IL86788A - N-(4-piperidinyl)bicyclic condensed 2-imidazolamine derivatives,their preparation and pharmaceutical compositions containing them - Google Patents
N-(4-piperidinyl)bicyclic condensed 2-imidazolamine derivatives,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL86788A IL86788A IL86788A IL8678888A IL86788A IL 86788 A IL86788 A IL 86788A IL 86788 A IL86788 A IL 86788A IL 8678888 A IL8678888 A IL 8678888A IL 86788 A IL86788 A IL 86788A
- Authority
- IL
- Israel
- Prior art keywords
- pharmaceutical compositions
- alk
- piperidinyl
- compositions containing
- 6alkyl
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- DEPDDPLQZYCHOH-UHFFFAOYSA-N 1h-imidazol-2-amine Chemical class NC1=NC=CN1 DEPDDPLQZYCHOH-UHFFFAOYSA-N 0.000 title abstract 2
- 125000002619 bicyclic group Chemical group 0.000 title abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 3
- 239000002253 acid Substances 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000000739 antihistaminic agent Substances 0.000 abstract 1
- 229940125715 antihistaminic agent Drugs 0.000 abstract 1
- 125000002541 furyl group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000002883 imidazolyl group Chemical group 0.000 abstract 1
- 125000003373 pyrazinyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000000335 thiazolyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
- Lubricants (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6389987A | 1987-06-19 | 1987-06-19 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL86788A0 IL86788A0 (en) | 1988-11-30 |
| IL86788A true IL86788A (en) | 1992-08-18 |
Family
ID=22052235
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL86788A IL86788A (en) | 1987-06-19 | 1988-06-17 | N-(4-piperidinyl)bicyclic condensed 2-imidazolamine derivatives,their preparation and pharmaceutical compositions containing them |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US4897401A (de) |
| EP (1) | EP0295742B1 (de) |
| JP (1) | JP2609464B2 (de) |
| KR (1) | KR970001158B1 (de) |
| CN (1) | CN1029964C (de) |
| AT (1) | ATE79878T1 (de) |
| AU (1) | AU600144B2 (de) |
| CA (1) | CA1324133C (de) |
| DE (1) | DE3874013T2 (de) |
| DK (1) | DK169761B1 (de) |
| ES (1) | ES2045083T3 (de) |
| FI (1) | FI90233C (de) |
| GR (1) | GR3006205T3 (de) |
| HU (1) | HU201755B (de) |
| IE (1) | IE61728B1 (de) |
| IL (1) | IL86788A (de) |
| NO (1) | NO167803C (de) |
| NZ (1) | NZ224928A (de) |
| PH (1) | PH25532A (de) |
| PT (1) | PT87742B (de) |
| SU (1) | SU1644717A3 (de) |
| ZA (1) | ZA884346B (de) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8716313D0 (en) * | 1987-07-10 | 1987-08-19 | Janssen Pharmaceutica Nv | 2-(heterocyclylalkyl)imidazopyridines |
| GB8900380D0 (en) * | 1989-01-09 | 1989-03-08 | Janssen Pharmaceutica Nv | 2-aminopyrimidinone derivatives |
| US5272150A (en) * | 1989-04-07 | 1993-12-21 | Janssen Pharmaceutica N.V. | Hydroxyalkylfuranyl derivatives |
| PH30434A (en) * | 1989-04-07 | 1997-05-09 | Janssen Pharmaceutica Nv | Hydroxyalkylfuranyl derivatives |
| KR100190299B1 (ko) * | 1990-07-19 | 1999-06-01 | 디르크 반테 | 신규한 옥사졸릴 유도체 |
| US5217980A (en) * | 1990-07-19 | 1993-06-08 | Janssen Pharmaceutica N.V. | Oxazolyl and piperidinyl substituted benimidazolyl compounds |
| NZ238863A (en) * | 1990-07-19 | 1993-03-26 | Janssen Pharmaceutica Nv | Substituted thiazolyl and pyridinyl derivatives |
| US5478858A (en) * | 1993-12-17 | 1995-12-26 | The Procter & Gamble Company | 5-(2-imidazolinylamino) benzimidazole compounds useful as alpha-2 adrenoceptor agonists |
| FR2725986B1 (fr) * | 1994-10-21 | 1996-11-29 | Adir | Nouveaux derives de piperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| EP1400519B1 (de) * | 1999-06-28 | 2007-03-07 | Janssen Pharmaceutica N.V. | Hemmer des Respiratorischen Syncytial Virus |
| ATE258928T1 (de) | 1999-06-28 | 2004-02-15 | Janssen Pharmaceutica Nv | Respiratorisches syncytialvirus replikation inhibitoren |
| EP1418175A1 (de) | 1999-06-28 | 2004-05-12 | Janssen Pharmaceutica N.V. | Replikationsinhibitoren des respiratorischen Synzytialvirus |
