IL64009A - Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them - Google Patents

Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them

Info

Publication number
IL64009A
IL64009A IL64009A IL6400981A IL64009A IL 64009 A IL64009 A IL 64009A IL 64009 A IL64009 A IL 64009A IL 6400981 A IL6400981 A IL 6400981A IL 64009 A IL64009 A IL 64009A
Authority
IL
Israel
Prior art keywords
alpha
dioxopenicillanoyloxymethyl
penicillanate
phenylacetamido
tosylate
Prior art date
Application number
IL64009A
Other languages
English (en)
Other versions
IL64009A0 (en
Original Assignee
Rech Applications Therap
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rech Applications Therap filed Critical Rech Applications Therap
Publication of IL64009A0 publication Critical patent/IL64009A0/xx
Publication of IL64009A publication Critical patent/IL64009A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL64009A 1980-10-31 1981-10-06 Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them IL64009A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8035156 1980-10-31

Publications (2)

Publication Number Publication Date
IL64009A0 IL64009A0 (en) 1982-01-31
IL64009A true IL64009A (en) 1984-09-30

Family

ID=10517019

Family Applications (1)

Application Number Title Priority Date Filing Date
IL64009A IL64009A (en) 1980-10-31 1981-10-06 Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them

Country Status (26)

Country Link
US (1) US4831025A (fr)
JP (1) JPS57126493A (fr)
KR (1) KR870001982B1 (fr)
AT (1) AT373893B (fr)
AU (1) AU543870B2 (fr)
BE (1) BE890938A (fr)
CA (1) CA1180696A (fr)
CH (1) CH647527A5 (fr)
DE (1) DE3143219A1 (fr)
DK (1) DK154219C (fr)
ES (1) ES506751A0 (fr)
FI (1) FI813331L (fr)
FR (1) FR2493322B1 (fr)
GB (1) GB2114969B (fr)
GR (1) GR75369B (fr)
IE (1) IE51640B1 (fr)
IL (1) IL64009A (fr)
IT (1) IT1193735B (fr)
LU (1) LU83727A1 (fr)
NL (1) NL8104938A (fr)
NO (1) NO813683L (fr)
NZ (1) NZ198622A (fr)
PH (1) PH17820A (fr)
PT (1) PT73913B (fr)
SE (1) SE452322B (fr)
ZA (1) ZA817091B (fr)

Families Citing this family (43)

