IL90552A - History of 3-oxo-propanitrile compressed pyrizole, their preparation and pharmaceutical preparations containing them - Google Patents

History of 3-oxo-propanitrile compressed pyrizole, their preparation and pharmaceutical preparations containing them

Info

Publication number
IL90552A
IL90552A IL9055289A IL9055289A IL90552A IL 90552 A IL90552 A IL 90552A IL 9055289 A IL9055289 A IL 9055289A IL 9055289 A IL9055289 A IL 9055289A IL 90552 A IL90552 A IL 90552A
Authority
IL
Israel
Prior art keywords
phenyl
group
oxo
cyano
dihydro
Prior art date
Application number
IL9055289A
Other languages
English (en)
Hebrew (he)
Other versions
IL90552A0 (en
Inventor
Gianfederico Doria
Anna Maria Isetta
Mario Ferrari
Domenico Trizio
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of IL90552A0 publication Critical patent/IL90552A0/xx
Publication of IL90552A publication Critical patent/IL90552A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cosmetics (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
IL9055289A 1988-06-20 1989-06-07 History of 3-oxo-propanitrile compressed pyrizole, their preparation and pharmaceutical preparations containing them IL90552A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888814587A GB8814587D0 (en) 1988-06-20 1988-06-20 Condensed pyrazole 3-oxo-propanenitrile derivatives & process for their preparation

Publications (2)

Publication Number Publication Date
IL90552A0 IL90552A0 (en) 1990-01-18
IL90552A true IL90552A (en) 1994-08-26

Family

ID=10638992

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9055289A IL90552A (en) 1988-06-20 1989-06-07 History of 3-oxo-propanitrile compressed pyrizole, their preparation and pharmaceutical preparations containing them

Country Status (21)

Country Link
US (1) US5424308A (de)
EP (2) EP0422051A1 (de)
JP (1) JPH03505205A (de)
KR (1) KR900701756A (de)
CN (1) CN1022322C (de)
AT (1) ATE88700T1 (de)
AU (1) AU634966B2 (de)
CZ (1) CZ284336B6 (de)
DE (1) DE68906200T2 (de)
DK (1) DK163581C (de)
ES (1) ES2054930T3 (de)
GB (1) GB8814587D0 (de)
HU (1) HU206872B (de)
IE (1) IE63189B1 (de)
IL (1) IL90552A (de)
NZ (1) NZ229450A (de)
PT (1) PT90905B (de)
RU (1) RU2109735C1 (de)
WO (1) WO1989012630A1 (de)
YU (1) YU46937B (de)
ZA (1) ZA894678B (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8907799D0 (en) * 1989-04-06 1989-05-17 Erba Carlo Spa Heteroaryl-3-oxo-propanenitrile derivatives useful in the treatment of rheumatoid arthritis and other autoimmune diseases
US5260328A (en) * 1989-04-06 1993-11-09 Farmitalia Carlo Erba Srl Phenyl-indenopurazol 3-oxo-propanamide derivatives useful in the treatment of rheumatoid arthritis
GB8916290D0 (en) * 1989-07-17 1989-08-31 Erba Carlo Spa Heteroaryl-3-oxo-propanenitrile derivatives useful in stimulating myelopoiesis
US6492411B1 (en) 1993-11-30 2002-12-10 G. D. Searle & Co. Substituted pyrazolyl benzenesulfonamides for the treatment of inflammation
US5466823A (en) 1993-11-30 1995-11-14 G.D. Searle & Co. Substituted pyrazolyl benzenesulfonamides
ES2193609T3 (es) * 1993-11-30 2003-11-01 Searle & Co Pirazolil-bencenosulfonamidas sustituidas y su uso como inhibidores de la ciclooxigenasa ii.
US6716991B1 (en) 1993-11-30 2004-04-06 G. D. Searle & Co. Process for preparing a substituted pyrazolyl benzenesulfonamide for the treatment of inflammation
US5547975A (en) * 1994-09-20 1996-08-20 Talley; John J. Benzopyranopyrazolyl derivatives for the treatment of inflammation
US5886016A (en) * 1995-09-15 1999-03-23 G.D. Searle & Co. Benzopyranopyrazolyl derivatives for the treatment of inflammation
US5756529A (en) * 1995-09-29 1998-05-26 G.D. Searle & Co. Substituted pyrazolyl benzenesulfonamides for use in veterinary therapies
GB9716103D0 (en) * 1997-07-30 1997-10-01 Pharmacia & Upjohn Spa Condensed heterocyclic compounds
EP1427706B1 (de) 2001-09-19 2007-05-30 Pharmacia Corporation Substituierte pyrazoloverbindungen zur behandlung von entzündungen
CA2461567C (en) 2001-09-19 2008-08-19 Pharmacia Corporation Substituted pyrazolyl benzenesulfamide compounds for the treatment of inflammation
JP2005506983A (ja) 2001-09-19 2005-03-10 ファルマシア・コーポレーション 炎症の治療のための置換ピラゾリル化合物
CN114718407A (zh) * 2022-03-01 2022-07-08 东风柳州汽车有限公司 车窗控制方法、装置、设备及存储介质

