IL234487A0 - Estrogen receptor modulators and their uses - Google Patents
Estrogen receptor modulators and their usesInfo
- Publication number
- IL234487A0 IL234487A0 IL234487A IL23448714A IL234487A0 IL 234487 A0 IL234487 A0 IL 234487A0 IL 234487 A IL234487 A IL 234487A IL 23448714 A IL23448714 A IL 23448714A IL 234487 A0 IL234487 A0 IL 234487A0
- Authority
- IL
- Israel
- Prior art keywords
- estrogen receptor
- receptor modulators
- modulators
- estrogen
- receptor
- Prior art date
Links
- 239000002834 estrogen receptor modulator Substances 0.000 title 1
Classifications
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Psychiatry (AREA)
- Immunology (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Obesity (AREA)
- Gastroenterology & Hepatology (AREA)
- Vascular Medicine (AREA)
- Otolaryngology (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261613442P | 2012-03-20 | 2012-03-20 | |
| PCT/US2013/031507 WO2013142266A1 (en) | 2012-03-20 | 2013-03-14 | Estrogen receptor modulators and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL234487A0 true IL234487A0 (en) | 2014-11-02 |
Family
ID=49223229
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL234487A IL234487A0 (en) | 2012-03-20 | 2014-09-07 | Estrogen receptor modulators and their uses |
Country Status (17)
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6154887B2 (ja) | 2012-03-20 | 2017-06-28 | セラゴン ファーマシューティカルズ,インク. | エストロゲン受容体モジュレーターおよびその使用 |
| KR20150129723A (ko) | 2013-03-14 | 2015-11-20 | 세라곤 파마슈티컬스, 인크. | 다환형 에스트로겐 수용체 조절제 및 이의 용도 |
| KR102090231B1 (ko) | 2013-03-15 | 2020-03-17 | 에피젠 바이오싸이언시즈, 아이엔씨. | 질환의 치료에 유용한 헤테로환식 화합물 |
| CN105451735B (zh) | 2013-06-19 | 2019-01-11 | 西拉根制药公司 | 氮杂环丁烷雌激素受体调节剂和其用途 |
| EA031077B1 (ru) | 2013-06-19 | 2018-11-30 | Серагон Фармасьютикалз, Инк. | Модулятор рецептора эстрогена и его применения |
| CA2932106A1 (en) | 2013-12-06 | 2015-06-11 | F. Hoffmann-La Roche Ag | Estrogen receptor modulator for the treatment of locally advanced or metastatic estrogen receptor positive breast cancer |
| WO2015136016A2 (en) | 2014-03-13 | 2015-09-17 | F. Hoffmann-La Roche Ag | Therapeutic combinations with estrogen receptor modulators |
| AU2015228860A1 (en) * | 2014-03-13 | 2016-09-08 | F. Hoffmann-La Roche Ag | Methods and compositions for modulating estrogen receptor mutants |
| MX2017001869A (es) | 2014-08-11 | 2017-05-17 | Hoffmann La Roche | Formas cristalinas de un modulador de receptor de estrogeno. |
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- 2013-03-14 WO PCT/US2013/031507 patent/WO2013142266A1/en not_active Ceased
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| EP2828243A4 (en) | 2015-10-28 |
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| CO7170179A2 (es) | 2015-01-28 |
| PE20142461A1 (es) | 2015-02-05 |
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| SG11201405918XA (en) | 2014-10-30 |
| HK1202535A1 (en) | 2015-10-02 |
| CA2866891A1 (en) | 2013-09-26 |
| KR20140138296A (ko) | 2014-12-03 |
| PH12014502095A1 (en) | 2014-11-24 |
| AU2013235499A1 (en) | 2014-09-25 |
| JP2015514072A (ja) | 2015-05-18 |
| CN104220426B (zh) | 2017-03-01 |
| NZ630124A (en) | 2016-01-29 |
| US20150105403A1 (en) | 2015-04-16 |
| WO2013142266A1 (en) | 2013-09-26 |
| EP2828243B1 (en) | 2018-10-17 |
| MX2014011217A (es) | 2015-03-10 |
| US9499538B2 (en) | 2016-11-22 |
| JP6154887B2 (ja) | 2017-06-28 |
| CR20140479A (es) | 2014-12-01 |
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