IL71617A0 - - Google Patents
Info
- Publication number
- IL71617A0 IL71617A0 IL8471617A IL7161784A IL71617A0 IL 71617 A0 IL71617 A0 IL 71617A0 IL 8471617 A IL8471617 A IL 8471617A IL 7161784 A IL7161784 A IL 7161784A IL 71617 A0 IL71617 A0 IL 71617A0
- Authority
- IL
- Israel
- Prior art keywords
- sup
- aralkyl
- formula
- lower alkyl
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Saccharide Compounds (AREA)
- External Artificial Organs (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/JP1983/000127 WO1984004306A1 (en) | 1983-04-22 | 1983-04-22 | Fused 7-membered ring compounds and process for their preparation |
| PCT/JP1983/000342 WO1985001730A1 (en) | 1983-10-13 | 1983-10-13 | Fused 7-membered ring compounds and process for their preparation |
| PCT/JP1984/000119 WO1985004402A1 (en) | 1984-03-24 | 1984-03-24 | Fused 7-membered ring compounds and process for their preparation |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL71617A0 true IL71617A0 (es) | 1984-07-31 |
| IL71617A IL71617A (en) | 1988-05-31 |
Family
ID=27304084
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL71617A IL71617A (en) | 1983-04-22 | 1984-04-22 | 3-(amino-1-carboxylalkyl)amino-4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepine-5-acetic acid derivatives,method for producing them and pharmaceutical compositions containing them |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4564612A (es) |
| EP (1) | EP0125056B1 (es) |
| KR (1) | KR910007965B1 (es) |
| AT (1) | ATE60061T1 (es) |
| AU (1) | AU565188B2 (es) |
| CA (1) | CA1209993A (es) |
| DE (1) | DE3483920D1 (es) |
| ES (2) | ES8602699A1 (es) |
| FI (1) | FI82455C (es) |
| GR (1) | GR79905B (es) |
| HU (1) | HU193008B (es) |
| IE (1) | IE57599B1 (es) |
| IL (1) | IL71617A (es) |
| NO (1) | NO162235C (es) |
| NZ (1) | NZ207915A (es) |
| PH (1) | PH21294A (es) |
| PT (1) | PT78454B (es) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1176345B (it) * | 1983-06-29 | 1987-08-18 | Mitsui Toatsu Chemicals | Derivati benzotiazepinici e loro metodo di preparazione |
| AU570710B2 (en) * | 1983-08-12 | 1988-03-24 | Takeda Chemical Industries Ltd. | 4-oxo-2, 3, 4, 5-tetrahydro-1, 5-benzoxazepine derivatives |
| US4512988A (en) * | 1984-03-01 | 1985-04-23 | E. R. Squibb & Sons, Inc. | Acylamino oxo or hydroxy substituted alkylamino thiazines and thiazepines |
| NO160712C (no) * | 1984-03-24 | 1989-05-24 | Takeda Chemical Industries Ltd | Analogifremgangsmaate for fremstilling av terapeutisk aktive benzotiazepin-forbindelser. |
| EP0187037A3 (en) * | 1984-12-21 | 1988-03-23 | Takeda Chemical Industries, Ltd. | Piperidine derivatives, their production and use |
| US4692522A (en) * | 1985-04-01 | 1987-09-08 | Merck & Co., Inc. | Benzofused lactams useful as cholecystokinin antagonists |
| JPH0657707B2 (ja) * | 1987-05-25 | 1994-08-03 | 吉富製薬株式会社 | ピペリジン化合物 |
| JPS6450872A (en) * | 1987-08-21 | 1989-02-27 | Tanabe Seiyaku Co | Production of 1,5-benzothiazepine derivative |
| EP0322779A3 (en) * | 1987-12-29 | 1991-05-08 | Yoshitomi Pharmaceutical Industries, Ltd. | Benzolactam compounds and pharmaceutical uses thereof |
| US5290927A (en) * | 1988-03-01 | 1994-03-01 | Ajinomoto Co., Inc. | Process for preparing 2',3'-dideoxyadenosine |
| AT393998B (de) * | 1990-02-16 | 1992-01-10 | Troendle Peter Paul | Buch |
| EP0648213A1 (en) * | 1992-07-01 | 1995-04-19 | Pfizer Inc. | Benzothiazepine and benzoxazepine derivatives as cholecystokinin receptor antagonists |
| IL108633A (en) * | 1993-02-15 | 1998-07-15 | Wellcome Found | History of Benzothiazepine Hypolipidemic Preparation and Pharmaceutical Preparations Containing Them |
| ZA956647B (en) * | 1994-08-10 | 1997-02-10 | Wellcome Found | Hypolipidaemic compounds. |
| FR2781483A1 (fr) * | 1998-07-21 | 2000-01-28 | Hoechst Marion Roussel Inc | Derives de thioazepinone, procede de preparation et intermediaires de ce procede, application a titre de medicament et compositions pharmaceutiques les renfermant |
