IN2014CN04945A - - Google Patents

Info

Publication number
IN2014CN04945A
IN2014CN04945A IN4945CHN2014A IN2014CN04945A IN 2014CN04945 A IN2014CN04945 A IN 2014CN04945A IN 4945CHN2014 A IN4945CHN2014 A IN 4945CHN2014A IN 2014CN04945 A IN2014CN04945 A IN 2014CN04945A
Authority
IN
India
Prior art keywords
formula
sitaxsentan
retains
formulas
represented
Prior art date
Application number
Other languages
English (en)
Inventor
Keigo Tanaka
Tomoki Nishioka
Original Assignee
Eisai R&D Man Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Man Co Ltd filed Critical Eisai R&D Man Co Ltd
Publication of IN2014CN04945A publication Critical patent/IN2014CN04945A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
IN4945CHN2014 2012-01-31 2013-01-29 IN2014CN04945A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261592923P 2012-01-31 2012-01-31
PCT/JP2013/051857 WO2013115162A1 (ja) 2012-01-31 2013-01-29 シタキセンタン誘導体

Publications (1)

Publication Number Publication Date
IN2014CN04945A true IN2014CN04945A (es) 2015-09-18

Family

ID=48870751

Family Applications (1)

Application Number Title Priority Date Filing Date
IN4945CHN2014 IN2014CN04945A (es) 2012-01-31 2013-01-29

Country Status (16)

Country Link
US (1) US8592470B2 (es)
EP (1) EP2810943B1 (es)
JP (1) JP6144631B2 (es)
KR (1) KR101933251B1 (es)
CN (1) CN104039781B (es)
AR (1) AR089838A1 (es)
AU (1) AU2013216122B9 (es)
BR (1) BR112014016204B1 (es)
CA (1) CA2861477C (es)
ES (1) ES2651293T3 (es)
IL (1) IL233171A (es)
IN (1) IN2014CN04945A (es)
MX (1) MX358151B (es)
RU (1) RU2622386C2 (es)
TW (1) TW201336496A (es)
WO (1) WO2013115162A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7531947B2 (ja) 2021-06-22 2024-08-13 株式会社アークメディスン 化合物、エンドセリンa受容体拮抗剤及び医薬組成物
TW202423432A (zh) * 2022-11-11 2024-06-16 日商亞克醫藥股份有限公司 化合物、內皮素a受體拮抗劑、血管收縮素ii第一型受體拮抗劑及醫藥組合物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4861366A (en) 1984-08-27 1989-08-29 E. I. Du Pont De Nemours And Company Herbicidal acetals and ketals
US4659369A (en) 1984-08-27 1987-04-21 E. I. Du Pont De Nemours And Company Herbicidal acetals and ketals
US4753672A (en) 1985-07-16 1988-06-28 E. I. Du Pont De Nemours And Company Herbicidal acetals and ketals
TW224462B (es) * 1992-02-24 1994-06-01 Squibb & Sons Inc
JP3233642B2 (ja) * 1995-04-04 2001-11-26 テキサス・バイオテクノロジー・コーポレイシヨン エンドセリンの活性を調整するチエニル−、フリル−、ピロリル−およびビフェニルスルホンアミドならびにその誘導体
PL197782B1 (pl) * 1999-12-31 2008-04-30 Encysive Pharmaceuticals Inc Sulfonoamidy, środek farmaceutyczny i zastosowanie sulfonoamidów
US20060205733A1 (en) * 2004-08-26 2006-09-14 Encysive Pharmaceuticals Endothelin a receptor antagonists in combination with phosphodiesterase 5 inhibitors and uses thereof
JP2009184924A (ja) 2006-05-31 2009-08-20 Eisai R & D Management Co Ltd 生物学的試薬用化合物
JP2010523694A (ja) * 2007-04-10 2010-07-15 オースペックス・ファーマシューティカルズ・インコーポレイテッド 高血圧治療のための置換重水素濃縮チオフェン

Also Published As

Publication number Publication date
CA2861477A1 (en) 2013-08-08
CA2861477C (en) 2018-01-02
CN104039781B (zh) 2016-08-17
CN104039781A (zh) 2014-09-10
US8592470B2 (en) 2013-11-26
MX2014007619A (es) 2014-09-15
JPWO2013115162A1 (ja) 2015-05-11
AU2013216122B2 (en) 2016-12-08
US20130197045A1 (en) 2013-08-01
KR101933251B1 (ko) 2018-12-27
KR20140117455A (ko) 2014-10-07
BR112014016204B1 (pt) 2020-09-24
ES2651293T3 (es) 2018-01-25
AR089838A1 (es) 2014-09-17
MX358151B (es) 2018-08-07
JP6144631B2 (ja) 2017-06-07
EP2810943B1 (en) 2017-09-27
BR112014016204A2 (pt) 2017-06-13
EP2810943A4 (en) 2015-09-02
IL233171A0 (en) 2014-07-31
RU2014126427A (ru) 2016-03-20
EP2810943A1 (en) 2014-12-10
AU2013216122A1 (en) 2014-07-24
BR112014016204A8 (pt) 2017-07-04
IL233171A (en) 2017-07-31
RU2622386C2 (ru) 2017-06-15
AU2013216122B9 (en) 2017-02-02
WO2013115162A1 (ja) 2013-08-08
TW201336496A (zh) 2013-09-16

Similar Documents

Publication Publication Date Title
CA2875877C (en) Syk inhibitors
PH12014501719A1 (en) Pyridone derivatives
MY180083A (en) Tetrahydropyrrolothiazine compounds
PH12016500169A1 (en) Polymorph of syk inhibitors
RS54526B1 (en) USE OF PIRAZOLOSPIROKETONE DERIVATIVES AS ACETYL-COA CARBOXYLASE INHIBITORS
MX2016006336A (es) Compuestos pirazolopirimidina.
RS53301B (en) TIOACETATE COMPOUNDS, COMPOSITIONS AND USE PROCEDURES
AU2012214029A8 (en) Rorgammat inhibitors
MX2017010735A (es) Inhibidores de inhibidores del factor beta de crecimiento de transformacion (tgf-beta).
IN2014MN01897A (es)
AU2012313888A8 (en) 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH
PH12016500148A1 (en) Plant disease control composition and its use
MA40171A (fr) Dérivés d'azamophinan et leur utilisation
IN2014DN07509A (es)
MX2014002833A (es) Derivados fungicidas de 3-fenil[(heterociclilmetoxi)imino]metil}-1 ,2,4-oxadiazol-5(4h)-ona sustituidos en 4.
RS54730B1 (sr) Inhibitori beta sekretaze
MA40170A (fr) Dérivés hétérocycliques de morphinan et leur utilisation
MX2017000330A (es) Derivado de piridona que tiene un grupo tetrahidropiranilmetilo.
IN2014CN04204A (es)
MA39866A (fr) Amides 2-amino-6-méthyl-4,4a,5,6-tétrahydropyrano[3,4-d][1,3]thiazin-8a(8h)-yl-1,3-thiazol-4-yle
SA517381678B1 (ar) مركبات داي هيدرو بيريميدين-2-أون واستخدامها الطبي
PH12015502429A1 (en) Dicarboxylic acid compound
MY185971A (en) Pyranodipyridine compound
IN2013CN01335A (es)
NZ605804A (en) New aminopyrazoloquinazolines