導体

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT02239689A IT1237772B (it) 1989-11-16 1989-11-16 Derivati di macrolidi polienici.

Publications (3)

Publication Number Publication Date
IT8922396A0 IT8922396A0 (it) 1989-11-16
IT8922396A1 IT8922396A1 (it) 1991-05-16
IT1237772B true IT1237772B (it) 1993-06-17

Family

ID=11195729

Family Applications (1)

Application Number Title Priority Date Filing Date
IT02239689A IT1237772B (it) 1989-11-16 1989-11-16 Derivati di macrolidi polienici.

Country Status (9)

Country Link
US (1) US5296597A (it)
EP (1) EP0434943B1 (it)
JP (1) JP3094065B2 (it)
KR (1) KR0185200B1 (it)
AT (1) ATE127471T1 (it)
DE (1) DE69022196T2 (it)
ES (1) ES2079417T3 (it)
IT (1) IT1237772B (it)
PT (1) PT95910B (it)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1243404B (it) * 1990-12-03 1994-06-10 Prodotti Antibiotici Spa Derivati della partricina
IT1283149B1 (it) * 1996-07-12 1998-04-07 Prodotti Antibiotici Spa Complessi di n'-dimetilaminoacetilpartricina a dimetilaminoetilamide, o suoi sali, e colesterol 3-solfato
IT1294740B1 (it) * 1997-09-16 1999-04-12 Prospa Bv Derivati della partricina per il trattamento profilattico e/o curativo delle contaminazioni fungine di colture cellulari e di tessuti
US6121244A (en) * 1997-09-19 2000-09-19 Prospa B.V. Antitumoral method by administration of partricin derivatives
WO2001051061A1 (en) 2000-01-14 2001-07-19 Intrabiotics Pharmaceuticals, Inc. Derivatives of polyene macrolides and preparation and use thereof
US6664241B2 (en) 2000-05-31 2003-12-16 Micrologix Biotech Inc. Water-soluble amide derivatives of polyene macrolides and preparation and uses thereof
ITMI20032280A1 (it) * 2003-11-24 2005-05-25 Tiberio Bruzzese Formulazioni farmaceutiche contenenti derivati della partricina e loro uso orale per il trattamento di infezioni fungine e protozoarie localizzate
MX365184B (es) * 2010-12-21 2019-05-21 Centro De Investig Y De Estudios Avanzados Del I P N Nuevos compuestos analogos de la anfotericina y composiciones farmaceuticas que los contienen.
GB201409451D0 (en) * 2014-05-28 2014-07-09 Ipabc Ltd Antimicrobial preparations, methods for preparing the same and uses thereof to combat microorganisms

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1406774A (en) * 1973-02-15 1975-09-17 Prodotti Antibiotici Spa Esters of patricin and of partricin derivatives
PL122086B1 (en) * 1979-04-09 1982-06-30 Politechnika Gdanska Process for preparing amides of antibiotics from the group of polyene macrolides and their derivativesvykh makrolidov i ikh proizvodnykh
JP5728715B2 (ja) 2011-08-11 2015-06-03 オリオン機械株式会社 乳量計

Also Published As

Publication number Publication date
IT8922396A0 (it) 1989-11-16
DE69022196T2 (de) 1996-02-01
EP0434943B1 (en) 1995-09-06
JPH03188096A (ja) 1991-08-16
KR0185200B1 (ko) 1999-05-15
IT8922396A1 (it) 1991-05-16
DE69022196D1 (de) 1995-10-12
EP0434943A1 (en) 1991-07-03
KR910009638A (ko) 1991-06-28
ES2079417T3 (es) 1996-01-16
ATE127471T1 (de) 1995-09-15
JP3094065B2 (ja) 2000-10-03
PT95910B (pt) 1998-01-30
PT95910A (pt) 1991-09-13
US5296597A (en) 1994-03-22

Similar Documents

Publication Publication Date Title
YU11997A (sh) Laktamski derivati i njihove farmaceutske kompozicije
ES2085876T3 (es) Derivado de bifenilmetano, su utilizacion y composiciones farmacologicas que contienen el mismo.
DK0582829T3 (da) 9-(Substitueret glycyl)amido-6-demethyl-6-deoxytetracycliner som antibiotiske midler
BR9914221A (pt) Derivados de glicopeptìdeos e composições farmacêuticas contendo os mesmos
LV12358A (lv) 7-(Aizvietoti)-9-(aizvietoti glicil)-amido-6-demetil-6-deoksitetraciklini
ES2067589T3 (es) Derivados de amidas de aminoacidos.
DK0582789T3 (da) Nye (7-substitueret)-8-(substitueret)-9-(substitueret glycyl)amido-6-demethyl-6-deoxytetracycliner
EA199800288A1 (ru) Производные 5-o-дезозаминил-6-o-метилэритронолида а, способ их получения и их применение для получения биологически активных продуктов
ATE158288T1 (de) Antiatherosklerotische und antithrombotische 1- benzopyran-4-on- und 2-amino-1,3-benzoxazin-4-on- derivate
PT688789E (pt) Processo de lipopeptideos processo para a sua preparacao e sua utilizacao
DE69021501D1 (de) Anti-entzündende 4-aminophenol-derivate.
IT1237772B (it) Derivati di macrolidi polienici.
DE69224234D1 (de) 4-a-Substutierte Avermectinderivate
ES2094974T3 (es) Derivados de 17-aril- y 17-heterociclil-14beta-5alfa-androstano, androsteno y androstadieno, activos sobre el sistema cardiovascular, procesos para su preparacion y composiciones farmaceuticas que contienen los mismos.
ES2097297T3 (es) Isoquinolein-5-il-sulfonamidas, su procedimiento de preparacion y las composiciones farmaceuticas que las contienen.
FI101376B1 (fi) Menetelmä 3-bentsyyliamino-2-fenyylipiperidiinijohdannaisten valmistamiseksi
DK81885D0 (da) Pyrido-benzothiazinderivater, fremgangsmaade til fremstilling deraf ogfarmaceutisk praeparat indeholdende mindst et saadant derivat
ES2135429T3 (es) Derivados de ciclohexano sustituidos para el tratamiento de enfermedades.
ES2062215T3 (es) Derivados aminoalcoxibencenicos sustituidos.
GR1001597B (el) Νέα βιολογικώς δραστικά παράγωγα εμπουρναμενίνης, φαρμακευτικές συν?έσεις οι οποίες περιέχουν αυτά και μέ?οδος δια την παρασκευή αυτών.
DK0736029T3 (da) Antikonvulsive pseudofructopyranosesulfamater
IT1301968B1 (it) Derivati di eritromicina ad attivita' antibiotica
UA39870C2 (uk) ПОХІДНІ 9а-N-/N`-КАРБАМOЇЛУ/ ТА 9а-N-/N`-ТІОКАРБАМOЇЛУ/ ВІД 9-ДЕОКСО-9а-А3А-9а ГОМОЕРИТРОМІЦИНУ А, СПОСІБ ОДЕРЖАННЯ ТА ФАРМАЦЕВТИЧНА КОМПОЗИЦІЯ
ES2100396T3 (es) Derivados de 17-(3-furil)- y 17-(4-piridazinil)-5beta,14beta-androstano activos sobre el sistema cardiovascular, procesos para su preparacion y composiciones farmaceuticas que los contienen.
MX9206816A (es) Derivados de cromano substituidos con piperidilmetilo, procedimiento para su obtencion y medicamentoque los contiene.

Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19951026