IL199557A - Use of 10 [(r 3) -1-azabicyclo [2.2.2] oct-3-ilmethyl] - h 10 - phenazazine for the preparation of a drug with selective inhibition of muscarinic receptors 1m, 2m and 3m - Google Patents
Use of 10 [(r 3) -1-azabicyclo [2.2.2] oct-3-ilmethyl] - h 10 - phenazazine for the preparation of a drug with selective inhibition of muscarinic receptors 1m, 2m and 3mInfo
- Publication number
- IL199557A IL199557A IL199557A IL19955709A IL199557A IL 199557 A IL199557 A IL 199557A IL 199557 A IL199557 A IL 199557A IL 19955709 A IL19955709 A IL 19955709A IL 199557 A IL199557 A IL 199557A
- Authority
- IL
- Israel
- Prior art keywords
- ylmethyl
- oct
- azabicyclo
- phenothiazine
- incontinence
- Prior art date
Links
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Urology & Nephrology (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Otolaryngology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0656002A FR2910814B1 (fr) | 2006-12-28 | 2006-12-28 | Utilisation du 10-°(r3)-1-azabicyclo°2.2.2!oct-3-ylmethyl!-10h- phenothiazine pour la preparation d'un medicament exercant une inhibition selective des recepteurs muscariniques m1,2,3 |
| PCT/EP2007/064553 WO2008080924A1 (fr) | 2006-12-28 | 2007-12-26 | Utilisation du 10-[(3r)-1-azabicyclo[2.2.2]oct-3-ylméthyl]-10h-phénothiazine pour la préparation d'un médicament exerçant une inhibition sélective des récepteurs muscariniques m1, m2 et m3 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL199557A true IL199557A (en) | 2014-09-30 |
Family
ID=37951872
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL199557A IL199557A (en) | 2006-12-28 | 2009-06-25 | Use of 10 [(r 3) -1-azabicyclo [2.2.2] oct-3-ilmethyl] - h 10 - phenazazine for the preparation of a drug with selective inhibition of muscarinic receptors 1m, 2m and 3m |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US8143245B2 (enExample) |
| EP (1) | EP2124956A1 (enExample) |
| JP (1) | JP5564263B2 (enExample) |
| KR (1) | KR101465277B1 (enExample) |
| CN (1) | CN101573120B (enExample) |
| AR (1) | AR064714A1 (enExample) |
| AU (1) | AU2007341274B2 (enExample) |
| BR (1) | BRPI0720591A2 (enExample) |
| CA (1) | CA2674162A1 (enExample) |
| FR (2) | FR2910814B1 (enExample) |
| IL (1) | IL199557A (enExample) |
| MA (1) | MA31026B1 (enExample) |
| MX (1) | MX2009006950A (enExample) |
| NO (1) | NO20092654L (enExample) |
| NZ (1) | NZ577915A (enExample) |
| RU (1) | RU2449794C2 (enExample) |
| TN (1) | TN2009000257A1 (enExample) |
| TW (1) | TWI423806B (enExample) |
| UA (1) | UA98131C2 (enExample) |
| WO (1) | WO2008080924A1 (enExample) |
| ZA (1) | ZA200904304B (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2015133989A (ja) * | 2015-04-28 | 2015-07-27 | 重泉 達志 | 健康食品 |
| KR101969263B1 (ko) | 2018-07-16 | 2019-04-15 | 이상호 | 산소 챔버용 산소 공급 장치 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1173445B (it) * | 1984-03-16 | 1987-06-24 | Guidotti & C Spa Labor | Agenti ad attivita' antibroncospastica e composizioni farmaceutiche che li contengono |
| IT1251161B (it) * | 1991-08-07 | 1995-05-04 | Derivati ammonio quaternari di (-) e (+)-3-(10 h-fenotiazin-10-ilmetil)-l-azabiciclo (2.2.2.)ottano e composizioni farmaceutiche che li contengono | |
