IL155400A0 - Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride and processes for preparing thereof - Google Patents

Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride and processes for preparing thereof

Info

Publication number
IL155400A0
IL155400A0 IL15540001A IL15540001A IL155400A0 IL 155400 A0 IL155400 A0 IL 155400A0 IL 15540001 A IL15540001 A IL 15540001A IL 15540001 A IL15540001 A IL 15540001A IL 155400 A0 IL155400 A0 IL 155400A0
Authority
IL
Israel
Prior art keywords
venlafaxine
preparing
processes
crystalline
base
Prior art date
Application number
IL15540001A
Other languages
English (en)
Original Assignee
Teva Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27500045&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL155400(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teva Pharma filed Critical Teva Pharma
Publication of IL155400A0 publication Critical patent/IL155400A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/42—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having amino groups or hydroxy groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/10—Separation; Purification; Stabilisation; Use of additives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/54—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C217/74—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with rings other than six-membered aromatic rings being part of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL15540001A 2000-10-19 2001-10-19 Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride and processes for preparing thereof IL155400A0 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US24157700P 2000-10-19 2000-10-19
US25886100P 2000-12-29 2000-12-29
US27872101P 2001-03-26 2001-03-26
US29246901P 2001-05-21 2001-05-21
PCT/US2001/051017 WO2002045658A2 (fr) 2000-10-19 2001-10-19 Base cristalline de venlafaxine et nouveaux polymorphes de chlorhydrate de venlafaxine, et preparation de ceux-ci

Publications (1)

Publication Number Publication Date
IL155400A0 true IL155400A0 (en) 2003-11-23

Family

ID=27500045

Family Applications (2)

Application Number Title Priority Date Filing Date
IL15540001A IL155400A0 (en) 2000-10-19 2001-10-19 Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride and processes for preparing thereof
IL196287A IL196287A0 (en) 2000-10-19 2008-12-31 Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride and processes for preparing thereof

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL196287A IL196287A0 (en) 2000-10-19 2008-12-31 Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride and processes for preparing thereof

Country Status (20)