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US4432987A (en) * 1982-04-23 1984-02-21 Pfizer Inc. Crystalline benzenesulfonate salts of sultamicillin
PH20068A (en) * 1982-12-06 1986-09-18 Pfizer Process and intermediates for sultamicillin and analogs
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
ES2161602B1 (es) * 1999-04-08 2003-02-16 Asturpharma S A Sintesis de 6-(d-alfa-(bencilidenaminofenilacetamido))penicilanato de 1,1-dioxopenicilanoiloximetilo y analogos. nuevos intermedios para la sintesis de sultamicilina.
US7025989B2 (en) * 2000-02-24 2006-04-11 Advancis Pharmaceutical Corp. Multiple-delayed released antibiotic product, use and formulation thereof
US6544555B2 (en) 2000-02-24 2003-04-08 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
JP2003523372A (ja) * 2000-02-24 2003-08-05 アドバンシス ファーマシューティカル コーポレイション 抗生物質及び抗真菌剤組成物
US6610328B2 (en) 2000-02-24 2003-08-26 Advancis Pharmaceutical Corp. Amoxicillin-clarithromycin antibiotic composition
US6730320B2 (en) 2000-02-24 2004-05-04 Advancis Pharmaceutical Corp. Tetracycline antibiotic product, use and formulation thereof
US6627222B2 (en) 2000-02-24 2003-09-30 Advancis Pharmaceutical Corp. Amoxicillin-dicloxacillin antibiotic composition
US6623758B2 (en) 2000-02-24 2003-09-23 Advancis Pharmaceutical Corp. Cephalosporin-metronidazole antibiotic composition
US6667042B2 (en) 2000-02-24 2003-12-23 Advancis Pharmaceutical Corp. Fluroquinilone antibiotic product, use and formulation thereof
US6663891B2 (en) 2000-02-24 2003-12-16 Advancis Pharmaceutical Corp. Erythromyacin antibiotic product, use and formulation thereof
US6669948B2 (en) 2000-02-24 2003-12-30 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
US6663890B2 (en) 2000-02-24 2003-12-16 Advancis Pharmaceutical Corp. Metronidazole antibiotic product, use and formulation thereof
US6638532B2 (en) 2000-02-24 2003-10-28 Advancis Pharmaceutical Corp. Tetracycline—doxycycline antibiotic composition
US6667057B2 (en) 2000-02-24 2003-12-23 Advancis Pharmaceutical Corp. Levofloxacin antibiotic product, use and formulation thereof
US6991807B2 (en) * 2000-02-24 2006-01-31 Advancis Pharmaceutical, Corp. Antibiotic composition
WO2001062229A1 (fr) * 2000-02-24 2001-08-30 Advanced Pharma, Inc. Produit therapeutique, son application et sa formulation
US6565882B2 (en) 2000-02-24 2003-05-20 Advancis Pharmaceutical Corp Antibiotic composition with inhibitor
US6632453B2 (en) 2000-02-24 2003-10-14 Advancis Pharmaceutical Corp. Ciprofoxacin-metronidazole antibiotic composition
US7105174B2 (en) * 2000-10-13 2006-09-12 Advancis Pharmaceutical Corporation Multiple-delayed release anti-neoplastic product, use and formulation thereof
US7157095B2 (en) * 2000-10-13 2007-01-02 Advancis Pharmaceutical Corporation Multiple-delayed release antifungal product, use and formulation thereof
US7074417B2 (en) * 2000-10-13 2006-07-11 Advancis Pharmaceutical Corporation Multiple-delayed release anti-viral product, use and formulation thereof
US6541014B2 (en) 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
US20020197314A1 (en) 2001-02-23 2002-12-26 Rudnic Edward M. Anti-fungal composition
US20040114368A1 (en) * 2002-12-13 2004-06-17 Shyu Shing Jy Light device having rotatable or movable view
US20040265323A1 (en) * 2003-05-16 2004-12-30 Mccormick Beth A. Compositions comprising pathogen elicited epithelial chemoattractant (eicosanoid hepoxilin A3), inhibitors thereof and methods of use thereof
AU2004258949B2 (en) 2003-07-21 2011-02-10 Shionogi, Inc. Antibiotic product, use and formulation thereof
CA2533292C (fr) 2003-07-21 2013-12-31 Advancis Pharmaceutical Corporation Produit antibiotique, utilisation et formulation correspondantes
EP1648418A4 (fr) 2003-07-21 2011-11-16 Middlebrook Pharmaceuticals Inc Produit antibiotique, utilisation et formulation associees
CA2535177A1 (fr) 2003-08-11 2005-02-24 Advancis Pharmaceutical Corporation Pastille robuste
EP1653924A4 (fr) 2003-08-12 2009-09-09 Middlebrook Pharmaceuticals In Antibiotique, utilisation et formulation associees
CA2535780A1 (fr) 2003-08-29 2005-03-17 Advancis Pharmaceuticals Corporation Produit antibiotique, son utilisation et sa formulation
US8460710B2 (en) 2003-09-15 2013-06-11 Shionogi, Inc. Antibiotic product, use and formulation thereof
CA2572292A1 (fr) 2004-07-02 2006-02-09 Advancis Pharmaceutical Corporation Comprime pour distribution par impulsion
WO2007004239A1 (fr) * 2005-07-06 2007-01-11 Morepen Laboratories Limited Nouvelle forme polymorphique du tosylate de sultamicilline et procede correspondant
US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en) 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
US8299052B2 (en) * 2006-05-05 2012-10-30 Shionogi Inc. Pharmaceutical compositions and methods for improved bacterial eradication
EP2874623B1 (fr) 2012-07-17 2018-12-12 Bayer New Zealand Limited Formulations antibiotiques injectables et leurs procédés d'utilisation
ES2752034T3 (es) 2012-07-17 2020-04-02 Bayer New Zealand Ltd Formaciones inyectables de antibiótico y sus procedimientos de uso
US11116737B1 (en) 2020-04-10 2021-09-14 University Of Georgia Research Foundation, Inc. Methods of using probenecid for treatment of coronavirus infections

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1532222A (fr) * 1963-10-28 1968-07-12 Bristol Myers Co Procédé de préparation de dérivés de la pénicilline
KR830001903B1 (ko) * 1979-02-13 1983-09-19 레오 파마슈티칼 프로덕츠 리미티드 페니실란산유도체의 제조방법
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate

Also Published As

Publication number Publication date
DK154219B (da) 1988-10-24
ZA817091B (en) 1982-10-27
NZ198622A (en) 1985-07-12
US4831025A (en) 1989-05-16
BE890938A (fr) 1982-04-30
DK154219C (da) 1989-03-20
FR2493322B1 (fr) 1986-06-13
IE812361L (en) 1982-04-30
PT73913B (en) 1984-05-29
NO813683L (no) 1982-05-03
IT8168383A0 (it) 1981-10-23
JPH027957B2 (fr) 1990-02-21
IL64009A0 (en) 1982-01-31
IE51640B1 (en) 1987-01-21
SE452322B (sv) 1987-11-23
GB2114969B (en) 1985-02-20
FI813331L (fi) 1982-05-01
DK472181A (da) 1982-05-01
ES8206531A1 (es) 1982-08-16
ES506751A0 (es) 1982-08-16
JPS57126493A (en) 1982-08-06
PT73913A (en) 1981-11-01
ATA447781A (de) 1983-07-15
NL8104938A (nl) 1982-05-17
CA1180696A (fr) 1985-01-08
GB2114969A (en) 1983-09-01
SE8106404L (sv) 1982-05-01
AU543870B2 (en) 1985-05-09
CH647527A5 (de) 1985-01-31
DE3143219C2 (fr) 1990-05-17
GR75369B (fr) 1984-07-13
FR2493322A1 (fr) 1982-05-07
LU83727A1 (fr) 1982-05-07
IT1193735B (it) 1988-08-24
KR830007671A (ko) 1983-11-04
KR870001982B1 (ko) 1987-10-24
AU7636581A (en) 1982-05-06
AT373893B (de) 1984-02-27
DE3143219A1 (de) 1982-08-12
PH17820A (en) 1985-01-07

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