IL31990A - Pyridyl 1,2,4-oxadiazole derivatives,process for the preparation thereof and pharmaceutical compositions containing same - Google Patents
Pyridyl 1,2,4-oxadiazole derivatives,process for the preparation thereof and pharmaceutical compositions containing sameInfo
- Publication number
- IL31990A IL31990A IL31990A IL3199069A IL31990A IL 31990 A IL31990 A IL 31990A IL 31990 A IL31990 A IL 31990A IL 3199069 A IL3199069 A IL 3199069A IL 31990 A IL31990 A IL 31990A
- Authority
- IL
- Israel
- Prior art keywords
- pyridyl
- preparation
- pharmaceutical compositions
- compositions containing
- containing same
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HUCI000796 | 1968-04-26 |
Publications (2)
Publication Number | Publication Date |
---|---|
IL31990A0 IL31990A0 (en) | 1969-06-25 |
IL31990A true IL31990A (en) | 1974-05-16 |
Family
ID=10994349
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL31990A IL31990A (en) | 1968-04-26 | 1969-04-08 | Pyridyl 1,2,4-oxadiazole derivatives,process for the preparation thereof and pharmaceutical compositions containing same |
Country Status (15)
Country | Link |
---|---|
US (1) | US3647809A (pt) |
JP (1) | JPS4824394B1 (pt) |
AT (2) | AT292727B (pt) |
BE (1) | BE732131A (pt) |
BR (1) | BR6908381D0 (pt) |
CA (1) | CA954858A (pt) |
CH (2) | CH542232A (pt) |
DE (1) | DE1920037A1 (pt) |
FR (1) | FR2007529B1 (pt) |
GB (1) | GB1271302A (pt) |
IL (1) | IL31990A (pt) |
NL (1) | NL6906401A (pt) |
NO (1) | NO124253B (pt) |
PL (1) | PL79435B1 (pt) |
SE (1) | SE368576B (pt) |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3853893A (en) * | 1973-04-02 | 1974-12-10 | Squibb & Sons Inc | Anthelmintic 5-(pyridyl)-3-(isothiocyanophenyl) oxadiazoles |
HU177086B (en) * | 1975-06-09 | 1981-07-28 | Eszakmagyar Vegyimuevek | Herbicide and fungicide preparation containing substituted 1,2,4-oxadiazolidin-3-one derivatives |
JPS58150576A (ja) * | 1982-03-03 | 1983-09-07 | Sumitomo Chem Co Ltd | 新規な1,2,4−オキサジアゾ−ル誘導体 |
DE3247118A1 (de) * | 1982-12-20 | 1984-06-20 | Cassella Ag, 6000 Frankfurt | Neue substituierte 1,4-dihydropyridine, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
EP1582519A3 (en) * | 1999-08-19 | 2005-12-21 | Nps Pharmaceuticals, Inc. | Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
WO2001012627A1 (en) * | 1999-08-19 | 2001-02-22 | Nps Pharmaceuticals, Inc. | Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
US6660753B2 (en) * | 1999-08-19 | 2003-12-09 | Nps Pharmaceuticals, Inc. | Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
DK1379525T3 (da) * | 2001-02-21 | 2007-12-27 | Astrazeneca Ab | Heteropolycykliske forbindelser og anvendelse deraf som metabotropiske glutamatreceptor-antagonister |
JP2006502134A (ja) * | 2002-08-09 | 2006-01-19 | アストラゼネカ アクチボラグ | 代謝調節型グルタミン酸受容体において活性を有する化合物 |
