IN2014MN01575A - - Google Patents

Info

Publication number
IN2014MN01575A
IN2014MN01575A IN1575MUN2014A IN2014MN01575A IN 2014MN01575 A IN2014MN01575 A IN 2014MN01575A IN 1575MUN2014 A IN1575MUN2014 A IN 1575MUN2014A IN 2014MN01575 A IN2014MN01575 A IN 2014MN01575A
Authority
IN
India
Prior art keywords
methyl
pyrido
dimethylbutyl
pyrimidin
methylamino
Prior art date
Application number
Other languages
English (en)
Inventor
Matthew Carl Allgeier
Daniel L Flynn
Michael D Kaufman
Phenil J Patel
Craig D Wolfangel
Original Assignee
Lilly Co Eli
Deciphera Pharmaceuticals Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47884613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014MN01575(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli, Deciphera Pharmaceuticals Llc filed Critical Lilly Co Eli
Publication of IN2014MN01575A publication Critical patent/IN2014MN01575A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
IN1575MUN2014 2012-03-07 2013-03-05 IN2014MN01575A (cg-RX-API-DMAC7.html)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261607702P 2012-03-07 2012-03-07
PCT/US2013/029084 WO2013134243A1 (en) 2012-03-07 2013-03-05 2-amino, 6-phenyl substituted pyrido [2, 3 - d] pyrimidine derivatives useful as raf kinase inhibitors

Publications (1)

Publication Number Publication Date
IN2014MN01575A true IN2014MN01575A (cg-RX-API-DMAC7.html) 2015-05-08

Family

ID=47884613

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1575MUN2014 IN2014MN01575A (cg-RX-API-DMAC7.html) 2012-03-07 2013-03-05

Country Status (39)

Country Link
US (2) US9334267B2 (cg-RX-API-DMAC7.html)
EP (1) EP2850082B1 (cg-RX-API-DMAC7.html)
JP (1) JP2015509536A (cg-RX-API-DMAC7.html)
KR (1) KR20140129087A (cg-RX-API-DMAC7.html)
CN (1) CN104302646B (cg-RX-API-DMAC7.html)
AP (1) AP2014007899A0 (cg-RX-API-DMAC7.html)
AR (1) AR090151A1 (cg-RX-API-DMAC7.html)
AU (1) AU2013230146B2 (cg-RX-API-DMAC7.html)
BR (1) BR112014018528A8 (cg-RX-API-DMAC7.html)
CA (1) CA2863673A1 (cg-RX-API-DMAC7.html)
CL (1) CL2014002220A1 (cg-RX-API-DMAC7.html)
CO (1) CO7010837A2 (cg-RX-API-DMAC7.html)
CR (1) CR20140378A (cg-RX-API-DMAC7.html)
CY (1) CY1117846T1 (cg-RX-API-DMAC7.html)
DK (1) DK2850082T3 (cg-RX-API-DMAC7.html)
DO (1) DOP2014000200A (cg-RX-API-DMAC7.html)
EA (1) EA024824B1 (cg-RX-API-DMAC7.html)
EC (1) ECSP14017584A (cg-RX-API-DMAC7.html)
ES (1) ES2584387T3 (cg-RX-API-DMAC7.html)
HK (1) HK1202541A1 (cg-RX-API-DMAC7.html)
HR (1) HRP20160654T1 (cg-RX-API-DMAC7.html)
HU (1) HUE028095T2 (cg-RX-API-DMAC7.html)
IL (1) IL234052A (cg-RX-API-DMAC7.html)
IN (1) IN2014MN01575A (cg-RX-API-DMAC7.html)
LT (1) LT2850082T (cg-RX-API-DMAC7.html)
MA (1) MA37316B1 (cg-RX-API-DMAC7.html)
ME (1) ME02423B (cg-RX-API-DMAC7.html)
MX (1) MX2014010701A (cg-RX-API-DMAC7.html)
NZ (1) NZ627454A (cg-RX-API-DMAC7.html)
PE (1) PE20142338A1 (cg-RX-API-DMAC7.html)
PH (1) PH12014501986A1 (cg-RX-API-DMAC7.html)
PT (1) PT2850082T (cg-RX-API-DMAC7.html)
RS (1) RS54840B1 (cg-RX-API-DMAC7.html)
SG (1) SG11201404969YA (cg-RX-API-DMAC7.html)
SI (1) SI2850082T1 (cg-RX-API-DMAC7.html)
TN (1) TN2014000375A1 (cg-RX-API-DMAC7.html)
TW (1) TW201348233A (cg-RX-API-DMAC7.html)
UA (1) UA112340C2 (cg-RX-API-DMAC7.html)
WO (2) WO2013134243A1 (cg-RX-API-DMAC7.html)

