IN2014CN02346A - - Google Patents
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- Publication number
- IN2014CN02346A IN2014CN02346A IN2346CHN2014A IN2014CN02346A IN 2014CN02346 A IN2014CN02346 A IN 2014CN02346A IN 2346CHN2014 A IN2346CHN2014 A IN 2346CHN2014A IN 2014CN02346 A IN2014CN02346 A IN 2014CN02346A
- Authority
- IN
- India
- Prior art keywords
- carboxamide
- imidazole
- hydroxy
- hydrate
- acidic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2011213501 | 2011-09-28 | ||
| JP2011213500 | 2011-09-28 | ||
| PCT/JP2012/075106 WO2013047758A1 (ja) | 2011-09-28 | 2012-09-28 | ５－ヒドロキシ－１ｈ－イミダゾール－４－カルボキサミド水和物の結晶及び５－ヒドロキシ－１ｈ－イミダゾール－４－カルボキサミド・３／４水和物の結晶及びその製造方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2014CN02346A true IN2014CN02346A (es) | 2015-06-19 |
Family
ID=47995783
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN2346CHN2014 IN2014CN02346A (es) | 2011-09-28 | 2012-09-28 |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US9108928B2 (es) |
| EP (1) | EP2762469B1 (es) |
| KR (1) | KR101970509B1 (es) |
| CN (1) | CN103827093B (es) |
| AU (1) | AU2012317424B2 (es) |
| BR (1) | BR112014007436A2 (es) |
| CA (1) | CA2850196A1 (es) |
| HK (1) | HK1197406A1 (es) |
| IL (2) | IL231677A (es) |
| IN (1) | IN2014CN02346A (es) |
| MX (1) | MX354498B (es) |
| RU (2) | RU2630682C2 (es) |
| SG (1) | SG11201400974VA (es) |
| WO (1) | WO2013047758A1 (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2630682C2 (ru) | 2011-09-28 | 2017-09-12 | Фуджифилм Корпорэйшн | Кристалл 5-гидрокси-1н-имидазол-4-карбоксамид•3/4 гидрата, способ его получения и кристалл 5-гидрокси-1н-имидазол-4-карбоксамида гидрата |
| EP2947069B1 (en) | 2013-01-15 | 2017-11-22 | FUJIFILM Corporation | Sulfate of 5-hydroxy-1h-imidazole-4-carboxamide |
| AU2015205151B2 (en) * | 2014-01-10 | 2018-02-01 | Fujifilm Corporation | 5-hydroxy-1H-imidazole-4-carboxamide effective-dose/sensitivity prediction method and prediction device, xanthosine-monophosphate-amount measurement method, and myelodysplastic-syndrome treatment agent and treatment method |
| WO2018051971A1 (ja) * | 2016-09-13 | 2018-03-22 | 富士フイルム株式会社 | Ｍｌｌ関連白血病の予防または治療のための医薬、方法、使用及び化合物 |
| WO2019082898A1 (ja) | 2017-10-27 | 2019-05-02 | 富士フイルム株式会社 | ５－ヒドロキシ－１ｈ－イミダゾール－４－カルボキサミド・３／４水和物の製造方法 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4181731A (en) * | 1976-09-07 | 1980-01-01 | Sumitomo Chemical Company, Limited | Novel therapeutic application of 4-carbamoyl-5-hydroxyimidazole |
| JPS5625165A (en) * | 1979-08-08 | 1981-03-10 | Sumitomo Chem Co Ltd | Novel imidazole derivative |
| JPS5824569A (ja) | 1981-08-05 | 1983-02-14 | Sumitomo Chem Co Ltd | イミダゾ−ル誘導体の精製方法 |
| US4503235A (en) * | 1983-03-11 | 1985-03-05 | Warner-Lambert Company | Process for producing 4-carbamoyl-1H-imidazolium-5-olate |
| JPS60185727A (ja) * | 1984-03-05 | 1985-09-21 | Sumitomo Chem Co Ltd | ４−カルバモイルイミダゾリウム−５−オレ−ト製剤の安定化法 |
| CA2152863A1 (en) | 1994-07-26 | 1996-01-27 | Yeun-Kwei Han | Preparation of acyclovir |
| US5567816A (en) | 1994-07-26 | 1996-10-22 | Syntex (U.S.A.) Inc. | Preparation of acyclovir using 1,3 dioxolane |
| SI1320527T1 (sl) | 2000-09-29 | 2008-12-31 | Basf Se | Postopek za proizvodnjo 1-substituiranega 5-klor-4 metil pirazolov |