| FR2807039A1 (fr) * | 2000-03-31 | 2001-10-05 | Adir | NOUVEAU PROCEDE DE PREPARATION DE LA 11-AMINO-3-CHLORO-6,11- DIHYDRO-5,5-DIOXO-6-METHYL-DIBENZO[c,f][1,2]-THIAZEPINE ET APPLICATION A LA SYNTHESE DE LA TIANEPTINE |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3341519A (en) * | 1965-04-28 | 1967-09-12 | Squibb & Sons Inc | Novel benzoxazines, benzothiazines, benzoxazepins and benzothiazepins |
| AU543804B2 (en) * | 1980-10-31 | 1985-05-02 | Takeda Chemical Industries Ltd. | Amides having bicyclic substituents on nitrogen |
| DE3260505D1 (en) * | 1981-01-23 | 1984-09-13 | Takeda Chemical Industries Ltd | Alicyclic compounds, their production and use |
| DE3260831D1 (en) * | 1981-06-05 | 1984-10-31 | Merck & Co Inc | Perhydro-1,4-thiazepin-5-one and perhydro-1,4-thiazocin-5-one derivatives, process for preparing and pharmceutical composition containing the same |
| EP0072352B1 (de) * | 1981-08-11 | 1986-03-05 | Ciba-Geigy Ag | Benzazepin-2-one, Verfahren zu ihrer Herstellung, pharmazeutische Präparate die diese Verbindungen enthalten, sowie die Verbindungen zur therapeutischen Verwendung |
| JPS5829779A (ja) * | 1981-08-17 | 1983-02-22 | Nippon Iyakuhin Kogyo Kk | Ｎ−アミノアルキル−１，５−ベンゾチアゼピン誘導体の製造法 |
| US4477464A (en) * | 1983-02-10 | 1984-10-16 | Ciba-Geigy Corporation | Hetero-benzazepine derivatives and their pharmaceutical use |
| US4460579A (en) * | 1983-02-28 | 1984-07-17 | E. R. Squibb & Sons, Inc. | Thiazine and thiazepine containing compounds |
| IT1176345B (it) * | 1983-06-29 | 1987-08-18 | Mitsui Toatsu Chemicals | Derivati benzotiazepinici e loro metodo di preparazione |
-
1984
- 1984-04-11 US US06/599,187 patent/US4564612A/en not_active Expired - Fee Related
- 1984-04-13 AT AT84302564T patent/ATE60061T1/de not_active IP Right Cessation
- 1984-04-13 EP EP84302564A patent/EP0125056B1/en not_active Expired - Lifetime
- 1984-04-13 IE IE927/84A patent/IE57599B1/en not_active IP Right Cessation
- 1984-04-13 DE DE8484302564T patent/DE3483920D1/de not_active Expired - Fee Related
- 1984-04-17 NO NO841555A patent/NO162235C/no unknown
- 1984-04-18 GR GR74460A patent/GR79905B/el unknown
- 1984-04-18 ES ES531740A patent/ES8602699A1/es not_active Expired
- 1984-04-18 PH PH30584A patent/PH21294A/en unknown
- 1984-04-19 FI FI841590A patent/FI82455C/fi not_active IP Right Cessation
- 1984-04-19 AU AU27092/84A patent/AU565188B2/en not_active Ceased
- 1984-04-19 PT PT78454A patent/PT78454B/pt not_active IP Right Cessation
- 1984-04-19 CA CA000452446A patent/CA1209993A/en not_active Expired
- 1984-04-19 NZ NZ207915A patent/NZ207915A/en unknown
- 1984-04-20 HU HU841550A patent/HU193008B/hu not_active IP Right Cessation
- 1984-04-21 KR KR1019840002110A patent/KR910007965B1/ko not_active IP Right Cessation
- 1984-04-22 IL IL71617A patent/IL71617A/xx unknown
-
1985
- 1985-07-01 ES ES544748A patent/ES8609290A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES531740A0 (es) | 1985-12-01 |
| FI841590A (fi) | 1984-10-23 |
| NO841555L (no) | 1984-10-23 |
| PH21294A (en) | 1987-09-28 |
| HU193008B (en) | 1987-08-28 |
| EP0125056A2 (en) | 1984-11-14 |
| FI841590A0 (fi) | 1984-04-19 |
| FI82455C (fi) | 1991-03-11 |
| EP0125056B1 (en) | 1991-01-16 |
| ES544748A0 (es) | 1986-07-16 |
| HUT34176A (en) | 1985-02-28 |
| PT78454A (en) | 1984-05-01 |
| NZ207915A (en) | 1986-10-08 |
| FI82455B (fi) | 1990-11-30 |
| ES8609290A1 (es) | 1986-07-16 |
| IE57599B1 (en) | 1993-01-27 |
| PT78454B (en) | 1986-08-28 |
| US4564612A (en) | 1986-01-14 |
| GR79905B (es) | 1984-10-31 |
| NO162235B (no) | 1989-08-21 |
| ATE60061T1 (de) | 1991-02-15 |
| IE840927L (en) | 1984-10-22 |
| EP0125056A3 (en) | 1986-04-16 |
| KR910007965B1 (ko) | 1991-10-04 |
| AU565188B2 (en) | 1987-09-10 |
| AU2709284A (en) | 1984-10-25 |
| CA1209993A (en) | 1986-08-19 |
| KR840008346A (ko) | 1984-12-14 |
| NO162235C (no) | 1989-11-29 |
| DE3483920D1 (de) | 1991-02-21 |
| ES8602699A1 (es) | 1985-12-01 |
| IL71617A (en) | 1988-05-31 |
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