IL205776A0 - Morpholino compounds and methods of producing morpholino oligomers - Google Patents

Morpholino compounds and methods of producing morpholino oligomers

Info

Publication number
IL205776A0
IL205776A0 IL205776A IL20577610A IL205776A0 IL 205776 A0 IL205776 A0 IL 205776A0 IL 205776 A IL205776 A IL 205776A IL 20577610 A IL20577610 A IL 20577610A IL 205776 A0 IL205776 A0 IL 205776A0
Authority
IL
Israel
Prior art keywords
morpholino
methods
producing
compounds
oligomers
Prior art date
Application number
IL205776A
Other languages
English (en)
Original Assignee
Avi Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Avi Biopharma Inc filed Critical Avi Biopharma Inc
Publication of IL205776A0 publication Critical patent/IL205776A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL205776A 2007-11-15 2010-05-13 Morpholino compounds and methods of producing morpholino oligomers IL205776A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US98820007P 2007-11-15 2007-11-15
US98819207P 2007-11-15 2007-11-15
PCT/US2008/012804 WO2009064471A1 (en) 2007-11-15 2008-11-14 Method of synthesis of morpholino oligomers

Publications (1)

Publication Number Publication Date
IL205776A0 true IL205776A0 (en) 2010-11-30

Family

ID=40293764

Family Applications (1)

Application Number Title Priority Date Filing Date
IL205776A IL205776A0 (en) 2007-11-15 2010-05-13 Morpholino compounds and methods of producing morpholino oligomers

Country Status (13)

Country Link
EP (1) EP2207779B1 (enExample)
JP (3) JP5512533B2 (enExample)
KR (1) KR101617472B1 (enExample)
CN (1) CN101861318A (enExample)
BR (1) BR122019021332A8 (enExample)
CA (2) CA2704261C (enExample)
DK (1) DK2207779T3 (enExample)
ES (1) ES2479393T3 (enExample)
HR (1) HRP20140646T1 (enExample)
IL (1) IL205776A0 (enExample)
MX (1) MX2010004955A (enExample)
RU (1) RU2606627C2 (enExample)
WO (1) WO2009064471A1 (enExample)

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KR102182663B1 (ko) 2010-05-28 2020-11-25 사렙타 쎄러퓨틱스, 인코퍼레이티드 변형된 서브유니트간 결합 및/또는 말단 그룹을 갖는 올리고뉴클레오타이드 유사체
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Also Published As

Publication number Publication date
CA2884340A1 (en) 2009-05-22
BRPI0819828A8 (pt) 2022-12-27
JP2011503184A (ja) 2011-01-27
RU2010123958A (ru) 2011-12-20
AU2008321409B2 (en) 2014-08-14
CN101861318A (zh) 2010-10-13
BR122019021332A8 (pt) 2022-12-06
CA2884340C (en) 2017-07-25
JP5512533B2 (ja) 2014-06-04
JP2014159432A (ja) 2014-09-04
MX2010004955A (es) 2010-06-30
KR101617472B1 (ko) 2016-05-02
CA2704261C (en) 2015-05-26
CA2704261A1 (en) 2009-05-22
BRPI0819828A2 (pt) 2015-05-26
AU2008321409A1 (en) 2009-05-22
HRP20140646T1 (hr) 2014-09-26
HK1144424A1 (en) 2011-02-18
BR122019021332A2 (enExample) 2015-05-26
JP2016196494A (ja) 2016-11-24
RU2606627C2 (ru) 2017-01-10
KR20100090681A (ko) 2010-08-16
JP6178744B2 (ja) 2017-08-09
EP2207779B1 (en) 2014-04-09
EP2207779A1 (en) 2010-07-21
WO2009064471A1 (en) 2009-05-22
DK2207779T3 (da) 2014-07-14
ES2479393T3 (es) 2014-07-24

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