IL142837A0 - Semi-hydrochloride of 8-cyan-1-cycloproyl-7-(1s,6s-2,8-diazabicyclo [4.3.0] nonan-8-yl)-6-fluoro-1,4-dihydro-4-oxo-3-quinoline carboxylic acid - Google Patents

Semi-hydrochloride of 8-cyan-1-cycloproyl-7-(1s,6s-2,8-diazabicyclo [4.3.0] nonan-8-yl)-6-fluoro-1,4-dihydro-4-oxo-3-quinoline carboxylic acid

Info

Publication number
IL142837A0
IL142837A0 IL14283799A IL14283799A IL142837A0 IL 142837 A0 IL142837 A0 IL 142837A0 IL 14283799 A IL14283799 A IL 14283799A IL 14283799 A IL14283799 A IL 14283799A IL 142837 A0 IL142837 A0 IL 142837A0
Authority
IL
Israel
Prior art keywords
cycloproyl
nonan
diazabicyclo
cyan
dihydro
Prior art date
Application number
IL14283799A
Other languages
English (en)
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of IL142837A0 publication Critical patent/IL142837A0/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL14283799A 1998-11-25 1999-11-15 Semi-hydrochloride of 8-cyan-1-cycloproyl-7-(1s,6s-2,8-diazabicyclo [4.3.0] nonan-8-yl)-6-fluoro-1,4-dihydro-4-oxo-3-quinoline carboxylic acid IL142837A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19854357A DE19854357A1 (de) 1998-11-25 1998-11-25 Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
PCT/EP1999/008778 WO2000031077A1 (de) 1998-11-25 1999-11-15 Semi-hydrochlorid von 8-cyan-1- cyclopropyl -7-(1s,6s-2, 8-diazabicyclo [4.3.0]nonan -8-yl)-6- fluor-1, 4-dihydro-4- oxo-3- chinolincarbonsäure

Publications (1)

Publication Number Publication Date
IL142837A0 true IL142837A0 (en) 2002-03-10

Family

ID=7888961

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14283799A IL142837A0 (en) 1998-11-25 1999-11-15 Semi-hydrochloride of 8-cyan-1-cycloproyl-7-(1s,6s-2,8-diazabicyclo [4.3.0] nonan-8-yl)-6-fluoro-1,4-dihydro-4-oxo-3-quinoline carboxylic acid
IL142837A IL142837A (en) 1998-11-25 2001-04-27 Partial Hydrochloride of 8 Acid 8 - Cyano - 1 - Cyclopropyl - 7 - (S1, S6 - 2, 8 - Diazabicyclo [0.3.4] Nonan - 8 - Il) - 6 - Fluoro - 1, 4 - Dihydro - 4 - Oxo Quinolinkerboxylic acid and pharmaceutical preparations containing it

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL142837A IL142837A (en) 1998-11-25 2001-04-27 Partial Hydrochloride of 8 Acid 8 - Cyano - 1 - Cyclopropyl - 7 - (S1, S6 - 2, 8 - Diazabicyclo [0.3.4] Nonan - 8 - Il) - 6 - Fluoro - 1, 4 - Dihydro - 4 - Oxo Quinolinkerboxylic acid and pharmaceutical preparations containing it

Country Status (28)