WO2004091480A2 (en) * | 2003-04-09 | 2004-10-28 | Exelixis, Inc. | Tie-2 modulators and methods of use |
JP2006528980A (ja) * | 2003-05-15 | 2006-12-28 | メルク エンド カムパニー インコーポレーテッド | S1p受容体作働薬としての3−(2−アミノ−1−アザシクロ)−5−アリール−1,2,4−オキサジアゾール類 |
US20060189661A1 (en) * | 2003-11-03 | 2006-08-24 | Wagenen Bradford V | Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
WO2005060961A2 (en) * | 2003-12-18 | 2005-07-07 | Astrazeneca Ab | Treatment of transient lower esophageal sphincter relaxations (tlesrs) and gastro-esophageal reflux disease (gerd) |
JP4958560B2 (ja) * | 2003-12-24 | 2012-06-20 | プロシディオン・リミテッド | Gpcr受容体作動薬としてのヘテロ環誘導体 |
WO2005077368A2 (en) * | 2004-02-03 | 2005-08-25 | Astrazeneca Ab | Treatment of gastro-esophageal reflux disease (gerd) |
AU2006239418A1 (en) * | 2005-04-26 | 2006-11-02 | Neurosearch A/S | Novel oxadiazole derivatives and their medical use |
IL169855A (en) * | 2005-07-25 | 2014-05-28 | Elta Systems Ltd | A system and method for locating a receiver location |
SI1907382T1 (sl) | 2005-07-26 | 2015-10-30 | Bial-Portela & Ca S.A., | Nitrokateholni derivati kot inhibitorji COMT |
EP1845097A1 (en) * | 2006-04-10 | 2007-10-17 | Portela & Ca., S.A. | Oxadiazole derivatives as COMT inhibitors |
CA2661105C (en) * | 2006-09-07 | 2015-01-06 | Actelion Pharmaceuticals Ltd | Pyridin-4-yl derivatives as immunomodulating agents |
RU2454413C2 (ru) * | 2006-09-08 | 2012-06-27 | Актелион Фармасьютиклз Лтд | Производные пиридин-3-ила в качестве иммуномодулирующих агентов |
EP2124947B1 (en) * | 2007-01-31 | 2017-07-19 | BIAL - Portela & Ca., S.A. | Dosage regimen for comt inhibitors |
WO2008114157A1 (en) * | 2007-03-16 | 2008-09-25 | Actelion Pharmaceuticals Ltd | Amino- pyridine derivatives as s1p1 /edg1 receptor agonists |
MY153975A (en) * | 2007-08-17 | 2015-04-30 | Actelion Pharmaceuticals Ltd | Pyridine derivatives as s1p1/edg1 receptor modulators |
US20110014282A1 (en) * | 2008-02-28 | 2011-01-20 | De Vasconcelos Teofilo Cardoso | Pharmaceutical composition for poorly soluble drugs |
ES2389042T3 (es) * | 2008-03-06 | 2012-10-22 | Actelion Pharmaceuticals Ltd. | Compuestos de piridina |
MX2010009644A (es) * | 2008-03-07 | 2010-09-22 | Actelion Pharmaceuticals Ltd | Derivados piridin-2-ilo como agentes inmunomoduladores. |
KR20110002462A (ko) | 2008-03-17 | 2011-01-07 | 바이알 - 포르텔라 앤드 씨에이 에스에이 | 5-[3-(2,5-디클로로-4,6-디메틸-1-옥시-피리딘-3-일)-[1,2,4]옥사디아졸-5-일]-3-나이트로벤젠-1,2-디올의 결정형 |
JP5837417B2 (ja) | 2008-05-14 | 2015-12-24 | ザ スクリプス リサーチ インスティテュート | スフィンゴシンリン酸受容体の新規なモジュレーター |
PL2396321T3 (pl) | 2009-02-10 | 2015-10-30 | Monsanto Technology Llc | Kompozycje i sposoby zwalczania nicieni |
CN102438595B (zh) * | 2009-04-01 | 2016-04-27 | 巴尔-波特拉及康邦亚股份有限公司 | 包括硝基儿茶酚衍生物的药物制剂及其制备方法 |
JP5864409B2 (ja) | 2009-04-01 | 2016-02-17 | ノヴィファーマ ソシエテ アノニム | ニトロカテコール誘導体を含む医薬製剤及びその製造方法 |
CA2767585C (en) | 2009-07-16 | 2017-09-26 | Actelion Pharmaceuticals Ltd | Pyridin-4-yl derivatives |
