IL152417A0 - Azabicyclic carbamates and their use as alpha-7 nicotinic acetylcholine receptor agonists - Google Patents

Azabicyclic carbamates and their use as alpha-7 nicotinic acetylcholine receptor agonists

Info

Publication number
IL152417A0
IL152417A0 IL15241701A IL15241701A IL152417A0 IL 152417 A0 IL152417 A0 IL 152417A0 IL 15241701 A IL15241701 A IL 15241701A IL 15241701 A IL15241701 A IL 15241701A IL 152417 A0 IL152417 A0 IL 152417A0
Authority
IL
Israel
Prior art keywords
alpha
receptor agonists
acetylcholine receptor
nicotinic acetylcholine
azabicyclic
Prior art date
Application number
IL15241701A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of IL152417A0 publication Critical patent/IL152417A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL15241701A 2000-05-05 2001-05-03 Azabicyclic carbamates and their use as alpha-7 nicotinic acetylcholine receptor agonists IL152417A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0010955.3A GB0010955D0 (en) 2000-05-05 2000-05-05 Organic compounds
PCT/EP2001/005008 WO2001085727A1 (en) 2000-05-05 2001-05-03 Azabicyclic carbamates and their use as alpha-7 nicotinic acetylcholine receptor agonists

Publications (1)

Publication Number Publication Date
IL152417A0 true IL152417A0 (en) 2003-05-29

Family

ID=9891092

Family Applications (1)

Application Number Title Priority Date Filing Date
IL15241701A IL152417A0 (en) 2000-05-05 2001-05-03 Azabicyclic carbamates and their use as alpha-7 nicotinic acetylcholine receptor agonists

Country Status (29)

Country Link
US (1) US6780861B2 (enExample)
EP (1) EP1282620B1 (enExample)
JP (1) JP4898062B2 (enExample)
KR (1) KR20020093974A (enExample)
CN (1) CN1167703C (enExample)
AR (1) AR028073A1 (enExample)
AT (1) ATE263167T1 (enExample)
AU (2) AU6225701A (enExample)
BR (1) BR0110521A (enExample)
CA (1) CA2407972C (enExample)
CZ (1) CZ20023622A3 (enExample)
DE (1) DE60102581T2 (enExample)
DK (1) DK1282620T3 (enExample)
ES (1) ES2218418T3 (enExample)
GB (1) GB0010955D0 (enExample)
HK (1) HK1054223B (enExample)
HU (1) HUP0301866A2 (enExample)
IL (1) IL152417A0 (enExample)
MX (1) MXPA02010892A (enExample)
NO (1) NO20025280L (enExample)
NZ (1) NZ522226A (enExample)
PE (1) PE20020221A1 (enExample)
PL (1) PL357435A1 (enExample)
PT (1) PT1282620E (enExample)
RU (1) RU2002131886A (enExample)
SK (1) SK15612002A3 (enExample)
TR (1) TR200401007T4 (enExample)
WO (1) WO2001085727A1 (enExample)
ZA (1) ZA200208969B (enExample)

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Also Published As

Publication number Publication date
JP2003532731A (ja) 2003-11-05
MXPA02010892A (es) 2003-03-27
PL357435A1 (en) 2004-07-26
CN1427840A (zh) 2003-07-02
DK1282620T3 (da) 2004-07-19
CN1167703C (zh) 2004-09-22
ES2218418T3 (es) 2004-11-16
DE60102581T2 (de) 2005-02-03
EP1282620A1 (en) 2003-02-12
US20030166654A1 (en) 2003-09-04
JP4898062B2 (ja) 2012-03-14
RU2002131886A (ru) 2004-04-10
HK1054223B (en) 2005-03-04
NO20025280D0 (no) 2002-11-04
AR028073A1 (es) 2003-04-23
CZ20023622A3 (cs) 2003-02-12
ATE263167T1 (de) 2004-04-15
DE60102581D1 (de) 2004-05-06
PT1282620E (pt) 2004-07-30
PE20020221A1 (es) 2002-04-23
NO20025280L (no) 2002-11-04
US6780861B2 (en) 2004-08-24
SK15612002A3 (sk) 2003-04-01
KR20020093974A (ko) 2002-12-16
AU6225701A (en) 2001-11-20
ZA200208969B (en) 2003-10-07
WO2001085727A1 (en) 2001-11-15
EP1282620B1 (en) 2004-03-31
CA2407972A1 (en) 2001-11-15
TR200401007T4 (tr) 2004-07-21
GB0010955D0 (en) 2000-06-28
AU2001262257B2 (en) 2004-11-04
NZ522226A (en) 2004-08-27
CA2407972C (en) 2010-03-09
HK1054223A1 (en) 2003-11-21
HUP0301866A2 (hu) 2003-09-29
BR0110521A (pt) 2003-04-08

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