TN2009000257A1 - Utilisation du 10-[(3r)-1-azabicyclo[2.2.2]oct-3-ylmethyl]-10h-phenothiazine pour la preparation d'un medicament exercant une inhibition selective des recepteurs muscariniques m1, m2 et m3. - Google Patents

Utilisation du 10-[(3r)-1-azabicyclo[2.2.2]oct-3-ylmethyl]-10h-phenothiazine pour la preparation d'un medicament exercant une inhibition selective des recepteurs muscariniques m1, m2 et m3.

Info

Publication number
TN2009000257A1
TN2009000257A1 TNP2009000257A TN2009000257A TN2009000257A1 TN 2009000257 A1 TN2009000257 A1 TN 2009000257A1 TN P2009000257 A TNP2009000257 A TN P2009000257A TN 2009000257 A TN2009000257 A TN 2009000257A TN 2009000257 A1 TN2009000257 A1 TN 2009000257A1
Authority
TN
Tunisia
Prior art keywords
azabicyclo
phenothiazine
ylmethyl
medicament
oct
Prior art date
Application number
TNP2009000257A
Other languages
English (en)
Inventor
Thierry Clerc
Jacky Tisne-Versailles
Christophe Przybylski
Original Assignee
Pf Medicament
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pf Medicament filed Critical Pf Medicament
Publication of TN2009000257A1 publication Critical patent/TN2009000257A1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La présente invention concerne l'utilisation du 10-[(3R)-]-azabicyclo[2.2.2.]oct-3-ylméthyl]-10- H phénothiazine ainsi que de ses sels pharmaceutiquement acceptables pour la préparation d'un médicament permettant en particulier de prévenir ou de traiter l'incontinence urinaire et ce par voie locale et/ou par voie orale.
TNP2009000257A 2006-12-28 2009-06-23 Utilisation du 10-[(3r)-1-azabicyclo[2.2.2]oct-3-ylmethyl]-10h-phenothiazine pour la preparation d'un medicament exercant une inhibition selective des recepteurs muscariniques m1, m2 et m3. TN2009000257A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0656002A FR2910814B1 (fr) 2006-12-28 2006-12-28 Utilisation du 10-°(r3)-1-azabicyclo°2.2.2!oct-3-ylmethyl!-10h- phenothiazine pour la preparation d'un medicament exercant une inhibition selective des recepteurs muscariniques m1,2,3
PCT/EP2007/064553 WO2008080924A1 (fr) 2006-12-28 2007-12-26 Utilisation du 10-[(3r)-1-azabicyclo[2.2.2]oct-3-ylméthyl]-10h-phénothiazine pour la préparation d'un médicament exerçant une inhibition sélective des récepteurs muscariniques m1, m2 et m3

Publications (1)

Publication Number Publication Date
TN2009000257A1 true TN2009000257A1 (fr) 2010-10-18

Family

ID=37951872

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2009000257A TN2009000257A1 (fr) 2006-12-28 2009-06-23 Utilisation du 10-[(3r)-1-azabicyclo[2.2.2]oct-3-ylmethyl]-10h-phenothiazine pour la preparation d'un medicament exercant une inhibition selective des recepteurs muscariniques m1, m2 et m3.

Country Status (22)

Country Link
US (1) US8143245B2 (fr)
EP (1) EP2124956A1 (fr)
JP (1) JP5564263B2 (fr)
KR (1) KR101465277B1 (fr)
CN (1) CN101573120B (fr)
AR (1) AR064714A1 (fr)
AU (1) AU2007341274B2 (fr)
BR (1) BRPI0720591A2 (fr)
CA (1) CA2674162A1 (fr)
FR (2) FR2910814B1 (fr)
HK (1) HK1133207A1 (fr)
IL (1) IL199557A (fr)
MA (1) MA31026B1 (fr)
MX (1) MX2009006950A (fr)
NO (1) NO20092654L (fr)
NZ (1) NZ577915A (fr)
RU (1) RU2449794C2 (fr)
TN (1) TN2009000257A1 (fr)
TW (1) TWI423806B (fr)
UA (1) UA98131C2 (fr)
WO (1) WO2008080924A1 (fr)
ZA (1) ZA200904304B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2015133989A (ja) * 2015-04-28 2015-07-27 重泉 達志 健康食品
KR101969263B1 (ko) 2018-07-16 2019-04-15 이상호 산소 챔버용 산소 공급 장치

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1173445B (it) * 1984-03-16 1987-06-24 Guidotti & C Spa Labor Agenti ad attivita' antibroncospastica e composizioni farmaceutiche che li contengono
IT1251161B (it) * 1991-08-07 1995-05-04 Derivati ammonio quaternari di (-) e (+)-3-(10 h-fenotiazin-10-ilmetil)-l-azabiciclo (2.2.2.)ottano e composizioni farmaceutiche che li contengono
AU6686700A (en) * 1999-08-23 2001-03-19 H. Lundbeck A/S Treatment of urinary incontinence
JP2005513080A (ja) * 2001-12-20 2005-05-12 フェムファーマ， インコーポレイテッド 薬物の膣送達

Also Published As

Publication number Publication date
KR101465277B1 (ko) 2014-11-27
US8143245B2 (en) 2012-03-27
RU2009128326A (ru) 2011-02-10
WO2008080924A1 (fr) 2008-07-10
RU2449794C2 (ru) 2012-05-10
MX2009006950A (es) 2009-07-14
NO20092654L (no) 2009-09-28
CN101573120B (zh) 2011-11-23
IL199557A (en) 2014-09-30
JP5564263B2 (ja) 2014-07-30
CA2674162A1 (fr) 2008-07-10
FR2953721A1 (fr) 2011-06-17
AU2007341274A1 (en) 2008-07-10
AR064714A1 (es) 2009-04-22
UA98131C2 (ru) 2012-04-25
BRPI0720591A2 (pt) 2014-02-25
FR2910814B1 (fr) 2011-06-17
KR20090103887A (ko) 2009-10-01
MA31026B1 (fr) 2009-12-01
TW200833331A (en) 2008-08-16
FR2910814A1 (fr) 2008-07-04
US20100063276A1 (en) 2010-03-11
AU2007341274B2 (en) 2012-09-20
NZ577915A (en) 2011-12-22
EP2124956A1 (fr) 2009-12-02
JP2010514730A (ja) 2010-05-06
HK1133207A1 (fr) 2010-03-19
ZA200904304B (en) 2010-06-30
CN101573120A (zh) 2009-11-04
TWI423806B (zh) 2014-01-21

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