IS5720A - Latar gegn peptídýli af VLA-4 skilyrtri frumutengingu gagnlegir til meðhöndlunar á bólguvaldandi-, sjálfónæmis, og öndunarsjúkdómum - Google Patents

Latar gegn peptídýli af VLA-4 skilyrtri frumutengingu gagnlegir til meðhöndlunar á bólguvaldandi-, sjálfónæmis, og öndunarsjúkdómum

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Publication number
IS5720A
IS5720A IS5720A IS5720A IS5720A IS 5720 A IS5720 A IS 5720A IS 5720 A IS5720 A IS 5720A IS 5720 A IS5720 A IS 5720A IS 5720 A IS5720 A IS 5720A
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Iceland
Prior art keywords
vla
autoimmune
latency
inflammatory
inhibitors
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IS5720A
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English (en)
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Jacob Duplantier Allen
John Milici Anthony
Stanley Chupak Louis
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Pfizer Products Inc.
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Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of IS5720A publication Critical patent/IS5720A/is

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IS5720A 1998-06-30 2000-11-21 Latar gegn peptídýli af VLA-4 skilyrtri frumutengingu gagnlegir til meðhöndlunar á bólguvaldandi-, sjálfónæmis, og öndunarsjúkdómum IS5720A (is)

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US9118098P 1998-06-30 1998-06-30
PCT/IB1999/000973 WO2000000477A1 (en) 1998-06-30 1999-05-31 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases

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US6518292B1 (en) * 1999-03-12 2003-02-11 Bristol-Myers Squibb Co. Heterocyclic aromatic compounds usefuls as growth hormone secretagogues
US6756378B2 (en) * 1999-06-30 2004-06-29 Pharmacopeia Drug Discovery, Inc. VLA-4 inhibitor compounds
CN1391473A (zh) * 1999-06-30 2003-01-15 第一制药株式会社 Vla-4抑制剂化合物
PL357109A1 (en) 1999-12-28 2004-07-12 Pfizer Products Inc. Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
AU2001234741A1 (en) * 2000-02-04 2001-08-14 Biogen, Inc. Integrin antagonists
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DE10111877A1 (de) * 2001-03-10 2002-09-12 Aventis Pharma Gmbh Neue Imidazolidinderivate, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate
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GB2377933A (en) 2001-07-06 2003-01-29 Bayer Ag Succinic acid derivatives useful as integrin antagonists
DE10137595A1 (de) 2001-08-01 2003-02-13 Aventis Pharma Gmbh Neue Imidazolidinderivate, ihre Herstellung und ihre Verwendung
WO2003024401A2 (en) * 2001-09-18 2003-03-27 Bristol-Myers Squibb Company Piperizinones as modulators of chemokine receptor activity
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WO2004004665A2 (en) * 2002-07-09 2004-01-15 Bristol-Myers Squibb Company Substituted heterocyclic derivatives useful as antidiabetic and antiobesity agents and method
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TW200610754A (en) * 2004-06-14 2006-04-01 Daiichi Seiyaku Co Vla-4 inhibitor
US7453002B2 (en) 2004-06-15 2008-11-18 Bristol-Myers Squibb Company Five-membered heterocycles useful as serine protease inhibitors
JP5107724B2 (ja) 2005-12-13 2012-12-26 第一三共株式会社 Vla−4阻害薬
WO2011020874A1 (en) 2009-08-20 2011-02-24 Inserm (Institut National De La Sante Et De La Recherche Medicale) Vla-4 as a biomarker for prognosis and target for therapy in duchenne muscular dystrophy
AU2018311976B2 (en) 2017-08-04 2022-10-13 Takeda Pharmaceutical Company Limited Inhibitors of Plasma Kallikrein and uses thereof
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PE20000762A1 (es) 2000-08-24
IL139584A0 (en) 2002-02-10
US6306887B1 (en) 2001-10-23
JP2002519344A (ja) 2002-07-02
ID27414A (id) 2001-04-05
EP1091943A1 (en) 2001-04-18
US6355662B1 (en) 2002-03-12
CN1308616A (zh) 2001-08-15
EP1091943B1 (en) 2005-11-30
KR20010083081A (ko) 2001-08-31
GT199900101A (es) 2000-12-16
DE69928667T2 (de) 2006-08-10
UA66864C2 (uk) 2004-06-15
AU758939B2 (en) 2003-04-03
DE69928667D1 (de) 2006-01-05
ATE311371T1 (de) 2005-12-15
MA26640A1 (fr) 2004-12-20
ZA993777B (en) 2000-12-04
JP3676677B2 (ja) 2005-07-27
YU77600A (sh) 2004-03-12
BR9911701A (pt) 2001-03-20
AR015312A1 (es) 2001-04-18
HUP0102477A3 (en) 2002-08-28
NZ508033A (en) 2002-12-20
AU3841699A (en) 2000-01-17
WO2000000477A1 (en) 2000-01-06
TR200003848T2 (tr) 2001-06-21
SK20052000A3 (sk) 2002-08-06
NO20006600L (no) 2001-02-21
CZ20004909A3 (cs) 2002-04-17
NO20006600D0 (no) 2000-12-22
EA200001238A1 (ru) 2001-08-27
BG105190A (en) 2001-12-29
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CO5320599A1 (es) 2003-09-30
PA8477001A1 (es) 2000-05-24
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AP9901561A0 (en) 1999-06-30
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