IT1184285B - Derivati steroidei sostituiti in posizione 11-beta,procedimento per la loro preparazione e loro applicazione come medicamenti - Google Patents

Derivati steroidei sostituiti in posizione 11-beta,procedimento per la loro preparazione e loro applicazione come medicamenti

Info

Publication number
IT1184285B
IT1184285B IT48298/85A IT4829885A IT1184285B IT 1184285 B IT1184285 B IT 1184285B IT 48298/85 A IT48298/85 A IT 48298/85A IT 4829885 A IT4829885 A IT 4829885A IT 1184285 B IT1184285 B IT 1184285B
Authority
IT
Italy
Prior art keywords
medications
procedure
preparation
application
beta position
Prior art date
Application number
IT48298/85A
Other languages
English (en)
Italian (it)
Other versions
IT8548298A0 (it
Inventor
Torelli Vesperto
Jean George Teutsch
Daniel Philibert
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of IT8548298A0 publication Critical patent/IT8548298A0/it
Application granted granted Critical
Publication of IT1184285B publication Critical patent/IT1184285B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • C07J41/0083Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT48298/85A 1984-06-29 1985-06-28 Derivati steroidei sostituiti in posizione 11-beta,procedimento per la loro preparazione e loro applicazione come medicamenti IT1184285B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8410304A FR2566779B2 (fr) 1984-06-29 1984-06-29 Nouveaux derives steroides substitues en 11b, leur procede de preparation et leur application comme medicaments

Publications (2)

Publication Number Publication Date
IT8548298A0 IT8548298A0 (it) 1985-06-28
IT1184285B true IT1184285B (it) 1987-10-22

Family

ID=9305596

Family Applications (1)

Application Number Title Priority Date Filing Date
IT48298/85A IT1184285B (it) 1984-06-29 1985-06-28 Derivati steroidei sostituiti in posizione 11-beta,procedimento per la loro preparazione e loro applicazione come medicamenti

Country Status (7)

Country Link
JP (1) JPS6118798A (nl)
CH (1) CH666277A5 (nl)
DE (1) DE3523297A1 (nl)
FR (1) FR2566779B2 (nl)
GB (1) GB2160873B (nl)
IT (1) IT1184285B (nl)
NL (1) NL8501868A (nl)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3619413C2 (de) * 1986-06-10 2000-04-06 Schering Ag 9alpha, 10alpha-Methylen-Estrene, deren Herstellung und diese enthaltende pharmazeutische Präparate
DE3621024C2 (de) * 1986-06-20 1999-10-28 Schering Ag 11beta-Phenylestradiene, deren Herstellung und diese enthaltende pharmazeutische Präparate
JP2785023B2 (ja) * 1987-12-30 1998-08-13 ルセル―ユクラフ 17α位置を置換された17β―OH―19―ノルステロイドの新誘導体、その製造方法、その薬剤としての使用及びそれを含有する製薬組成物
JP3202224B2 (ja) * 1989-08-04 2001-08-27 シエーリング アクチエンゲゼルシヤフト 11β―アリール―ゴナ―4,9―ジエン―3―オン、その製造方法及びそれを含有する調剤学的調製剤
FR2651233B1 (fr) * 1989-08-23 1991-12-13 Roussel Uclaf Nouveaux acides omega-phenylamino alcanouiques substitues sur le noyau aromatique par un radical derive de 19-norsterouides, leur procede de preparation, leur application a titre de medicaments et les compositions les renfermant.
FR2651435A1 (fr) * 1989-09-07 1991-03-08 Roussel Uclaf Nouvelle utilisation de composes anti-progestomimetiques.
FR2654337B1 (fr) * 1989-11-15 1994-08-05 Roussel Uclaf Nouvelles microspheres injectables biodegradables procede de preparation et suspensions injectables les renfermant.
US5407928A (en) * 1990-08-15 1995-04-18 Schering Aktiengesellschaft 11β-aryl-gona-4,9-dien-3-ones

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2377418A1 (fr) * 1977-01-13 1978-08-11 Roussel Uclaf Nouveaux derives steroides 4,9-dieniques 11b-substitues, leur procede de preparation et leur application comme medicaments
FR2528434B1 (fr) * 1982-06-11 1985-07-19 Roussel Uclaf Nouveaux 19-nor steroides substitues en 11b et eventuellement en 2, leur procede de preparation et leur application comme medicament
ZA8231B (en) * 1981-01-09 1982-11-24 Roussel Uclaf New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained
DE3321826A1 (de) * 1983-06-15 1984-12-20 Schering AG, 1000 Berlin und 4709 Bergkamen 13(alpha)-alkylgonane, deren herstellung und diese enthaltende pharmazeutische praeparate

Also Published As

Publication number Publication date
FR2566779B2 (fr) 1987-03-06
FR2566779A2 (fr) 1986-01-03
JPS6118798A (ja) 1986-01-27
IT8548298A0 (it) 1985-06-28
NL8501868A (nl) 1986-01-16
GB2160873B (en) 1988-03-09
CH666277A5 (fr) 1988-07-15
GB8516387D0 (en) 1985-07-31
DE3523297A1 (de) 1986-01-09
GB2160873A (en) 1986-01-02

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19960517