SG191742A1 (en) | 2011-01-19 | 2013-08-30 | Actelion Pharmaceuticals Ltd | 2-methoxy-pyridin-4-yl derivatives |
US20140045900A1 (en) | 2011-02-11 | 2014-02-13 | Bial-Portela & Ca, S.A. | Administration regime for nitrocatechols |
DK2791134T3 (da) | 2011-12-13 | 2019-12-09 | BIAL PORTELA & Cª S A | Kemisk forbindelse, der er anvendelig som mellemprodukt til fremstilling af en catechol-o-methyltransferasehæmmer |
CA2901006A1 (en) * | 2013-02-15 | 2014-08-21 | Monsanto Technology Llc | 3,5-disubstituted-4,5-dihydro-1,2,4-oxadiazoles for controlling nematode pests |
WO2016083863A1 (en) | 2014-11-28 | 2016-06-02 | Bial - Portela & Ca, S.A. | Medicaments for slowing parkinson's disease |
KR102220848B1 (ko) | 2015-05-20 | 2021-02-26 | 이도르시아 파마슈티컬스 리미티드 | 화합물 (s)-3-{4-[5-(2-시클로펜틸-6-메톡시-피리딘-4-일)-[1,2,4]옥사디아졸-3-일]-2-에틸-6-메틸-페녹시}-프로판-1,2-디올의 결정형 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL256329A (pt) * | 1959-09-29 | |||
US3227725A (en) * | 1962-04-17 | 1966-01-04 | Union Carbide Corp | Certain 3,5-disubstituted 1,2,4-oxadiazole compounds |
-
1969
- 1969-04-08 IL IL31990A patent/IL31990A/xx unknown
- 1969-04-08 US US815520A patent/US3647809A/en not_active Expired - Lifetime
- 1969-04-14 GB GB09047/69A patent/GB1271302A/en not_active Expired
- 1969-04-18 AT AT375469A patent/AT292727B/de not_active IP Right Cessation
- 1969-04-18 AT AT815670A patent/AT292728B/de not_active IP Right Cessation
- 1969-04-19 DE DE19691920037 patent/DE1920037A1/de active Pending
- 1969-04-24 CH CH1476972A patent/CH542232A/de not_active IP Right Cessation
- 1969-04-24 CH CH627569A patent/CH540925A/de not_active IP Right Cessation
- 1969-04-24 FR FR696912994A patent/FR2007529B1/fr not_active Expired
- 1969-04-25 NL NL6906401A patent/NL6906401A/xx unknown
- 1969-04-25 BR BR208381/69A patent/BR6908381D0/pt unknown
- 1969-04-25 SE SE05909/69A patent/SE368576B/xx unknown
- 1969-04-25 JP JP44032259A patent/JPS4824394B1/ja active Pending
- 1969-04-25 NO NO1733/69A patent/NO124253B/no unknown
- 1969-04-25 CA CA049,755A patent/CA954858A/en not_active Expired
- 1969-04-25 PL PL1969133199A patent/PL79435B1/pl unknown
- 1969-04-25 BE BE732131D patent/BE732131A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
JPS4824394B1 (pt) | 1973-07-20 |
FR2007529A1 (pt) | 1970-01-09 |
US3647809A (en) | 1972-03-07 |
PL79435B1 (en) | 1975-06-30 |
CH540925A (de) | 1973-08-31 |
CH542232A (de) | 1973-11-15 |
GB1271302A (en) | 1972-04-19 |
BE732131A (pt) | 1969-10-01 |
BR6908381D0 (pt) | 1973-02-08 |
CA954858A (en) | 1974-09-17 |
NO124253B (pt) | 1972-03-27 |
IL31990A0 (en) | 1969-06-25 |
FR2007529B1 (pt) | 1973-03-16 |
NL6906401A (pt) | 1969-10-28 |
SE368576B (pt) | 1974-07-08 |
AT292728B (de) | 1971-09-10 |
DE1920037A1 (de) | 1970-11-12 |
AT292727B (de) | 1971-09-10 |
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