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2989538A (en) * 1960-02-10 1961-06-20 Smith Kline French Lab Process for preparing pyrazoloindenone hydrazones
US3004983A (en) * 1960-05-16 1961-10-17 Smith Kline French Lab 4-aminopyrazolo [3, 4-a] indene derivatives
US4140785A (en) * 1978-05-08 1979-02-20 E. I. Du Pont De Nemours And Company N-(benzothienopyrazol)amide antirhinoviral agents
US4173634A (en) * 1979-02-23 1979-11-06 E. R. Squibb & Sons, Inc. Basically-substituted tricyclic pyrazoles useful as antiinflammatory agents
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
US4420476A (en) * 1982-05-24 1983-12-13 Averst McKenna & Harrison, Inc. Benzofuro[3,2-c]pyrazol-3-amine derivatives
US4816467A (en) * 1987-01-09 1989-03-28 Farmitalia Carlo Erba S.R.L Heteroaryl 3-oxo-propanenitrile derivatives, pharmaceutical compositions and use
ES2061644T3 (es) * 1987-04-09 1994-12-16 Du Pont Indazoles sustituidos insecticidas.
GB8814586D0 (en) * 1988-06-20 1988-07-27 Erba Carlo Spa Tricyclic 3-oxo-propanenitrile derivatives & process for their preparation
GB8916290D0 (en) * 1989-07-17 1989-08-31 Erba Carlo Spa Heteroaryl-3-oxo-propanenitrile derivatives useful in stimulating myelopoiesis

Also Published As

Publication number Publication date
PT90905B (pt) 1994-12-30
KR900701756A (ko) 1990-12-04
CZ284336B6 (cs) 1998-10-14
CN1038642A (zh) 1990-01-10
ATE88700T1 (de) 1993-05-15
IL90552A0 (en) 1990-01-18
YU46937B (sh) 1994-06-24
ZA894678B (en) 1991-02-27
DE68906200D1 (de) 1993-06-03
DK300890D0 (da) 1990-12-19
CN1022322C (zh) 1993-10-06
YU125489A (en) 1991-04-30
EP0347773B1 (de) 1993-04-28
DK163581B (da) 1992-03-16
DK163581C (da) 1992-08-10
DE68906200T2 (de) 1993-08-05
HUT56076A (en) 1991-07-29
CZ370189A3 (cs) 1998-07-15
JPH03505205A (ja) 1991-11-14
NZ229450A (en) 1990-08-28
EP0422051A1 (de) 1991-04-17
HU894019D0 (en) 1991-06-28
IE63189B1 (en) 1995-03-22
US5424308A (en) 1995-06-13
GB8814587D0 (en) 1988-07-27
ES2054930T3 (es) 1994-08-16
AU3769289A (en) 1990-01-12
AU634966B2 (en) 1993-03-11
DK300890A (da) 1991-02-20
PT90905A (pt) 1989-12-29
RU2109735C1 (ru) 1998-04-27
HU206872B (en) 1993-01-28
WO1989012630A1 (en) 1989-12-28
EP0347773A1 (de) 1989-12-27

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