Country Link
US (1) US6995170B1 (cs)
EP (1) EP1133495B1 (cs)
JP (1) JP2002530408A (cs)
KR (1) KR100740956B1 (cs)
CN (1) CN1176921C (cs)
AR (1) AR023709A1 (cs)
AT (1) ATE225790T1 (cs)
AU (1) AU759769B2 (cs)
BR (1) BR9915684A (cs)
CA (1) CA2351714C (cs)
CZ (1) CZ300058B6 (cs)
DE (2) DE19854357A1 (cs)
DK (1) DK1133495T3 (cs)
ES (1) ES2181488T3 (cs)
HK (1) HK1042704B (cs)
HU (1) HUP0104367A3 (cs)
IL (2) IL142837A0 (cs)
NO (1) NO318053B1 (cs)
NZ (1) NZ511863A (cs)
PL (1) PL196508B1 (cs)
PT (1) PT1133495E (cs)
RU (1) RU2242475C2 (cs)
SK (1) SK285561B6 (cs)
TR (1) TR200101443T2 (cs)
TW (1) TWI234565B (cs)
UA (1) UA67875C2 (cs)
WO (1) WO2000031077A1 (cs)
ZA (1) ZA013317B (cs)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19854357A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE10224086A1 (de) * 2002-05-31 2003-12-11 Bayer Ag Pharmazeutische Zubereitungen zur oralen Anwendung enthaltend wirkstoffbeladene Ionentauscherharze sowie strukturviskose Gelbildner als Verdicker
DE102004015981A1 (de) * 2004-04-01 2005-10-20 Bayer Healthcare Ag Neue kirstalline Form von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE102006049520A1 (de) * 2006-10-20 2008-04-24 Bayer Healthcare Ag Verfahren zur Herstellung von Pradofloxacin
BR112019016543A2 (pt) 2017-02-13 2020-03-31 Bayer Animal Health Gmbh Composição líquida que contém pradofloxacina
CN116813614A (zh) * 2023-05-31 2023-09-29 天津大学 一种盐酸普拉沙星二水合物晶体及其制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3906365A1 (de) * 1988-07-15 1990-01-18 Bayer Ag 7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
DE4120646A1 (de) * 1991-06-22 1992-12-24 Bayer Ag 7-isoindolinyl-chinolon- und naphthyridoncarbonsaeure-derivate
DE19546249A1 (de) * 1995-12-12 1997-06-19 Bayer Ag Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen
IL125444A (en) * 1996-02-23 2001-03-19 Bayer Ag Optionally substituted 8-cyano-1-cyclopropyl-7- (2,8-diazabicyclo ¬4.3.0¾ nonan-8-yl)-6- floro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids and their derivatives their preparation and medicaments containing them
DE19633805A1 (de) * 1996-02-23 1997-08-28 Bayer Ag Gegenenenfalls substituierte 8-Cyan-l-cyclopropyl-7-(2,8-diazabicyclo-[4.3.0]-nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäuren und ihre Derivate
DE19854357A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure

Also Published As

Publication number Publication date
CZ20011753A3 (cs) 2001-09-12
NO20012532L (no) 2001-07-02
SK285561B6 (sk) 2007-03-01
CN1328557A (zh) 2001-12-26
HUP0104367A2 (hu) 2002-02-28
NO20012532D0 (no) 2001-05-23
TWI234565B (en) 2005-06-21
HUP0104367A3 (en) 2002-12-28
DE19854357A1 (de) 2000-05-31
NZ511863A (en) 2003-05-30
EP1133495A1 (de) 2001-09-19
EP1133495B1 (de) 2002-10-09
CZ300058B6 (cs) 2009-01-21
US6995170B1 (en) 2006-02-07
CA2351714C (en) 2010-06-15
AU759769B2 (en) 2003-05-01
UA67875C2 (uk) 2004-07-15
CA2351714A1 (en) 2000-06-02
AU1271600A (en) 2000-06-13
HK1042704B (zh) 2005-09-09
HK1042704A1 (en) 2002-08-23
ZA013317B (en) 2002-06-26
ES2181488T3 (es) 2003-02-16
KR100740956B1 (ko) 2007-07-19
JP2002530408A (ja) 2002-09-17
CN1176921C (zh) 2004-11-24
PL347799A1 (en) 2002-04-22
WO2000031077A1 (de) 2000-06-02
IL142837A (en) 2006-08-01
PT1133495E (pt) 2003-02-28
RU2242475C2 (ru) 2004-12-20
DK1133495T3 (da) 2003-02-10
TR200101443T2 (tr) 2001-09-21
DE59903063D1 (de) 2002-11-14
SK6842001A3 (en) 2001-12-03
PL196508B1 (pl) 2008-01-31
AR023709A1 (es) 2002-09-04
ATE225790T1 (de) 2002-10-15
BR9915684A (pt) 2001-08-14
NO318053B1 (no) 2005-01-24
KR20010075694A (ko) 2001-08-09

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