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CN118903436A (zh) 2018-01-31 2024-11-08 德西费拉制药有限责任公司 治疗肥大细胞增多症的组合疗法
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JP7451543B2 (ja) 2019-02-06 2024-03-18 イーライ リリー アンド カンパニー Kcnq増強剤としての1-((2-(2,2,2-トリフルオロエトキシ)ピリジン-4-イル)メチル)尿素誘導体
TWI756636B (zh) * 2019-02-18 2022-03-01 美商建南德克公司 嘧啶并嘧啶化合物及使用方法
IL330104A (en) 2019-03-11 2026-08-01 Deciphera Pharmaceuticals Llc Crystalline forms of rifatinib
CN114072148A (zh) * 2019-05-03 2022-02-18 金耐特生物制药公司 Raf激酶的抑制剂
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Also Published As

Publication number Publication date
HK1202541A1 (en) 2015-10-02
ES2584387T3 (es) 2016-09-27
HUE028095T2 (en) 2016-11-28
RS54840B1 (sr) 2016-10-31
EP2850082B1 (en) 2016-05-18
CR20140378A (es) 2014-11-27
CA2863673A1 (en) 2013-09-12
NZ627454A (en) 2016-09-30
ECSP14017584A (es) 2016-01-29
PH12014501986B1 (en) 2014-11-24
WO2013134252A1 (en) 2013-09-12
CN104302646A (zh) 2015-01-21
AR090151A1 (es) 2014-10-22
MX2014010701A (es) 2015-03-10
BR112014018528A8 (pt) 2017-07-11
MA37316B1 (fr) 2017-03-31
MA37316A1 (fr) 2016-06-30
JP2015509536A (ja) 2015-03-30
CY1117846T1 (el) 2017-05-17
IL234052A (en) 2016-05-31
AU2013230146A1 (en) 2014-08-14
PT2850082T (pt) 2016-07-15
AP2014007899A0 (en) 2014-08-31
US20150119392A1 (en) 2015-04-30
LT2850082T (lt) 2016-09-12
US20130252977A1 (en) 2013-09-26
US9334267B2 (en) 2016-05-10
DK2850082T3 (en) 2016-08-15
EA201491456A1 (ru) 2014-12-30
PE20142338A1 (es) 2015-01-10
WO2013134243A1 (en) 2013-09-12
UA112340C2 (uk) 2016-08-25
SG11201404969YA (en) 2014-10-30
BR112014018528A2 (cg-RX-API-DMAC7.html) 2017-06-20
EA024824B1 (ru) 2016-10-31
ME02423B (me) 2016-09-20
DOP2014000200A (es) 2014-10-15
TW201348233A (zh) 2013-12-01
US8741911B2 (en) 2014-06-03
TN2014000375A1 (en) 2015-12-21
CN104302646B (zh) 2016-05-04
SI2850082T1 (sl) 2016-07-29
KR20140129087A (ko) 2014-11-06
AU2013230146B2 (en) 2015-09-10
CO7010837A2 (es) 2014-07-31
CL2014002220A1 (es) 2015-06-05
PH12014501986A1 (en) 2014-11-24
HRP20160654T1 (hr) 2016-07-01
EP2850082A1 (en) 2015-03-25

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