IN2012DN00539A - - Google Patents

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Publication number
IN2012DN00539A
IN2012DN00539A IN539DEN2012A IN2012DN00539A IN 2012DN00539 A IN2012DN00539 A IN 2012DN00539A IN 539DEN2012 A IN539DEN2012 A IN 539DEN2012A IN 2012DN00539 A IN2012DN00539 A IN 2012DN00539A
Authority
IN
India
Prior art keywords
fluoropyrimidinones
fungicides
acyl
derivatives
compounds
Prior art date
Application number
Other languages
English (en)
Inventor
Boebel Timothy
Bryan Kristy
Lorsbach Beth
Martin Timothy
Owen W
Pobanz Mark
Thornburgh Scott
Webster Jeffery
Yao Chenglin
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2012DN00539(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of IN2012DN00539A publication Critical patent/IN2012DN00539A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IN539DEN2012 2009-08-07 2010-08-05 IN2012DN00539A (en:Method)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
IN2012DN00539A true IN2012DN00539A (en:Method) 2015-06-12

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
IN539DEN2012 IN2012DN00539A (en:Method) 2009-08-07 2010-08-05

Country Status (33)

Country Link
US (1) US8470839B2 (en:Method)
EP (1) EP2519512B1 (en:Method)
JP (1) JP5748754B2 (en:Method)
KR (1) KR101792285B1 (en:Method)
CN (1) CN102548981B (en:Method)
AU (1) AU2010279402B2 (en:Method)
BR (1) BR112012002810B1 (en:Method)
CA (1) CA2768510C (en:Method)
CL (1) CL2012000316A1 (en:Method)
CO (1) CO6491117A2 (en:Method)
CR (1) CR20120030A (en:Method)
CY (1) CY1122115T1 (en:Method)
DK (1) DK2519512T3 (en:Method)
EA (1) EA023411B1 (en:Method)
EC (1) ECSP12011653A (en:Method)
ES (1) ES2728966T3 (en:Method)
HN (1) HN2012000269A (en:Method)
HR (1) HRP20190919T1 (en:Method)
HU (1) HUE045290T2 (en:Method)
IL (1) IL217952A (en:Method)
IN (1) IN2012DN00539A (en:Method)
LT (1) LT2519512T (en:Method)
MX (1) MX2012001620A (en:Method)
NI (1) NI201200022A (en:Method)
NZ (1) NZ597570A (en:Method)
PE (1) PE20120688A1 (en:Method)
PL (1) PL2519512T3 (en:Method)
PT (1) PT2519512T (en:Method)
SI (1) SI2519512T1 (en:Method)
TR (1) TR201908180T4 (en:Method)
UA (1) UA106889C2 (en:Method)
WO (1) WO2011017538A1 (en:Method)
ZA (1) ZA201200819B (en:Method)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2769073C (en) * 2009-08-07 2018-07-24 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
CN103874413B (zh) * 2011-08-17 2017-03-08 阿达玛马克西姆股份有限公司 5‑氟‑4‑亚氨基‑3‑(取代的)‑3,4‑二氢嘧啶‑2(1h)酮衍生物
CN110003118A (zh) 2012-12-28 2019-07-12 阿达玛马克西姆股份有限公司 制备羧酸酯衍生物的方法
CA2893776A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
KR20150100869A (ko) 2012-12-28 2015-09-02 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복스아미드 유도체
CA2894553C (en) * 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
SG11201605372QA (en) 2013-12-31 2016-08-30 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
HUE072634T2 (hu) 2013-12-31 2025-11-28 Adama Makhteshim Ltd Szinergikus fungicid keverékek gomba elleni védekezésre gabonafélékben
US10011617B2 (en) 2014-09-26 2018-07-03 The Chemours Company Fc, Llc Isocyanate derived organosilanes
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
MA54148A (fr) 2018-11-05 2022-02-09 Adama Makhteshim Ltd Mélanges et compositions comprenant de la 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one et leurs procédés d'utilisation
TWI808347B (zh) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (en:Method) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
MX9800136A (es) 1995-07-05 1998-03-29 Du Pont Pirimidinonas fungicidas.
US6262058B1 (en) 1996-03-11 2001-07-17 Syngenta Crop Protection, Inc. Pyrimidin-4-one derivatives as pesticide
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
EP1731523A4 (en) 2004-04-01 2009-08-12 Takeda Pharmaceutical THIAZOLOPYRIMIDINDERIVAT
WO2008005303A2 (en) 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
PT2562162E (pt) 2008-01-22 2015-10-21 Dow Agrosciences Llc Derivados de n-ciano-4-amino-5-fluoro-pirimidina como fungicidas
JP5580310B2 (ja) 2008-08-01 2014-08-27 ダウ アグロサイエンシィズ エルエルシー 殺真菌剤としての5−フルオロシトシンの使用
PT2389375E (pt) 2009-01-23 2015-09-17 Euro Celtique Sa Derivados de ácido hidroxâmico
CA2769073C (en) 2009-08-07 2018-07-24 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives

Also Published As

Publication number Publication date
NI201200022A (es) 2012-05-22
CN102548981A (zh) 2012-07-04
US20110034490A1 (en) 2011-02-10
AU2010279402A1 (en) 2012-02-02
ES2728966T3 (es) 2019-10-29
WO2011017538A1 (en) 2011-02-10
HK1172894A1 (en) 2013-05-03
UA106889C2 (uk) 2014-10-27
NZ597570A (en) 2014-04-30
DK2519512T3 (da) 2019-05-27
TR201908180T4 (tr) 2019-06-21
JP5748754B2 (ja) 2015-07-15
US8470839B2 (en) 2013-06-25
JP2013501723A (ja) 2013-01-17
PE20120688A1 (es) 2012-06-06
ZA201200819B (en) 2013-05-29
EP2519512A1 (en) 2012-11-07
BR112012002810A2 (pt) 2015-09-15
SI2519512T1 (sl) 2019-09-30
PL2519512T3 (pl) 2019-09-30
CL2012000316A1 (es) 2014-06-27
MX2012001620A (es) 2012-04-11
IL217952A (en) 2017-11-30
IL217952A0 (en) 2012-03-29
EP2519512B1 (en) 2019-03-20
KR20120041786A (ko) 2012-05-02
BR112012002810B1 (pt) 2018-12-11
CY1122115T1 (el) 2020-11-25
EA201270253A1 (ru) 2012-07-30
CN102548981B (zh) 2015-05-13
EA023411B1 (ru) 2016-06-30
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
HRP20190919T1 (hr) 2019-09-20
CA2768510A1 (en) 2011-02-10
KR101792285B1 (ko) 2017-10-31
AU2010279402B2 (en) 2015-04-16
CA2768510C (en) 2018-05-15
CR20120030A (es) 2012-03-28
EP2519512A4 (en) 2013-01-16
CO6491117A2 (es) 2012-07-31
PT2519512T (pt) 2019-06-04
LT2519512T (lt) 2019-07-25
HN2012000269A (es) 2015-04-27

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