| AU6686700A (en) | 1999-08-23 | 2001-03-19 | H. Lundbeck A/S | Treatment of urinary incontinence |
| AU2002366800B2 (en) * | 2001-12-20 | 2006-08-03 | Femmepharma Holding Company, Inc. | Vaginal delivery of drugs |
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2006
- 2006-12-28 FR FR0656002A patent/FR2910814B1/fr not_active Expired - Fee Related
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2007
- 2007-12-13 TW TW096147644A patent/TWI423806B/zh not_active IP Right Cessation
- 2007-12-26 NZ NZ577915A patent/NZ577915A/en not_active IP Right Cessation
- 2007-12-26 US US12/521,067 patent/US8143245B2/en not_active Expired - Fee Related
- 2007-12-26 RU RU2009128326/15A patent/RU2449794C2/ru not_active IP Right Cessation
- 2007-12-26 JP JP2009543465A patent/JP5564263B2/ja not_active Expired - Fee Related
- 2007-12-26 KR KR1020097013047A patent/KR101465277B1/ko not_active Expired - Fee Related
- 2007-12-26 WO PCT/EP2007/064553 patent/WO2008080924A1/fr not_active Ceased
- 2007-12-26 BR BRPI0720591-0A patent/BRPI0720591A2/pt not_active IP Right Cessation
- 2007-12-26 MX MX2009006950A patent/MX2009006950A/es active IP Right Grant
- 2007-12-26 AU AU2007341274A patent/AU2007341274B2/en not_active Ceased
- 2007-12-26 CN CN2007800467680A patent/CN101573120B/zh not_active Expired - Fee Related
- 2007-12-26 EP EP07858150A patent/EP2124956A1/fr not_active Withdrawn
- 2007-12-26 CA CA002674162A patent/CA2674162A1/fr not_active Abandoned
- 2007-12-26 UA UAA200907928A patent/UA98131C2/ru unknown
- 2007-12-28 AR ARP070105989A patent/AR064714A1/es unknown
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2009
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- 2009-06-23 TN TNP2009000257A patent/TN2009000257A1/fr unknown
- 2009-06-25 IL IL199557A patent/IL199557A/en not_active IP Right Cessation
- 2009-06-26 MA MA32046A patent/MA31026B1/fr unknown
- 2009-07-13 NO NO20092654A patent/NO20092654L/no not_active Application Discontinuation
-
2011
- 2011-03-17 FR FR1152199A patent/FR2953721A1/fr active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US8143245B2 (en) | 2012-03-27 |
| JP2010514730A (ja) | 2010-05-06 |
| KR101465277B1 (ko) | 2014-11-27 |
| MX2009006950A (es) | 2009-07-14 |
| AR064714A1 (es) | 2009-04-22 |
| AU2007341274A1 (en) | 2008-07-10 |
| RU2009128326A (ru) | 2011-02-10 |
| JP5564263B2 (ja) | 2014-07-30 |
| RU2449794C2 (ru) | 2012-05-10 |
| FR2953721A1 (fr) | 2011-06-17 |
| AU2007341274B2 (en) | 2012-09-20 |
| HK1133207A1 (en) | 2010-03-19 |
| BRPI0720591A2 (pt) | 2014-02-25 |
| NZ577915A (en) | 2011-12-22 |
| CN101573120A (zh) | 2009-11-04 |
| TWI423806B (zh) | 2014-01-21 |
| UA98131C2 (ru) | 2012-04-25 |
| KR20090103887A (ko) | 2009-10-01 |
| TN2009000257A1 (fr) | 2010-10-18 |
| WO2008080924A1 (fr) | 2008-07-10 |
| NO20092654L (no) | 2009-09-28 |
| EP2124956A1 (fr) | 2009-12-02 |
| FR2910814B1 (fr) | 2011-06-17 |
| CN101573120B (zh) | 2011-11-23 |
| TW200833331A (en) | 2008-08-16 |
| FR2910814A1 (fr) | 2008-07-04 |
| ZA200904304B (en) | 2010-06-30 |
| CA2674162A1 (fr) | 2008-07-10 |
| US20100063276A1 (en) | 2010-03-11 |
| MA31026B1 (fr) | 2009-12-01 |
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| FF | Patent granted | ||
| KB | Patent renewed | ||
| MM9K | Patent not in force due to non-payment of renewal fees |