| JP2004525109A (ja) | 2001-02-15 | 2004-08-19 | キング・ファーマシューティカルズ・インコーポレイティッド | 安定化された甲状腺ホルモン医薬組成物、及びその製法 |
| US7101569B2 (en) | 2001-08-14 | 2006-09-05 | Franz G Andrew | Methods of administering levothyroxine pharmaceutical compositions |
| EP1479676A1 (de) * | 2003-05-19 | 2004-11-24 | Aventis Pharma Deutschland GmbH | Benzimidazolderivate als Faktor Xa-Inhibitoren |
| WO2004113322A1 (en) * | 2003-06-24 | 2004-12-29 | Pfizer Products Inc. | Processes for the preparation of 1-[(benzoimidazole-1yl) quinolin-8-yl] piperidin-4-ylamine derivatives |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4219559A (en) * | 1979-01-10 | 1980-08-26 | Janssen Pharmaceutica N.V. | N-Heterocyclyl-4-piperidinamines |
| US4556660A (en) * | 1982-07-12 | 1985-12-03 | Janssen Pharmaceutica N.V. | N-(Bicyclic heterocyclyl)-4-piperidinamines |
| US4634704A (en) * | 1983-10-06 | 1987-01-06 | Janssen Pharmaceutica, N.V. | Anti-allergic five membered heterocyclic ring containing N-(bicyclic heterocycyl)-4-piperidinamines |
| US4695569A (en) * | 1983-11-30 | 1987-09-22 | Janssen Pharmaceutica N.V. | Bicyclic heterocyclyl containing N-(bicyclic heterocyclyl)-4-piperidinamines |
| US4588722A (en) * | 1984-01-09 | 1986-05-13 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives |
| CA1327579C (en) * | 1986-02-03 | 1994-03-08 | Frans Eduard Janssens | Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines |
| CA1317939C (en) * | 1987-07-01 | 1993-05-18 | Janssen Pharmaceutica Naamloze Vennootschap | ¬(bicyclic heterocyclyl)methyl and -hetero| substituted hexahydro-1h-azepines and pyrrolidines |
-
1988
- 1988-04-18 US US07/182,814 patent/US4897401A/en not_active Expired - Lifetime
- 1988-05-05 CA CA000565978A patent/CA1324133C/en not_active Expired - Fee Related
- 1988-06-07 NZ NZ224928A patent/NZ224928A/en unknown
- 1988-06-08 EP EP88201172A patent/EP0295742B1/de not_active Expired - Lifetime
- 1988-06-08 AT AT88201172T patent/ATE79878T1/de active
- 1988-06-08 DE DE8888201172T patent/DE3874013T2/de not_active Expired - Fee Related
- 1988-06-08 ES ES88201172T patent/ES2045083T3/es not_active Expired - Lifetime
- 1988-06-14 SU SU884355903A patent/SU1644717A3/ru active
- 1988-06-15 JP JP63145933A patent/JP2609464B2/ja not_active Expired - Fee Related
- 1988-06-15 NO NO882641A patent/NO167803C/no unknown
- 1988-06-16 PT PT87742A patent/PT87742B/pt not_active IP Right Cessation
- 1988-06-17 DK DK333288A patent/DK169761B1/da not_active IP Right Cessation
- 1988-06-17 HU HU883118A patent/HU201755B/hu not_active IP Right Cessation
- 1988-06-17 CN CN88103784A patent/CN1029964C/zh not_active Expired - Fee Related
- 1988-06-17 IL IL86788A patent/IL86788A/xx not_active IP Right Cessation
- 1988-06-17 AU AU18109/88A patent/AU600144B2/en not_active Ceased
- 1988-06-17 KR KR1019880007315A patent/KR970001158B1/ko not_active Expired - Fee Related
- 1988-06-17 ZA ZA884346A patent/ZA884346B/xx unknown
- 1988-06-17 IE IE184988A patent/IE61728B1/en not_active IP Right Cessation
- 1988-06-17 PH PH37085A patent/PH25532A/en unknown
- 1988-06-17 FI FI882909A patent/FI90233C/fi not_active IP Right Cessation
-
1992
- 1992-11-11 GR GR920402534T patent/GR3006205T3/el unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL92730A0 (en) | 2-aminopyrimidinone derivatives,their preparation and pharmaceutical compositions containing them | |
| IL92208A0 (en) | 3-piperidinyl-1,2-benzisoxazoles,their preparation and pharmaceutical compositions containing them | |
| IL86788A0 (en) | N-(4-piperidinyl)bicyclic condensed 2-imidazolamine derivatives,their preparation and pharmaceutical compositions containing them | |
| HU900063D0 (en) | Process for preparation of new 2-amino-pyrimidinone-derivatives | |
| IL91194A0 (en) | 3-piperazinylbenzazole derivatives,their preparation and pharmaceutical compositions containing them | |
| NO176608C (no) | Analogifremgangsmåte for fremstilling av terapeutisk aktive 3-piperidinylindazol-derivater |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RH | Patent void |