IS7726A - Pyrazólólpyridín og aðferðir til þess að búa þau til og nota - Google Patents

Pyrazólólpyridín og aðferðir til þess að búa þau til og nota

Info

Publication number
IS7726A
IS7726A IS7726A IS7726A IS7726A IS 7726 A IS7726 A IS 7726A IS 7726 A IS7726 A IS 7726A IS 7726 A IS7726 A IS 7726A IS 7726 A IS7726 A IS 7726A
Authority
IS
Iceland
Prior art keywords
pyrazolol
pyridine
preparation
methods
pyrazolol pyridine
Prior art date
Application number
IS7726A
Other languages
English (en)
Inventor
Lee Wen-Cherng
Lyne Paul
Singh Juswinder
Beth Carter Mary
Chuaqui Claudio
Somerville
Boriack-Sjodin Paula
Sun Lihong
Zheng Zhongli
Original Assignee
Biogen Idec Ma, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biogen Idec Ma, Inc. filed Critical Biogen Idec Ma, Inc.
Publication of IS7726A publication Critical patent/IS7726A/is

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/04Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Oncology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IS7726A 2002-09-06 2005-03-04 Pyrazólólpyridín og aðferðir til þess að búa þau til og nota IS7726A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40881102P 2002-09-06 2002-09-06
PCT/US2003/027722 WO2004022054A1 (en) 2002-09-06 2003-09-05 Pyrazolopyridines and methods of making and using the same

Publications (1)

Publication Number Publication Date
IS7726A true IS7726A (is) 2005-03-04

Family

ID=31978684

Family Applications (2)

Application Number Title Priority Date Filing Date
IS7726A IS7726A (is) 2002-09-06 2005-03-04 Pyrazólólpyridín og aðferðir til þess að búa þau til og nota
IS7725A IS7725A (is) 2002-09-06 2005-03-04 Imidazólópyridín og aðferðir við framleiðslu og notkun þeirra

Family Applications After (1)

Application Number Title Priority Date Filing Date
IS7725A IS7725A (is) 2002-09-06 2005-03-04 Imidazólópyridín og aðferðir við framleiðslu og notkun þeirra

Country Status (20)

Country Link
US (1) US7691865B2 (is)
EP (1) EP1551398A4 (is)
JP (1) JP2006502165A (is)
KR (1) KR20050057235A (is)
CN (1) CN1694698A (is)
AR (1) AR041207A1 (is)
AU (1) AU2003268447B2 (is)
BR (1) BR0314053A (is)
CA (1) CA2497970A1 (is)
EA (1) EA009441B1 (is)
GE (1) GEP20074125B (is)
IS (2) IS7726A (is)
MX (1) MXPA05002443A (is)
NO (1) NO20051503D0 (is)
NZ (1) NZ539069A (is)
PL (1) PL375699A1 (is)
RS (1) RS20050200A (is)
UA (1) UA80295C2 (is)
WO (1) WO2004022054A1 (is)
ZA (1) ZA200501856B (is)

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JP2010540451A (ja) * 2007-09-20 2010-12-24 ワイス・エルエルシー ピラゾロ[5,1−c][1,2,4]トリアジン、その調製法および使用法
TWI436767B (zh) * 2008-03-14 2014-05-11 Otsuka Pharma Co Ltd 基質金屬蛋白酶-2(mmp-2)及/或基質金屬蛋白酶-9(mmp-9)抑制劑
CN101544634B (zh) * 2008-03-27 2011-08-10 天津药物研究院 2-苯基-3-取代吡唑并[1,5-a]吡啶类衍生物及其制备方法和用途
EP2402335A1 (en) * 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
EP2402344A1 (en) * 2010-06-29 2012-01-04 Basf Se Pyrazole fused bicyclic compounds
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KR102455518B1 (ko) * 2014-03-27 2022-10-14 얀센 파마슈티카 엔.브이. ROS1 저해제로서 치환된 4,5,6,7-테트라히드로피라졸로[1,5-a]피리미딘 유도체 및 2,3-디히드로-1H-이미다조[1,2-b]피라졸 유도체
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CN112707902B (zh) * 2020-03-23 2022-04-15 杭州阿诺生物医药科技有限公司 TGF-β受体抑制剂

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CA2497970A1 (en) 2004-03-18
EP1551398A1 (en) 2005-07-13
MXPA05002443A (es) 2005-09-30
EA200500450A1 (ru) 2005-08-25
NZ539069A (en) 2007-03-30
AR041207A1 (es) 2005-05-11
KR20050057235A (ko) 2005-06-16
EA009441B1 (ru) 2007-12-28
WO2004022054A1 (en) 2004-03-18
AU2003268447A1 (en) 2004-03-29
RS20050200A (en) 2007-08-03
US20060106033A1 (en) 2006-05-18
PL375699A1 (en) 2005-12-12
EP1551398A4 (en) 2006-06-07
AU2003268447B2 (en) 2008-07-24
IS7725A (is) 2005-03-04
NO20051503L (no) 2005-03-21
JP2006502165A (ja) 2006-01-19
ZA200501856B (en) 2006-04-26
US7691865B2 (en) 2010-04-06
CN1694698A (zh) 2005-11-09
GEP20074125B (en) 2007-06-11
UA80295C2 (en) 2007-09-10
BR0314053A (pt) 2005-07-19
NO20051503D0 (no) 2005-03-21

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