| JP2002265601A (ja) | 2001-03-07 | 2002-09-18 | Rikogaku Shinkokai | イミド樹脂 |
| RU2410377C2 (ru) * | 2005-02-16 | 2011-01-27 | Солвей Фармасьютикалс Б.В. | Производные 1н-имидазола как модуляторы рецептора каннабиноидов св2 |
| CN101395141A (zh) * | 2006-02-24 | 2009-03-25 | 莱西肯医药有限公司 | 咪唑基化合物，包含其的组合物和它们的使用方法 |
| JP5266010B2 (ja) * | 2007-09-14 | 2013-08-21 | 富士フイルム株式会社 | ４−カルバモイル−５−ヒドロキシ−イミダゾール誘導体のスルホン酸塩化合物 |
| KR100982720B1 (ko) * | 2008-02-04 | 2010-09-17 | 주식회사 파마코스텍 | 4-카르바모일-1-β-Ｄ-리보푸라노실이미다졸륨-5-올레이트의 생산을 위한 중간체로서의 2-아미노말론아미드의제조방법 |
| RU2630682C2 (ru) | 2011-09-28 | 2017-09-12 | Фуджифилм Корпорэйшн | Кристалл 5-гидрокси-1н-имидазол-4-карбоксамид•3/4 гидрата, способ его получения и кристалл 5-гидрокси-1н-имидазол-4-карбоксамида гидрата |
| TWI573791B (zh) | 2011-09-28 | 2017-03-11 | 富士軟片股份有限公司 | ５－羥基－１ｈ－咪唑－４－甲醯胺．３／４水合物及其結晶之製造方法 |
-
2012
- 2012-09-28 RU RU2014111810A patent/RU2630682C2/ru not_active IP Right Cessation
- 2012-09-28 CA CA2850196A patent/CA2850196A1/en active Pending
- 2012-09-28 RU RU2017125796A patent/RU2672560C1/ru not_active IP Right Cessation
- 2012-09-28 WO PCT/JP2012/075106 patent/WO2013047758A1/ja active Application Filing
- 2012-09-28 SG SG11201400974VA patent/SG11201400974VA/en unknown
- 2012-09-28 AU AU2012317424A patent/AU2012317424B2/en not_active Ceased
- 2012-09-28 MX MX2014003638A patent/MX354498B/es active IP Right Grant
- 2012-09-28 KR KR1020147008200A patent/KR101970509B1/ko active IP Right Grant
- 2012-09-28 IN IN2346CHN2014 patent/IN2014CN02346A/en unknown
- 2012-09-28 CN CN201280047308.0A patent/CN103827093B/zh not_active Expired - Fee Related
- 2012-09-28 EP EP12835728.2A patent/EP2762469B1/en active Active
- 2012-09-28 BR BR112014007436A patent/BR112014007436A2/pt not_active Application Discontinuation
-
2014
- 2014-03-24 IL IL231677A patent/IL231677A/en active IP Right Grant
- 2014-03-26 US US14/226,364 patent/US9108928B2/en active Active
- 2014-10-30 HK HK14110905.7A patent/HK1197406A1/zh not_active IP Right Cessation
-
2015
- 2015-07-10 US US14/796,602 patent/US9567303B2/en active Active
-
2016
- 2016-07-13 IL IL246754A patent/IL246754A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| BR112014007436A2 (pt) | 2017-04-04 |
| EP2762469A1 (en) | 2014-08-06 |
| KR101970509B1 (ko) | 2019-04-19 |
| SG11201400974VA (en) | 2014-09-26 |
| US20150315156A1 (en) | 2015-11-05 |
| MX2014003638A (es) | 2014-05-21 |
| IL231677A0 (en) | 2014-05-28 |
| EP2762469A4 (en) | 2015-01-14 |
| HK1197406A1 (zh) | 2015-01-16 |
| RU2014111810A (ru) | 2015-11-10 |
| US9567303B2 (en) | 2017-02-14 |
| MX354498B (es) | 2018-03-08 |
| RU2672560C1 (ru) | 2018-11-16 |
| NZ622928A (en) | 2015-04-24 |
| AU2012317424B2 (en) | 2017-05-18 |
| CA2850196A1 (en) | 2013-04-04 |
| AU2012317424A8 (en) | 2014-07-03 |
| WO2013047758A1 (ja) | 2013-04-04 |
| KR20140069052A (ko) | 2014-06-09 |
| CN103827093A (zh) | 2014-05-28 |
| EP2762469B1 (en) | 2016-11-23 |
| IL246754A (en) | 2017-08-31 |
| IL231677A (en) | 2017-01-31 |
| RU2630682C2 (ru) | 2017-09-12 |
| US20140275568A1 (en) | 2014-09-18 |
| CN103827093B (zh) | 2016-06-15 |
| US9108928B2 (en) | 2015-08-18 |
| AU2012317424A1 (en) | 2014-04-17 |
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