Country Link
US (1) US20020143211A1 (fr)
EP (1) EP1334082A4 (fr)
JP (2) JP2004530638A (fr)
KR (1) KR20030059206A (fr)
CN (1) CN1620420A (fr)
AU (1) AU2002241764A1 (fr)
CA (1) CA2426158A1 (fr)
CZ (1) CZ20031298A3 (fr)
DE (1) DE01988460T1 (fr)
ES (1) ES2206082T1 (fr)
HR (1) HRP20030392A2 (fr)
HU (1) HUP0303496A3 (fr)
IL (2) IL155400A0 (fr)
IS (1) IS6789A (fr)
MX (1) MXPA03003459A (fr)
NO (1) NO20031743L (fr)
PL (1) PL365895A1 (fr)
SK (1) SK5762003A3 (fr)
WO (1) WO2002045658A2 (fr)
YU (1) YU30203A (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020183553A1 (en) * 2000-10-19 2002-12-05 Ben-Zion Dolitzky Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride, processes for preparing thereof
EP1330427A1 (fr) * 2000-10-31 2003-07-30 Ciba SC Holding AG Formes cristallines de chlorhydrate de venlafaxine
HUP0104872A3 (en) * 2001-11-13 2004-04-28 Egis Gyogyszergyar Nyilvanosan New polymorphic forms of venlafaxine, process for their preparation, pharmaceutical compositions containing them and their use
UA77234C2 (en) * 2001-12-05 2006-11-15 Wyeth Corp Monohydrate of venlafaxine hydrochloride and methods for its preparation (variants)
KR20050044673A (ko) 2001-12-05 2005-05-12 와이어쓰 벤라팍신 하이드로클로라이드의 신규한 결정 다형체 및이의 제조방법
WO2003050074A1 (fr) * 2001-12-13 2003-06-19 Cadila Healthcare Limited Fabrication de l'hydrochlorure venlafaxine et de polymorphes cristallins de celui-ci
AU2003226748A1 (en) * 2002-03-28 2003-10-13 Synthon B.V. Compositions of venlafaxine base
AR039163A1 (es) 2002-03-28 2005-02-09 Synthon Bv Besilato de venlafaxina
WO2003082805A1 (fr) 2002-03-28 2003-10-09 Synthon B.V. Sels de venlafaxine faiblement solubles dans l'eau
DE10359154A1 (de) 2003-12-16 2005-07-28 Krka Tovarna Zdravil, D.D. Verfahren zur Herstellung von Venlafaxin und Venlafaxinhydrochlorid der Form I
US7468428B2 (en) 2004-03-17 2008-12-23 App Pharmaceuticals, Llc Lyophilized azithromycin formulation
JP4889501B2 (ja) * 2004-10-20 2012-03-07 田辺三菱製薬株式会社 フェニルエタノールアミン化合物の製造方法及びその中間体
KR20080056311A (ko) * 2005-10-19 2008-06-20 테바 파마슈티컬 인더스트리즈 리미티드 고순도1-[2-디메틸아미노-(4-메톡시페닐)에틸)시클로헥산올염산염의 제조 방법
WO2007049302A2 (fr) * 2005-10-28 2007-05-03 Ind-Swift Laboratories Limited Procede ameliore pour la preparation de venlafaxine pure
SI2032521T1 (sl) 2006-06-27 2010-02-26 Sandoz Ag Nov postopek za pripravo soli
EP2081885A2 (fr) * 2006-07-14 2009-07-29 Medichem, S.A. Procedes ameliores servant a preparer de la venlafaxine sous forme de base et des sels de celle-ci
CA2860747C (fr) * 2010-10-01 2015-08-11 Shan Dong Luye Pharmaceutical Co., Ltd. Formes polymorphiques du chlorhydrate de 4-methylbenzoate de 4-[2-dimethylamino-1-(1-hydroxycyclohexyl)ethyl]phenyle, leurs procedes de synthese et leur utilisation
AU2014348523B2 (en) 2013-11-15 2019-01-03 Akebia Therapeutics, Inc. Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino}acetic acid, compositions, and uses thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4535186A (en) * 1983-04-19 1985-08-13 American Home Products Corporation 2-Phenyl-2-(1-hydroxycycloalkyl or 1-hydroxycycloalk-2-enyl)ethylamine derivatives
US4611078A (en) * 1983-10-26 1986-09-09 American Home Products Corporation Substituted phenylacetonitriles
AR255595A1 (fr) 1994-07-13 2002-05-24 Gador Sa
PE57198A1 (es) * 1996-03-25 1998-10-10 American Home Prod Formula de liberacion prolongada
US6197828B1 (en) * 1998-12-01 2001-03-06 Sepracor, Inc. Derivatives of (+)-venlafaxine and methods of preparing and using the same
US20020183553A1 (en) * 2000-10-19 2002-12-05 Ben-Zion Dolitzky Crystalline venlafaxine base and novel polymorphs of venlafaxine hydrochloride, processes for preparing thereof
EP1330427A1 (fr) * 2000-10-31 2003-07-30 Ciba SC Holding AG Formes cristallines de chlorhydrate de venlafaxine
AU2001235970A1 (en) * 2000-12-07 2002-06-18 Dr. Reddy's Research Foundation Novel crystalline polymorphic forms of venlafaxine hydrochloride and a process for their preparation

Also Published As

Publication number Publication date
HUP0303496A2 (hu) 2004-01-28
AU2002241764A1 (en) 2002-06-18
NO20031743L (no) 2003-06-18
KR20030059206A (ko) 2003-07-07
WO2002045658A2 (fr) 2002-06-13
ES2206082T1 (es) 2004-05-16
DE01988460T1 (de) 2004-04-22
IL196287A0 (en) 2011-08-01
JP2004530638A (ja) 2004-10-07
EP1334082A4 (fr) 2006-02-01
NO20031743D0 (no) 2003-04-15
SK5762003A3 (en) 2003-11-04
HRP20030392A2 (en) 2005-04-30
WO2002045658A3 (fr) 2003-01-16
CA2426158A1 (fr) 2002-06-13
MXPA03003459A (es) 2005-04-29
IS6789A (is) 2003-04-15
YU30203A (sh) 2006-08-17
HUP0303496A3 (en) 2005-08-29
CZ20031298A3 (cs) 2003-10-15
US20020143211A1 (en) 2002-10-03
JP2008239629A (ja) 2008-10-09
CN1620420A (zh) 2005-05-25
PL365895A1 (en) 2005-01-10
EP1334082A2 (fr) 2003-08-13

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